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EMA 上市药物库

EMA 上市药物库

产品编号 L1020 EMA Approved Drug Library
  库化合物信息   Excel SDF

EMA 上市药物库收录了 670 个欧洲药品监督管理局(EMA)批准的化合物,所有化合物通过临床验证,靶点明确,具有较好的安全性和生物利用度,是进行老药新用理想的工具,可以大大提高药物研发的成功率,能够缩短药物研发周期,节约研发成本。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
咨询化合物库
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产品描述

  • 657个EMA批准药物的独特集合,可用于高通量筛选和高内涵筛选;
  • 经过了严格的临床前研究和临床试验,生物活性和安全性得到保障;
  • 涵盖多个研究领域:肿瘤、心血管药物、抗炎、免疫、神经系统药物、呼吸系统药物等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L1020)
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化合物库组成

Autophagy (121)
Apoptosis (87)
Antibacterial (52)
Antibiotic (51)
HIV Protease (50)
5-HT Receptor (34)
Adrenergic Receptor (32)
c-Kit (26)
VEGFR (24)
Endogenous Metabolite (23)
DNA/RNA Synthesis (22)
PDGFR (22)
Sodium Channel (21)
Dopamine Receptor (19)
SARS-CoV (19)
Ferroptosis (18)
HCV Protease (17)
Reverse Transcriptase (17)
Potassium Channel (16)
EGFR (16)
COX (16)
FLT (15)
P450 (15)
JAK (14)
Calcium Channel (13)
Antifungal (13)
Histamine Receptor (12)
Mitophagy (12)
Proteasome (12)
PDE (12)
AChR (12)
Src (12)
Topoisomerase (11)
Glucocorticoid Receptor (11)
Bcr-Abl (11)
Estrogen/progestogen Receptor (11)
PPAR (10)
Tyrosine Kinases (10)
Raf (10)
FGFR (10)
Thrombin (10)
Nucleoside Antimetabolite/Analog (10)
c-RET (9)
c-Met/HGFR (9)
Estrogen Receptor/ERR (9)
PARP (8)
Serotonin Transporter (8)
SGLT (8)
DPP-4 (8)
RAAS (8)
TAM Receptor (7)
CDK (7)
CFTR (7)
NF-κB (7)
ALK (7)
HBV (7)
MEK (7)
Influenza Virus (7)
Factor Xa (7)
ribosome (7)
Parasite (7)
Androgen Receptor (6)
MAO (6)
P2Y Receptor (6)
Dehydrogenase (6)
ROS (6)
Prostaglandin Receptor (6)
Antifolate (6)
Transferase (6)
Microtubule Associated (6)
TNF (6)
HSV (5)
Monoamine Oxidase (5)
NMDAR (5)
P-gp (5)
Norepinephrine (5)
S1P Receptor (5)
TRP/TRPV Channel (5)
Progesterone Receptor (5)
LPL Receptor (5)
Ligand for E3 Ligase (4)
DNA Alkylator/Crosslinker (4)
AMPK (4)
Reactive Oxygen Species (4)
ERK (4)
BCL (4)
Endothelin Receptor (4)
Neurokinin receptor (4)
Molecular Glues (4)
GABA Receptor (4)
DHFR (4)
BTK (4)
Carbonic Anhydrase (4)
Proton pump (4)
ROS Kinase (4)
Virus Protease (4)
Hydroxylase (3)
Cysteine Protease (3)
MMP (3)
Decarboxylase (3)
Trk receptor (3)
Adenosine Receptor (3)
mTOR (3)
Retinoid Receptor (3)
Hedgehog/Smoothened (3)
DNA Alkylation (3)
Ras (3)
HER (3)
ATPase (3)
iGluR (3)
Melatonin Receptor (3)
PI3K (3)
HIF (3)
Adenosine deaminase (2)
AChE (2)
ABC (2)
Antioxidant (2)
Phosphatase (2)
Protease-activated Receptor (2)
DNA Methyltransferase (2)
GPR (2)
Nrf2 (2)
RSV (2)
GHSR (2)
ROR (2)
Syk (2)
Ligands for Target Protein for PROTAC (2)
c-Fms (2)
CETP (2)
Ephrin Receptor (2)
CaSR (2)
Guanylate cyclase (2)
IL Receptor (2)
CCR (2)
FXR (2)
Fatty Acid Synthase (2)
Integrase (2)
Smo (2)
Opioid Receptor (2)
ROCK (2)
GluR (2)
Antifection (2)
Mitochondrial Metabolism (2)
DNA gyrase (2)
Aryl Hydrocarbon Receptor (2)
MT Receptor (2)
Drug Metabolite (2)
IRE1 (2)
Xanthine Oxidase (2)
PAK (2)
Rho (2)
Thrombopoietin Receptor (2)
NPC1L1 (1)
GNRH Receptor (1)
OAT (1)
CRM1 (1)
Monoamine Transporter (1)
Anti-infection (1)
Interleukin (1)
TGF-beta/Smad (1)
NADPH-oxidase (1)
MAPK (1)
HMG-CoA Reductase (1)
Monocarboxylate transporter (1)
Sigma receptor (1)
Tyrosinase (1)
Cannabinoid Receptor (1)
Beta-Secretase (1)
PGE Synthase (1)
Akt (1)
HIF/HIF Prolyl-Hydroxylase (1)
FAK (1)
NOD-like Receptor (NLR) (1)
CSF-1R (1)
AhR (1)
Telomerase (1)
Imidazoline Receptor (1)
Chloride channel (1)
PAFR (1)
PKM (1)
Amino Acids and Derivatives (1)
Complement System (1)
p38 MAPK (1)
CXCR (1)
Neprilysin (1)
GST (1)
Beta Amyloid (1)
Glutathione Peroxidase (1)
ACK (1)
STAT (1)
Cell wall (1)
GluCls (1)
HDAC (1)
Chk (1)
IFNAR (1)
CRISPR/Cas9 (1)
OX Receptor (1)
IGF-1R (1)
JNK (1)
Phospholipase (1)
CaMK (1)
Myosin (1)
Caspase (1)
ATP Citrate Lyase (1)
PKC (1)
Serine Protease (1)
Isocitrate Dehydrogenase (IDH) (1)
TLR (1)
YAP (1)
Arginase (1)
CGRP Receptor (1)
VDA (1)
UGT (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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