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Search Results for " apen "

Targets Recommended: Calcium Channel GABA Receptor

33

抑制剂 & 化合物

7

天然产物

4

重组蛋白

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Cat. No.	Product Name	Target	Signaling Pathways
T6507	Gabapentin hydrochloride 加巴喷丁盐酸盐,Neurontin HCl,Gabapentin HCl	Calcium Channel; GABA Receptor	Membrane transporter/Ion channel; Metabolism; Neuroscience
	Gabapentin hydrochloride (Neurontin HCl) 是GABA 类似物，可用于缓解神经性疼痛。
T40622	Mapenterol hydrochloride	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Mapenterol hydrochloride 是 β2 肾上腺素受体激动剂。
T1629	Rifapentine MDL473,Rifapentina,Rifapentinum,DL 473,利福喷丁,Priftin,Cyclopentylrifampicin	DNA/RNA Synthesis; Antibacterial; Antibiotic	Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
	Rifapentine (Rifapentinum) 是可用于肺结核的抗生素。
T6411	Biapenem CLI 86815,比阿培南,Biapenern,Omegacin,L 627,LJC 10627	Antibacterial; Antibiotic	Microbiology/Virology
	Biapenem (CLI 86815) 是不经肠道的广谱碳青霉烯抗生素。
T0464	Carbetapentane citrate 托可拉斯,Pentoxyverine citrate,咳必清	AChR	Neuroscience
	Carbetapentane citrate (Pentoxyverine citrate) 能够选择性抑制咳嗽中枢，具有轻度的阿托品样作用和局麻作用。
T4990	Cefcapene pivoxil hydrochloride hydrate Cefcapene Pivoxil Hydrochloride,盐酸头孢卡品酯	Antibacterial; Antibiotic	Microbiology/Virology
	Cefcapene pivoxil hydrochloride hydrate 是一种头孢菌素的前药，具有口服活性和广谱抗菌活性。它可研究掌跖脓疱病等感染性疾病。
T68165	Trapencaine
	Trapencaine 是一种新合成的氨基甲酸型局部麻醉剂，诱导的肥大细胞膜上钠通道的构象变化。
T4991	Ertapenem sodium 厄他培南钠,MK-826,L-749345,尔他培南钠	Antibacterial; Antibiotic	Microbiology/Virology
	Ertapenem sodium (MK-826) 是碳青霉烯，是一种 β-内酰胺抗生素，具有广谱抗菌活性。
T0702	Gabapentin Neurontin,Gabapentine,加巴喷丁,Aclonium	Calcium Channel; GABA Receptor	Membrane transporter/Ion channel; Metabolism; Neuroscience
	Gabapentin (Neurontin) 是GABA 类似物，是一种抗癫痫药，可用于缓解神经性疼痛。
T8833	2-chloro-5-(16,18-dioxo-17-azapentacyclo[6.6.5.0~2,7~.0~9,14~.0~15,19~]nonadeca-2,4,6,9,11,13-hexaen-17-yl)benzoic acid	Others	Others
	2-chloro-5-(16,18-dioxo-17-azapentacyclo[6.6.5.0~2,7~.0~9,14~.0~15,19~]nonadeca-2,4,6,9,11,13-hexaen-17-yl)benzoic acid 可用于合成多种有机化合物。
T36999	7(S),17(S)-dihydroxy-8(E),10(Z),13(Z),15(E),19(Z)-Docosapentaenoic Acid
	Novel oxylipins, referred to as docosanoids, have been derived from C22polyunsaturated fatty acids 7(S),17(S)-dihydroxy-8(E),10(Z),13(Z),15(E),19(Z)-Docosapentaenoic acid (7(S),17(S)-hydroxy DPA) is a DPA-derived analog of the 17(S)-dihydroxy series of docosanoids known as protectins. Protectin D1, a DHA-derived dihydroxy fatty acid, exhibits potent anti-inflammatory activities.1,2,3Potentially, 7(S),17(S)-hydroxy DPA demonstrates similar properties; however, its biological activity has yet to b...
T4991L	Ertapenem (sodium salt)
	Ertapenem (sodium salt) 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T4991L，CAS号为 153832-38-3。
T16322	Nicodicosapent	Others	Others
	Nicodicosapent is a fatty acid niacin conjugate. It is also an inhibitor of the sterol regulatory element-binding protein (SREBP). The sterol regulatory element-binding protein (SREBP) is a key regulator of cholesterol metabolism proteins such as PCSK9, H
T27813	Lenapenem carbapenem
	Lenapenem is a broad-spectrum, carbapenem antibiotic with bactericidal activity by weakens the bacterial cell wall and leads to lytic cell death.
T37634	17-oxo-7(Z),10(Z),13(Z),15(E),19(Z)-Docosapentaenoic Acid
	Docosapentaenoic acid (DPA) is a ω-3 fatty acid found in fish oils. 17-oxo-7(Z),10(Z),13(Z),15(E),19(Z)-docosapentaenoic acid is a metabolite of lipoxygenase-mediated oxidation of DPA that is produced endogenously by aspirin-enhanced COX-2 activity. It has been shown to activate Nrf2-dependent antioxidant gene expression, to act as a PPARγ agonist (EC50 = ~200 nM), and to inhibit pro-inflammatory cytokine and nitric oxide production at biological concentration ranges (5-25 μM).
T37382	1,2,3-Trieicosapentaenoyl-rac-glycerol
	1,2,3-Trieicosapentaenoyl-rac-glycerol (EPA-TG) is a glycerol ester of eicosapentaenoic acid , which is an ω-3 fatty acid. An EPA-TG emulsion, administered i.v., lowers leukotriene B4 production by 40% in polymorphonuclear leukocytes from rabbits and reduces platelet aggregation. It suppresses natural killer cell activity both in vitro and in vivo, in human lymphocytes and murine spleens, respectively, with the in vivo effects lasting up to seven days.
T13284	Vapendavir diphosphate BTA798 diphosphate	Others	Others
	Vapendavir diphosphate is a potent enteroviral capsid binder (CB) and has a potent antiviral activity for enterovirus 71 (EV71) replication (EC50: 0.5-1.4 μM in different EV71 strains).
T131540	Capensin
	Capensin 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T131540。
T68149	tacapenem
	Tacapenem 是一种β-内酰胺类抗菌剂。它具有广谱抗菌活性，对β-内酰胺酶具有很高的稳定性。
T38278	9(Z),12(Z),15(Z),18(Z),21(Z)-Tetracosapentaenoic Acid
	9(Z),12(Z),15(Z),18(Z),21(Z)-Tetracosapentaenoic acid is an ω-3 very long-chain polyunsaturated fatty acid. It has been used to study the desaturation and elongation of ω-3 polyunsaturated fatty acids. It is elongated to form C26:5 or acted on by δ6 desaturase to form C24:6. 9(Z),12(Z),15(Z),18(Z),21(Z)-Tetracosapentaenoic acid is found at low levels in mouse brain and spleen and levels decrease in the brain and spleen of old and exceptionally old mice.
T20107	Ertapenem Invanz,MK0826,MK-0826,MK 0826
	Ertapenem is a parenteral carbapenem. It has a broad spectrum of antimicrobial activity. It is highly resistant to inactivation by a wide variety of beta-lactamases.
T65455	2,5,8,11,14-Pentaoxapentadecane
	2,5,8,11,14-Pentaoxapentadecane 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T65455，CAS号为 143-24-8。
T13284L	Vapendavir BTA798	Others	Others
	Vapendavir is a potent enteroviral capsid binder. Vapendavir has an effective antiviral activity for enterovirus 71 replication (EC50: 0.5-1.4 μM in different EV71 strains).
T36426	Eicosapentaenoyl 1-propanol-2-amide
	Monoacylglycerols (MAGs) of ω-3 polyunsaturated fatty acids have diverse physiological and health effects. In particular, MAGs containing docosahexaenoic acid or eicosapentaenoic acid have anti-proliferative properties against colon and lung cancer cell lines. Eicosapentaenoyl 1-propanol-2-amide is an EPA-containing MAG amide analog that inhibits the growth of human lung carcinoma A549 cells, producing 98.4% growth inhibition when applied at 3 μM. It is an analog of eicosapentaenoyl ethanolamide...
T37371	4(Z),7(Z),10(Z),13(Z),16(Z)-Nonadecapentaenoic Acid
	4(Z),7(Z),10(Z),13(Z),16(Z)-Nonadecapentaenoic acid is an unusual polyunsaturated fatty acid (PUFA) generated during the synthesis of docosahexaenoic acid-d5 . While the physiological properties of this compound are not known, dietary intake of n-3 long-chain PUFAs provides potential health benefits.
T10134	4,7,10,13,16-Docosapentaenoic acid	Others	Others
	4,7,10,13,16-Docosapentaenoic acid is an endogenous metabolite.
T70806	Metformin icosapent
	Metformin icosapent is an AMP-activated protein kinase (AMPK) activator that improves glycemic control by improving insulin sensitivity and decreasing intestinal absorption of glucose.
T29330	25-Desacetylrifapentine L14583,L-14583
	25-Desacetylrifapentine is the main metabolite of DL 473-IT in plasma.
T62218	Parapenzolate bromide
	Parapenzolate bromide 是一种口服具有活力的 mAChR 拮抗剂。Parapenzolate bromide 是一种抗胆碱能剂，也是一种解痉挛剂。
T15366	Gabapentin enacarbil XP-13512,加巴喷丁酯	Others; Calcium Channel	Membrane transporter/Ion channel; Metabolism; Others
	Gabapentin enacarbil (XP-13512) 是抗惊厥和镇痛药物加巴喷丁的前药。Gabapentin enacarbil 提供持续剂量比例的 Gabapentin 暴露和可预测的生物利用度。
T38208	Heneicosapentaenoic Acid
	Heneicosapentaenoic Acid (HPA) is a 21:5 ω-3 fatty acid present in trace amounts in the green alga B. pennata and in fish oils. Its chemical composition is similar to eicosapentaenoic acid (EPA) except elongated with one carbon on the carboxyl end, placing the first double bond in the δ6 position. HPA can be used to study the significance of the position of the double bonds in ω-3 fatty acids. It incorporates into phospholipids and into triacylglycerol in vivo with the same efficiency as EPA and...
T70473	Parapenzolate Free Base
	Parapenzolate Free Base is a safe and effective anticholinergic drug possessing antisecretory and antimotility properties and prolonged duration of action. Clinical investigation has shown that after an oral dose of the drug there was inhibition of both basal and histamine-stimulated acid outputs.
T37125	1,3-Dipalmitoyl-2-Eicosapentaenoyl-rac-glycerol
	1,3-Dipalmitoyl-2-eicosapentaenoyl-rac-glycerol is a triacylglycerol that contains palmitic acid at the sn-1 and sn-3 positions and eicosapentaenoic acid at the sn-2 position. Dietary administration of 1,3-dipalmitoyl-2-eicosapentaenoyl-rac-glycerol decreases hepatic triacylglycerol levels in mice.

化合物

Gabapentin hydrochloride

Cat.No: T6507

Synonym: 加巴喷丁盐酸盐,Neurontin HCl,Gabapentin HCl

Target: Calcium Channel, GABA Receptor

Mapenterol hydrochloride

Cat.No: T40622

Target: Adrenergic Receptor

Cat.No: T1629

Synonym: MDL473,Rifapentina,Rifapentinum,DL 473,利福喷丁,Priftin,Cyclopentylrifampicin

Target: DNA/RNA Synthesis, Antibacterial, Antibiotic

Cat.No: T6411

Synonym: CLI 86815,比阿培南,Biapenern,Omegacin,L 627,LJC 10627

Target: Antibacterial, Antibiotic

Carbetapentane citrate

Cat.No: T0464

Synonym: 托可拉斯,Pentoxyverine citrate,咳必清

Target: AChR

Cefcapene pivoxil hydrochloride hydrate

Cat.No: T4990

Synonym: Cefcapene Pivoxil Hydrochloride,盐酸头孢卡品酯

Target: Antibacterial, Antibiotic

Cat.No: T68165

Ertapenem sodium

Cat.No: T4991

Synonym: 厄他培南钠,MK-826,L-749345,尔他培南钠

Target: Antibacterial, Antibiotic

Cat.No: T0702

Synonym: Neurontin,Gabapentine,加巴喷丁,Aclonium

Target: Calcium Channel, GABA Receptor

2-chloro-5-(16,18-dioxo-17-azapentacyclo[6.6.5.0~2,7~.0~9,14~.0~15,19~]nonadeca-2,4,6,9,11,13-hexaen-17-yl)benzoic acid

Cat.No: T8833

Target: Others

7(S),17(S)-dihydroxy-8(E),10(Z),13(Z),15(E),19(Z)-Docosapentaenoic Acid

Cat.No: T36999

Ertapenem (sodium salt)

Cat.No: T4991L

Cat.No: T16322

Target: Others

Cat.No: T27813

Synonym: carbapenem

17-oxo-7(Z),10(Z),13(Z),15(E),19(Z)-Docosapentaenoic Acid

Cat.No: T37634

1,2,3-Trieicosapentaenoyl-rac-glycerol

Cat.No: T37382

Vapendavir diphosphate

Cat.No: T13284

Synonym: BTA798 diphosphate

Target: Others

Cat.No: T131540

Cat.No: T68149

9(Z),12(Z),15(Z),18(Z),21(Z)-Tetracosapentaenoic Acid

Cat.No: T38278

Cat.No: T20107

Synonym: Invanz,MK0826,MK-0826,MK 0826

2,5,8,11,14-Pentaoxapentadecane

Cat.No: T65455

Cat.No: T13284L

Synonym: BTA798

Target: Others

Eicosapentaenoyl 1-propanol-2-amide

Cat.No: T36426

4(Z),7(Z),10(Z),13(Z),16(Z)-Nonadecapentaenoic Acid

Cat.No: T37371

4,7,10,13,16-Docosapentaenoic acid

Cat.No: T10134

Target: Others

Metformin icosapent

Cat.No: T70806

25-Desacetylrifapentine

Cat.No: T29330

Synonym: L14583,L-14583

Parapenzolate bromide

Cat.No: T62218

Gabapentin enacarbil

Cat.No: T15366

Synonym: XP-13512,加巴喷丁酯

Target: Others, Calcium Channel

Heneicosapentaenoic Acid

Cat.No: T38208

Parapenzolate Free Base

Cat.No: T70473

1,3-Dipalmitoyl-2-Eicosapentaenoyl-rac-glycerol

Cat.No: T37125

Cat. No.	Product Name	Target	Signaling Pathways
T19295	Docosapentaenoic acid 22n-3	Endogenous Metabolite	Metabolism
	Docosapentaenoic acid 22n-3 是在所有动物细胞膜中发现的磷脂组成成分。
T7068	Eicosapentaenoic acid ethyl ester Icosapent ethyl,顺-二十碳五烯酸乙酯,EPA ethyl ester,Ethyl eicosapentaenoate	Others; Endogenous Metabolite	Metabolism; Others
	Eicosapentaenoic acid ethyl ester (Ethyl eicosapentaenoate) 是一种ω-3 脂肪酸剂和人内源性代谢物。
T5368	Eicosapentaenoic Acid	Histone Demethylase; Others; Endogenous Metabolite	Chromatin/Epigenetic; Metabolism; Others
	Eicosapentaenoic Acid 是一种 ω-3 脂肪酸。
TN4338	Isovouacapenol C	Others	Others
	Isovouacapenol C是一种天然产物，属于豆科云实属，其产品编号为 TN4338，CAS号为 455255-15-9。Isovouacapenol C可用作对照参考。
T40347	Eicosapentaenoic acid methyl ester
	Eicosapentaenoic acid methyl ester is a degradation product derived from monogalactosyl diacylglycerol, which is an apoptosis-inducing anticancer compound.
T72152	Eicosapentaenoic Acid sodium 二十碳五烯酸钠盐,Timnodonic acid sodium,EPA sodium
	Eicosapentaenoic Acid (EPA) sodium 为口服活性 ω-3 长链多不饱和脂肪酸 (ω-3 LC-PUFAs)。其通过DNA去甲基化，促进肿瘤抑制基因CCAAT/增强子结合蛋白δ (C/EBPδ)的重新表达，并通过H-RAS内含子1 CpG岛的去甲基化，激活U937白血病细胞中RAS/ERK/C/EBPβ途径。此外，该化合物能够促进血管平滑肌细胞松弛和血管舒张。
T83660	3(Z),6(Z),9(Z),12(Z),15(Z)-Octadecapentaenoic Acid C18:5 n-3,C18:5(3Z,6Z,9Z,12Z,15Z),all-cis-3,6,9,12,15-Octadecapentaenoic Acid
	3(Z),6(Z),9(Z),12(Z),15(Z)-Octadecapentaenoic acid 是一种在 G. kowalevskii 中发现的微藻 PUFA，常作为微藻和甲藻的化学分类生物标志物使用。

天然产物

Docosapentaenoic acid 22n-3

Cat.No: T19295

Target: Endogenous Metabolite

Eicosapentaenoic acid ethyl ester

Cat.No: T7068

Synonym: Icosapent ethyl,顺-二十碳五烯酸乙酯,EPA ethyl ester,Ethyl eicosapentaenoate

Target: Others, Endogenous Metabolite

Eicosapentaenoic Acid

Cat.No: T5368

Target: Histone Demethylase, Others, Endogenous Metabolite

Isovouacapenol C

Cat.No: TN4338

Target: Others

Eicosapentaenoic acid methyl ester

Cat.No: T40347

Eicosapentaenoic Acid sodium

Cat.No: T72152

Synonym: 二十碳五烯酸钠盐,Timnodonic acid sodium,EPA sodium

3(Z),6(Z),9(Z),12(Z),15(Z)-Octadecapentaenoic Acid

Cat.No: T83660

Synonym: C18:5 n-3,C18:5(3Z,6Z,9Z,12Z,15Z),all-cis-3,6,9,12,15-Octadecapentaenoic Acid

Species：

Expression System：

Tag：

Cat. No.	Product Name	Species	Expression System
TMPY-02433	APE1/APEX1 Protein, Human, Recombinant (His) APEX,HAP1,APX,APE,APEX nuclease (multifunctional DNA repair ...	Human	E. coli
	The enzyme is known to be a redox factor (Ref-1) stimulating DNA binding activity of AP-1 binding proteins such as Fos and Jun as well as a multifunctional DNA repair enzyme having 5' AP endonuclease, DNA 3' repair diesterase, 3'-5' exonuclease and DNA 3'-phosphatase activities.Although Apex mRNA was expressed ubiquitously, the levels varied significantly, suggesting organ- or tissue-specific expression of the Apex gene. The highest level was observed in the testis, relatively high levels in the...
TMPJ-00464	APE Protein, Human, Recombinant APEX,Apurinic-Apyrimidinic Endonuclease 1,APEN,DNA-...	Human	E. coli
	Apurinic-Apyrimidinic Endonuclease 1 (APE1) is required for efficient DNA base excision repair. When the DNA glycosylase remove the damaged bases, APE1 cleaves the AP site to allow resynthesis and ligation to complete repair. APE1 stimulates the DNA binding activity of many transcription factors, which participate in cancer promotion and progression. APE1 regulates the redox state of multiple transcription factors, such as c-Jun, c-Fos, NF-kB, p53. APEN is also involved in calcium-dependent down...
TMPY-05947	Influenza A H1N2 (A/swine/Papenburg/IDT12653/2010) Neuraminidase/NA Protein (His)	H1N2	HEK293 Cells
	Influenza A H1N2 (A/swine/Papenburg/IDT12653/2010) Neuraminidase/NA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 50.6 kDa and the accession number is V5J546.
TMPY-06675	Met e 1 Protein, Metapenaeus ensis, Recombinant	Metapenaeus ensis	E. coli
	Met e 1 Protein, Metapenaeus ensis, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 32.7 kDa.

重组蛋白

APE1/APEX1 Protein, Human, Recombinant (His)

Cat.No: TMPY-02433

Species: Human

Expression System: E. coli

APE Protein, Human, Recombinant

Cat.No: TMPJ-00464

Species: Human

Expression System: E. coli

Influenza A H1N2 (A/swine/Papenburg/IDT12653/2010) Neuraminidase/NA Protein (His)

Cat.No: TMPY-05947

Species: H1N2

Expression System: HEK293 Cells

Met e 1 Protein, Metapenaeus ensis, Recombinant

Cat.No: TMPY-06675

Species: Metapenaeus ensis

Expression System: E. coli

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