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已知活性化合物库

已知活性化合物库

产品编号 L4010 Bioactive Compounds Library Max
  库化合物信息   Excel SDF

已知活性库是 20980 个具有生物活性,能引起细胞、组织甚至个体生物学反应的化合物的集合。包括了正在进行临床前研究的药物分子,临床期的药物分子和已经上市的药物。靶点明确,信息全面,非常适合完成药物功能重定位、小分子诱导细胞分化以及机制研究中蛋白靶点确认等科研工作。

由于活性明确,靶点已知,很多科学家会从已知活性库中选择可以用于细胞诱导分化的小分子;通过单一或几个小分子的联合作用,筛选出能将各种体细胞诱导成为诱导多能干细胞,神经前体细胞,心肌细胞等的分子;甚至还有使用小分子组合在体内完成诱导分化的成功尝试。

已知活性库是对经典已知活性库的补充,添加了 TargetMol 特有,新颖的化合物(Part C),所有化合物靶点明确,且都进行过细胞水平活性测试,比上市药物库结构更为新颖,比类药化合物库更易发现活性化合物。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
我们的产品含有多种规格,如需了解具体的规格以及价格信息,请联系我们咨询订购,对于大额的订购,我们还有额外的优惠!
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如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
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产品描述

  • 20980个已知活性化合物的集合,可用于高通量筛选、高内涵筛选、细胞诱导和靶点确认;
  • 所有化合物都有相应的靶点信息的描述,活性研究更有保障和依据;
  • 是老药新用、细胞诱导靶点筛选的有效工具;
  • 涵盖多个疾病研究领域,如癌症、代谢、免疫和心血管系统等;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • 结构多样,药效显著,可渗透细胞;

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L4010)
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化合物库组成

Apoptosis (1047)
Antibacterial (831)
Autophagy (797)
Endogenous Metabolite (759)
Antibiotic (512)
5-HT Receptor (317)
AChR (281)
Antifungal (260)
Parasite (257)
COX (248)
DNA/RNA Synthesis (230)
Adrenergic Receptor (227)
NF-κB (225)
Dopamine Receptor (209)
HIV Protease (194)
CDK (185)
PI3K (178)
Potassium Channel (177)
EGFR (163)
Reactive Oxygen Species (161)
Calcium Channel (160)
P450 (155)
VEGFR (150)
Histamine Receptor (148)
Epigenetic Reader Domain (143)
Dehydrogenase (137)
Influenza Virus (134)
Sodium Channel (133)
PDE (133)
GABA Receptor (128)
Histone Methyltransferase (116)
PPAR (116)
Antioxidant (112)
HDAC (110)
Microtubule Associated (109)
GluR (107)
TRP/TRPV Channel (107)
TNF (101)
JAK (99)
Ferroptosis (96)
mTOR (95)
Akt (94)
Topoisomerase (94)
Src (93)
ERK (91)
STAT (90)
p38 MAPK (90)
Estrogen/progestogen Receptor (90)
GPR (89)
PDGFR (89)
FLT (88)
Wnt/beta-catenin (88)
Prostaglandin Receptor (86)
Phosphatase (85)
SARS-CoV (83)
AMPK (82)
PKC (79)
AChE (78)
Estrogen Receptor/ERR (77)
Adenosine Receptor (76)
FGFR (76)
Opioid Receptor (76)
HCV Protease (76)
iGluR (75)
PARP (73)
IL Receptor (71)
Caspase (70)
NMDAR (70)
Raf (70)
Virus Protease (69)
BCL (68)
c-Met/HGFR (67)
c-Kit (67)
NO Synthase (66)
RAAS (66)
MMP (65)
Androgen Receptor (64)
Nucleoside Antimetabolite/Analog (63)
Anti-infection (61)
Ras (60)
Proteasome (60)
Bcr-Abl (59)
TLR (59)
GSK-3 (58)
Sirtuin (58)
HSV (57)
ATPase (57)
Beta Amyloid (57)
HSP (56)
Mitochondrial Metabolism (56)
Phospholipase (55)
HBV (55)
MAO (55)
Glucocorticoid Receptor (53)
Aurora Kinase (53)
Mitophagy (53)
Lipoxygenase (53)
TGF-beta/Smad (51)
ROS (51)
ALK (51)
Tyrosinase (50)
E1/E2/E3 Enzyme (49)
Cannabinoid Receptor (48)
Antiviral (47)
HIF/HIF Prolyl-Hydroxylase (47)
JNK (47)
MAPK (46)
Drug Metabolite (46)
Interleukin (44)
MEK (44)
HER (43)
Reverse Transcriptase (42)
Monoamine Oxidase (41)
IκB/IKK (41)
P-gp (41)
DUB (41)
Nrf2 (41)
p53 (41)
CCR (41)
Antifection (40)
Tyrosine Kinases (40)
CXCR (40)
BTK (40)
Transferase (40)
NOS (39)
Histone Demethylase (38)
Casein Kinase (38)
DNA-PK (38)
Retinoid Receptor (37)
Serine/threonin kinase (37)
IGF-1R (37)
PKA (37)
HIF (36)
ROCK (36)
Serotonin Transporter (36)
Gamma-secretase (35)
S1P Receptor (35)
Integrin (34)
CaMK (34)
Cysteine Protease (34)
Carbonic Anhydrase (33)
c-RET (33)
LPL Receptor (32)
Immunology/Inflammation related (32)
TAM Receptor (32)
Serine Protease (31)
S6 Kinase (31)
Norepinephrine (31)
P2X Receptor (31)
ribosome (31)
Trk receptor (31)
Histone Acetyltransferase (29)
Proton pump (29)
Hedgehog/Smoothened (29)
Chloride channel (28)
PLK (28)
Progesterone Receptor (27)
Sigma receptor (27)
FAAH (26)
Fatty Acid Synthase (26)
FAK (26)
c-Fms (25)
Glucosidase (25)
Mdm2 (25)
DNA Alkylator/Crosslinker (25)
Aryl Hydrocarbon Receptor (25)
RIP kinase (25)
DPP-4 (24)
Neurokinin receptor (24)
NADPH (24)
Reductase (24)
ATM/ATR (23)
Syk (23)
Protease-activated Receptor (23)
Neuropeptide Y Receptor (23)
Thyroid hormone receptor(THR) (23)
Indoleamine 2,3-Dioxygenase (IDO) (23)
transporter (22)
DNA Methyltransferase (22)
Smo (22)
Chk (22)
Glucokinase (22)
HMG-CoA Reductase (21)
AhR (21)
Amino Acids and Derivatives (21)
Complement System (21)
NOD (21)
FXR (21)
Thrombin (20)
Kinesin (20)
SGLT (20)
CFTR (20)
Pim (20)
STING (19)
PDK (19)
Rho (19)
Lipase (19)
Endothelin Receptor (19)
P2Y Receptor (19)
MRP (19)
Acyltransferase (18)
ROR (18)
Glutathione Peroxidase (18)
Guanylate cyclase (18)
LRRK2 (18)
Hydroxylase (17)
DNA Alkylation (17)
OX Receptor (16)
PERK (16)
Glucagon Receptor (16)
PAK (16)
IRAK (16)
Epoxide Hydrolase (16)
Antifolate (16)
Leukotriene Receptor (16)
c-Myc (15)
LPA Receptor (15)
Melanocortin Receptor (15)
NOD-like Receptor (NLR) (15)
Xanthine Oxidase (15)
IRE1 (15)
DNA (14)
DYRK (14)
LTR (14)
Ephrin Receptor (14)
Liver X Receptor (14)
DHFR (14)
BACE (14)
PGE Synthase (14)
PD-1/PD-L1 (14)
cAMP (13)
Vasopressin Receptor (13)
GNRH Receptor (13)
Factor Xa (13)
CSF-1R (13)
Myosin (13)
IAP (12)
Ligand for E3 Ligase (12)
Telomerase (12)
DNA gyrase (12)
Platelet aggregation (12)
RSV (12)
Aminopeptidase (12)
Beta-Secretase (12)
ABC (12)
Isocitrate Dehydrogenase (IDH) (11)
GTPase (11)
Free radical scavengers (11)
ROS Kinase (11)
GPCR19 (11)
PI4K (11)
IDO (11)
Stearoyl-CoA Desaturase (SCD) (11)
CaSR (10)
cholecystokinin (10)
Aromatase (10)
PAI-1 (10)
IFNAR (10)
Phosphorylase (10)
YAP (10)
Monocarboxylate transporter (10)
Acetyl-CoA Carboxylase (10)
Neurotensin Receptor (10)
Lipid (10)
LDL (9)
Bradykinin Receptor (9)
GRK (9)
Melatonin Receptor (9)
Imidazoline Receptor (9)
Discoidin Domain Receptor (DDR) (9)
UGT (9)
GHSR (9)
Monoamine Transporter (9)
SGK (9)
ATP Citrate Lyase (9)
Adenylyl cyclase (8)
GST (8)
Porcupine (8)
NADPH-oxidase (8)
MT Receptor (8)
PKM (8)
CAT (8)
PTEN (8)
BCRP (8)
NAMPT (8)
CETP (8)
Tie-2 (7)
SIK (7)
Ligands for Target Protein for PROTAC (7)
Na+/Ca2+ Exchanger (7)
PAD (7)
ASK (7)
Gap Junction Protein (7)
MLK (7)
Neprilysin (7)
Arginase (7)
p97 (7)
Carboxypeptidase (6)
Wee1 (6)
PAFR (6)
Dynamin (6)
OCT (6)
GlyT (6)
MAGL (6)
OAT (6)
CRISPR/Cas9 (6)
CRFR (6)
Somatostatin (6)
BMI-1 (5)
MELK (5)
cGAS (5)
DprE1 (5)
MTH1 (5)
CRM1 (5)
VDAC (5)
MyD88 (5)
Aquaporin (5)
Oxytocin Receptor (5)
FLAP (5)
Adenosine deaminase (5)
Apelin receptor (5)
Bombesin Receptor (5)
TOPK (5)
RAR/RXR  (5)
MNK (5)
PROTACs (5)
APC (5)
GPX (5)
LIM Kinase (5)
Glutaminase (5)
Decarboxylase (5)
Galectin (4)
KSP (4)
Hippo pathway (4)
PYK2 (4)
DAPK (4)
Annexin A (4)
OXPHOS (4)
ACK (4)
MALT (4)
NEDD8 (4)
CGRP Receptor (4)
NPC1L1 (4)
Adiponectin receptor (4)
Pyroptosis (4)
cell cycle arrest (4)
Molecular Glues (4)
TSH Receptor (4)
Hck (4)
advanced glycation end products (4)
CD73 (4)
Survivin (3)
KLF (3)
Melanin-concentrating Hormone Receptor (MCHR) (3)
PROTAC Linker (3)
AAK1 (AP2 associated kinase 1) (3)
Thrombopoietin Receptor (3)
Hexokinase (3)
Cell wall (3)
Methionine Adenosyltransferase (MAT) (3)
Na-K-Cl cotransporter (3)
Angiotensin-converting Enzyme (ACE) (3)
CD38 (3)
Haspin Kinase (2)
Motilin Receptor (2)
GluCls (2)
lysosomal autophagy (2)
RANKL/RANK (2)
Taste receptor (2)
PGC-1α (2)
ATTECs (2)
VDA (2)
Necroptosis (2)
Integrase (2)
HCN Channel (2)
gp120/CD4 (2)
Glutathione reductase (2)
Transaminase (2)
EBI2/GPR183 (2)
hCE (2)
Prolyl Endopeptidase (PREP) (2)
Fas/FasL (2)
Thioredoxin (1)
FABP (1)
stilbene oxidase (1)
N-Acetylglucosaminyltransferase (1)
FOXO1 (1)
Piezo Channel (1)
Protease (1)
Fer/FerT kinase (1)
GSNOR (1)
aconitase (1)
LHRH (1)
Anion Exchanger (1)
Neuropeptide W (1)
NUDIX hydrolase (1)
Hydrogenase (1)
Stemness kinase (1)
NMU2R (1)
CYP19A1 (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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