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已知活性化合物库

已知活性化合物库

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产品编号 L4010 Bioactive Compounds Library Max
  库化合物信息   Excel SDF

已知活性库是 22555 个具有生物活性,能引起细胞、组织甚至个体生物学反应的化合物的集合。包括了正在进行临床前研究的药物分子,临床期的药物分子和已经上市的药物。靶点明确,信息全面,非常适合完成药物功能重定位、小分子诱导细胞分化以及机制研究中蛋白靶点确认等科研工作。

由于活性明确,靶点已知,很多科学家会从已知活性库中选择可以用于细胞诱导分化的小分子;通过单一或几个小分子的联合作用,筛选出能将各种体细胞诱导成为诱导多能干细胞,神经前体细胞,心肌细胞等的分子;甚至还有使用小分子组合在体内完成诱导分化的成功尝试。

已知活性库是对经典已知活性库的补充,添加了 TargetMol 特有,新颖的化合物(Part B),所有化合物靶点明确,且都进行过细胞水平活性测试,比上市药物库结构更为新颖,比类药化合物库更易发现活性化合物。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
咨询化合物库
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产品描述

  • 22555个已知活性化合物的集合,可用于高通量筛选、高内涵筛选、细胞诱导和靶点确认;
  • 所有化合物都有相应的靶点信息的描述,活性研究更有保障和依据;
  • 是老药新用、细胞诱导靶点筛选的有效工具;
  • 涵盖多个疾病研究领域,如癌症、代谢、免疫和心血管系统等;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • 结构多样,药效显著,可渗透细胞;

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L4010)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

Apoptosis (1130)
Antibacterial (875)
Autophagy (811)
Endogenous Metabolite (789)
Antibiotic (526)
5-HT Receptor (351)
AChR (302)
Antifungal (287)
Parasite (282)
COX (269)
Adrenergic Receptor (249)
DNA/RNA Synthesis (241)
NF-κB (239)
Dopamine Receptor (221)
CDK (218)
HIV Protease (211)
PI3K (199)
Potassium Channel (194)
Calcium Channel (192)
EGFR (181)
Reactive Oxygen Species (172)
P450 (168)
Histamine Receptor (166)
PDE (165)
VEGFR (158)
Epigenetic Reader Domain (158)
Dehydrogenase (154)
Sodium Channel (145)
Influenza Virus (143)
Antioxidant (135)
GABA Receptor (133)
GluR (128)
PPAR (127)
Histone Methyltransferase (125)
TRP/TRPV Channel (121)
Microtubule Associated (119)
HDAC (118)
JAK (111)
TNF (110)
mTOR (106)
GPR (103)
Wnt/beta-catenin (103)
Akt (102)
ERK (101)
p38 MAPK (101)
FLT (100)
Prostaglandin Receptor (99)
Topoisomerase (99)
Phosphatase (98)
Estrogen/progestogen Receptor (97)
Src (97)
Ferroptosis (96)
PDGFR (92)
Adenosine Receptor (91)
AChE (91)
SARS-CoV (89)
STAT (88)
iGluR (87)
PKC (86)
Estrogen Receptor/ERR (85)
PARP (84)
HCV Protease (84)
AMPK (83)
GSK-3 (82)
FGFR (82)
IL Receptor (79)
Nucleoside Antimetabolite/Analog (78)
RAAS (78)
Opioid Receptor (78)
Raf (77)
Caspase (77)
NMDAR (76)
Virus Protease (76)
NO Synthase (74)
MMP (73)
c-Kit (73)
BCL (73)
c-Met/HGFR (70)
Ras (68)
MAO (68)
Glucocorticoid Receptor (67)
Androgen Receptor (66)
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Phospholipase (64)
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HSV (61)
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Mitochondrial Metabolism (60)
Anti-infection (60)
TGF-beta/Smad (58)
ROS (58)
Aurora Kinase (57)
ALK (56)
Mitophagy (53)
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JNK (51)
BTK (50)
HIF/HIF Prolyl-Hydroxylase (50)
E1/E2/E3 Enzyme (49)
DUB (49)
MEK (48)
Antifection (47)
Tyrosine Kinases (47)
HER (47)
Casein Kinase (47)
CCR (46)
ROCK (46)
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PKA (46)
Monoamine Oxidase (46)
Nrf2 (46)
NOS (46)
Transferase (45)
Interleukin (45)
Reverse Transcriptase (44)
IκB/IKK (43)
HIF (42)
P-gp (42)
Histone Demethylase (42)
p53 (42)
Gamma-secretase (41)
IGF-1R (41)
Retinoid Receptor (41)
Serine/threonin kinase (41)
Serotonin Transporter (39)
P2X Receptor (39)
DNA-PK (39)
Integrin (38)
CXCR (37)
c-RET (36)
S1P Receptor (36)
Norepinephrine (35)
TAM Receptor (35)
Cysteine Protease (35)
Immunology/Inflammation related (34)
Serine Protease (33)
LPL Receptor (33)
Reductase (33)
S6 Kinase (32)
Hedgehog/Smoothened (32)
CaMK (32)
ribosome (32)
FAK (31)
Histone Acetyltransferase (31)
Trk receptor (31)
RIP kinase (30)
PROTACs (30)
Chloride channel (30)
FAAH (30)
Glucosidase (30)
Proton pump (29)
Progesterone Receptor (29)
PLK (29)
Sigma receptor (29)
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transporter (27)
Fatty Acid Synthase (27)
NADPH (27)
Thrombin (26)
Glucokinase (26)
NOD (26)
CFTR (26)
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Aryl Hydrocarbon Receptor (25)
DPP-4 (25)
Syk (25)
ATM/ATR (25)
Mdm2 (24)
Protease-activated Receptor (24)
Kinesin (24)
Ligand for E3 Ligase (23)
Rho (23)
Amino Acids and Derivatives (23)
Pim (23)
DNA Methyltransferase (23)
ROR (22)
PDK (22)
Endothelin Receptor (22)
PERK (22)
Smo (22)
HMG-CoA Reductase (22)
Indoleamine 2,3-Dioxygenase (IDO) (22)
FXR (21)
Thyroid hormone receptor(THR) (21)
Glutathione Peroxidase (21)
DNA (21)
DNA Alkylator/Crosslinker (21)
P2Y Receptor (21)
Lipase (21)
SGLT (21)
IRAK (20)
AhR (20)
Epoxide Hydrolase (20)
Glucagon Receptor (20)
LTR (19)
LRRK2 (19)
Factor Xa (19)
Complement System (19)
DYRK (19)
Hydroxylase (19)
Guanylate cyclase (19)
Neurokinin receptor (19)
Xanthine Oxidase (19)
MRP (19)
STING (18)
cAMP (18)
PAK (18)
OX Receptor (17)
LPA Receptor (17)
PD-1/PD-L1 (17)
Leukotriene Receptor (16)
NOD-like Receptor (NLR) (16)
DHFR (16)
Neuropeptide Y Receptor (16)
YAP (15)
Antifolate (15)
c-Myc (15)
Lipid (15)
IRE1 (15)
BACE (15)
IAP (15)
Myosin (15)
DNA Alkylation (15)
Liver X Receptor (14)
PI4K (14)
Aromatase (14)
Platelet aggregation (14)
DNA gyrase (14)
PGE Synthase (14)
CSF-1R (14)
GTPase (14)
Ephrin Receptor (14)
ROS Kinase (13)
Vasopressin Receptor (13)
RSV (13)
ABC (13)
cholecystokinin (13)
Aminopeptidase (13)
Beta-Secretase (12)
Telomerase (12)
CETP (12)
NADPH-oxidase (11)
Discoidin Domain Receptor (DDR) (11)
Stearoyl-CoA Desaturase (SCD) (11)
Bradykinin Receptor (11)
Free radical scavengers (11)
Isocitrate Dehydrogenase (IDH) (11)
Monocarboxylate transporter (11)
GPCR19 (11)
Neurotensin Receptor (11)
Melanocortin Receptor (11)
GHSR (11)
Monoamine Transporter (11)
Acetyl-CoA Carboxylase (11)
Phosphorylase (11)
PAI-1 (11)
IDO (10)
PKM (10)
NAMPT (10)
Imidazoline Receptor (10)
Melatonin Receptor (10)
LDL (10)
IFNAR (10)
UGT (9)
MT Receptor (9)
ATP Citrate Lyase (9)
SGK (9)
MLK (9)
CaSR (9)
CAT (9)
BCRP (9)
GRK (9)
Arrestin (8)
Dynamin (8)
Glutaminase (8)
Adenylyl cyclase (8)
Neprilysin (8)
ASK (8)
Ligands for Target Protein for PROTAC (8)
Wee1 (8)
GST (8)
Porcupine (8)
Tie-2 (7)
GlyT (7)
p97 (7)
Na+/Ca2+ Exchanger (7)
PAD (7)
OCT (7)
PTEN (7)
SIK (7)
MNK (7)
Annexin A (7)
Arginase (7)
GPX (6)
Adenosine deaminase (6)
OAT (6)
MyD88 (6)
Aquaporin (6)
RAR/RXR  (6)
Molecular Glues (6)
FLAP (6)
Somatostatin (6)
MELK (6)
Carboxypeptidase (6)
MAGL (6)
CRISPR/Cas9 (6)
APC (6)
Oxytocin Receptor (5)
NPC1L1 (5)
DprE1 (5)
Gap Junction Protein (5)
VDAC (5)
BMI-1 (5)
cell cycle arrest (5)
Hippo pathway (5)
TOPK (5)
Amylase (5)
GNRH Receptor (5)
CRM1 (5)
AAK1 (AP2 associated kinase 1) (5)
Methionine Adenosyltransferase (MAT) (5)
Angiotensin-converting Enzyme (ACE) (5)
Decarboxylase (5)
Bombesin Receptor (5)
ACK (5)
CRFR (5)
TSH Receptor (5)
PYK2 (5)
MTH1 (5)
PAFR (5)
CGRP Receptor (5)
LIM Kinase (5)
cGAS (5)
Cell wall (4)
Melanin-concentrating Hormone Receptor (MCHR) (4)
Thrombopoietin Receptor (4)
Pyroptosis (4)
Adiponectin receptor (4)
Survivin (4)
KSP (4)
NEDD8 (4)
PROTAC Linker (4)
Galectin (4)
MALT (4)
CD73 (4)
DAPK (4)
advanced glycation end products (4)
Transaminase (3)
Haspin Kinase (3)
RANKL/RANK (3)
Na-K-Cl cotransporter (3)
Hexokinase (3)
Hck (3)
CPT (3)
HCN Channel (3)
CD38 (3)
Necroptosis (3)
Glutathione reductase (3)
OXPHOS (3)
GluCls (3)
KLF (3)
AIM2 (3)
VDA (2)
Taste receptor (2)
gp120/CD4 (2)
lysosomal autophagy (2)
Protease (2)
Apelin receptor (2)
Prolyl Endopeptidase (PREP) (2)
PGC-1α (2)
Fas/FasL (2)
GSNOR (2)
hCE (2)
EBI2/GPR183 (2)
ATTECs (2)
Integrase (2)
NUDIX hydrolase (2)
FABP (1)
N-Acetylglucosaminyltransferase (1)
Stemness kinase (1)
CYP19A1 (1)
RXFP receptor (1)
FOXO1 (1)
aconitase (1)
Piezo Channel (1)
PACAP (1)
Hydrogenase (1)
NMU2R (1)
Motilin Receptor (1)
HuR (1)
Thioredoxin (1)
Anion Exchanger (1)
Procollagen C Proteinase (1)
Neuropeptide W (1)
Fer/FerT kinase (1)
stilbene oxidase (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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