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PGC-1α

PGC-1α是一种在人类中由PPARGC1A基因编码的蛋白质。PGC-1α是线粒体生物合成的主要调节因子。PGC-1α也是肝脏糖异生的主要调节因子,诱导糖异生基因表达增加。

SR-18292
T43532095432-55-4
SR-18292 是一种 PPARγ 共激活因子-1α (PGC-1α) 抑制剂,可增加 PGC-1α 乙酰化,抑制糖异生基因表达并减少肝细胞中的葡萄糖生成。
  • ¥ 235
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TargetMol | Inhibitor Sale
ZLN005
T180249671-76-3
ZLN005 是一种有效的组织特异性 PGC-1α 转录激活剂。
  • ¥ 128
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TargetMol | Inhibitor Sale
11-Oxoisomogroside V
T799652149606-15-3
11-Oxoisomogroside V(compound 3)是从罗汉果粗提物中分离的一种葫芦苷,能够激活PGC-1α的转录活性。荧光素酶实验表明,10 μM 和 20 μM 浓度的11-Oxoisomogroside V分别将荧光素酶活性提高至 133.79% 和 143.81%。
  • 待询
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Neuroprotective agent 8
T206923
Neuroprotective agent 8 (compound AA-9) 是一种口服活性神经保护剂,通过抗氧化应激和抗炎机制发挥作用。在大鼠 MCAO 缺血性卒中模型中,该化合物可以激活 PGC-1α 并抑制 NLRP3 炎症小体。
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