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Rotenone (Rotocide) 属于天然产物，是一种植物杀虫剂。Rotenone 是一种线粒体电子传递复合物 I 抑制剂，可以促进线粒体产生活性氧，并诱导细胞凋亡。

Bazinaprine 是一种选择性的、可逆的单胺氧化酶抑制剂(MAOI)，是治疗抑郁症的候选化合物。Bazinaprine 对A 型单胺氧化酶显示出较强的抑制作用，对b 型单胺氧化酶只显示出较弱的抑制作用。Bazinaprine 在体内可逆，但在体外不可逆。

Vardenafil (Vivanza) 是选择性、高效的、具有口服活性的磷酸二酯酶5抑制剂，IC50=0.7 nM。它能够非竞争性地抑制环磷酸鸟苷水解，从而提高 cGMP 水平。它对 PDE1 (180 nM)，PDE6 (11 nM)，PDE2，PDE3，PDE4 (>1000 nM) 具有选择性。它可用于研究勃起功能障碍。

PMSF (Phenylmethylsulfonyl fluoride) 是一种丝氨酸 半胱氨酸蛋白酶不可逆抑制剂，常用于制备细胞裂解物。

Aniline-d5(苯胺-d5)是Aniline的氘代同位素标记物，可用于同位素示踪。Aniline 通过铁过载和通过血红素加氧酶 1 上调诱导氧化应激对脾脏产生毒性，能够导致 p-IKKα 和 p-IKKβ 显着增加，进而增加 NF-κB 和 AP-1 结合活性。

Tripterin (Celastrol) 属于天然产物，是一种蛋白酶体抑制剂，抑制 20S 蛋白酶体的胰凝乳蛋白酶样活性 (IC50=2.5 μM)。Tripterin 具有抗炎、抗感染和免疫调节的作用。

1,2,3,4,6-O-Pentagalloylglucose (Penta-O-galloyl-β-D-glucose) 存在于多种植物中，具有重要的药理作用。Pentagalloylglucose 表现出显著的抗狂犬病病毒 (RABV) 活性。

Calcifediol (U 32070E) 属于天然产物，由 vitamin D3 在肝脏中代谢得到，是一种 VDR 配体。Calcifediol 适用于所有 vitamin D 缺乏症患者的维生素补充。

Bumetanide D5 is a deuterium-labeled Bumetanide. Bumetanide is a Na+-K+-Cl- (NKCC1) inhibitor (IC50s: 0.68 and 4.0 μM for hNKCC1A and hNKCC2A).

Edaravone, a novel and potent free radical scavenger, effectively prevents MMP-9-related brain hemorrhage in rats treated with tissue plasminogen activator. Its deuterium-labeled variant, Edaravone D5, retains the original compound's attributes while offering isotopic labeling benefits.

Nateglinide D5 is a deuterium labeled Nateglinide.

Nimesulide D5 is a deuterium labeled Nimesulide. Nimesulide is a selective inhibitor OF COX-2(IC50s of 70 nM-70 μM)

Phenindione D5 is deuterium labeled Phenindione, which functions as a Vitamin K antagonist.

Phenylacetylglutamine-D5 is a deuterated form of Phenylacetylglutamine.

Pirfenidone D5 is a deuterium labeled Pirfenidone. Pirfenidone is an antifibrotic agent that attenuates CCL2 and CCL12 production in fibrocyte cells.

Posaconazole-D5, a deuterium-labeled variant of Posaconazole, is a second-generation, broad-spectrum triazole compound with antifungal activity.

(rel)-Tranylcypromine D5 hydrochloride is a deuterium labeled (rel)-Tranylcypromine hydrochloride. (rel)-Tranylcypromine hydrochloride is an irreversible, nonselective inhibitor of monoamine oxidase (MAO) used in the treatment of depression.

Trandolaprilate D5 is a deuterium-labeled Trandolaprilate. Trandolaprilate is an inhibitor of angiotensin-converting enzyme (ACE).

5-Hydroxy Propafenone D5 HCl is the deuterium labeled 5-Hydroxy Propafenone.

Glycerol phenylbutyrate-D5 is a deuterium-labeled Glycerol phenylbutyrate. Glycerol phenylbutyrate is a sigma-2 (σ2) receptor ligand (pKi: 8.02).

Repaglinide D5 is deuterium labeled Repaglinide. Repaglinide is an insulin secretagogue for treatment type-2 diabetes mellitus.

Triamterene D5 is a deuterium-labeled Triamterene and can block epithelial Na+ channel (ENaC) in a voltage-dependent manner, used as a mild diuretic.

16α-Hydroxydehydroepiandrosterone-d5 (16α-Hydroxy-DHEA-d5) 是 16α-Hydroxydehydroepiandrosterone 的氘代形式。

D-CPP-ene is a NMDA antagonist.