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TargetMol | Compound Library

代谢化合物库现货

Metabolism Compound Library
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货号 L2560

代谢是生物体内发生的用于维持生命的一系列有序化学反应的总称。这些反应使得生物体能够生长、繁殖以及对外界环境做出反应。代谢通常分为两类:分解代谢和合成代谢;分解代谢又称为异化作用,可以将环境中或细胞存储的营养物质进行分解以获得能量;合成代谢又称为同化作用,可以利用能量来合成细胞中的各个组分,二者的平衡使生物体保持自身的稳定,以适应环境。代谢中的化学反应几乎都是在酶的催化下进行的,从一个代谢物到另一个代谢物的代谢过程是通过一系列连续的酶促反应实现的,这种连续的酶促反应称为代谢途径。代谢紊乱、机体代谢途径的失调或中断会引发一系列代谢相关疾病。如糖尿病、肥胖、高血压、心血管疾病、癌症等。
Targetmol 代谢化合物库收集了3059 种代谢途径相关的化合物,是研究代谢相关疾病有用的工具。

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货号 L2560

代谢化合物库

规格

  • 1 mg
  • 10 μL x 10 mM (in DMSO)
  • 20 μL x 10 mM (in DMSO)
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

特点 特点

  • 3059种代谢途径相关生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 靶向糖代谢、脂质代谢、核苷酸代谢等多个代谢途径;靶点包括GLUT、Hexokinase、Pyruvate Kinase;ATGL、MAGL、FAAH等代谢相关热门靶点;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;

优势介绍 优势介绍

靶向脂代谢、糖代谢、核苷酸代谢、线粒体代谢等代谢通路相关靶点。

 Metabolism Compound Library
注:仅分析分布数量大于等于10个以上的通路。

涉及靶点相关性高,靶点数量多,包括Fatty Acid Synthase、Lipoxygenase、Mitochondrial Metabolism、α-glucosidase等。

 Metabolism Compound Library
注:仅分析分布数量大于等于20个以上的靶点。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

Apoptosis
Autophagy
Calcium Channel
PI3K
ROS
Reactive Oxygen Species
Dehydrogenase
Cytochromes P450
PDE
PPAR
Antibacterial
Endogenous Metabolite
Phosphatase
Akt
mTOR
NF-κB
AMPK
GSK-3
HIF/HIF Prolyl-Hydroxylase
Lipoxygenase
COX
Parasite
Phospholipase
Mitochondrial Metabolism
HSP
Antibiotic
CDK
DNA/RNA Synthesis
ERK
Casein Kinase
Glucosidase
Antifungal
Ferroptosis
Carbonic Anhydrase
Potassium Channel
p53
Reductase
Transferase
Retinoid Receptor
HIF
IGF-1R
MDM-2/p53
Serine/threonin kinase
Caspase
glycosidase
DNA-PK
S6 Kinase
FAAH
TNF
Acyltransferase
AChR
Glucokinase
Antioxidant
Fatty Acid Synthase
Interleukin
Influenza Virus
ATM/ATR
transporter
HIV Protease
Proteasome
p38 MAPK
PKA
PKC
NADPH
DPP-4
FXR
Wnt/beta-catenin
HMG-CoA Reductase
VEGFR
Sodium Channel
Virus Protease
Glutathione Peroxidase
Indoleamine 2,3-Dioxygenase (IDO)
IDO
PDK
ROR
Hydroxylase
DHFR
Lipase
Factor Xa
Bcl-2 Family
Src
JNK
SGLT
STAT
Mitophagy
GABA Receptor
MAGL
Epoxide Hydrolase
Glucocorticoid Receptor
Ras
Nrf2
NO Synthase
SARS-CoV
Adrenergic Receptor
Amino Acids and Derivatives
Serine Protease
IL Receptor
PARP
Liver X Receptor
Isocitrate Dehydrogenase (IDH)
Prostaglandin Receptor
Histamine Receptor
MMP
5-HT Receptor
PI4K
EGFR
Xanthine Oxidase
Antifolate
TGF-beta/Smad
TRP/TRPV Channel
Mdm2
HSV
Sirtuin
Stearoyl-CoA Desaturase (SCD)
Cannabinoid Receptor
Cholinesterase (ChE)
Aminopeptidase
Microtubule Associated
Anti-infection
Angiotensin-converting Enzyme (ACE)
PAI-1
P-gp
Acetyl-CoA Carboxylase
Tyrosinase
Aurora Kinase
Lipid
Beta Amyloid
MAPK
Adenosine Receptor
ALK
LDL
PKM
E1/E2/E3 Enzyme
FAK
Estrogen Receptor/ERR
MEK
FLT
c-Met/HGFR
NAMPT
PTEN
ATP Citrate Lyase
HDAC
Estrogen/progestogen Receptor
Drug Metabolite
ROCK
CaMK
Immunology/Inflammation related
GPCR
HCV Protease
OXPHOS
TLR
HBV
UGT
Antifection
Androgen Receptor
Neprilysin
IκB/IKK
Phosphorylase
SGK
Monoamine Oxidase
Chk
MAO
Leukotriene Receptor
Topoisomerase
ATPase
Dopamine Receptor
FGFR
SIK
MTP
Amylase
Aryl Hydrocarbon Receptor
Opioid Receptor
LTR
iGluR
RAAS
Vitamin
Trk receptor
Syk
DYRK
MELK
ROS Kinase
Proton pump
RAR/RXR
Bcr-Abl
Integrin
Hedgehog/Smoothened
Adenosine Deaminase
GPCR19
RSV
GST
Reverse Transcriptase
Chloride channel
FKBP
NADPH-oxidase
PERK
Tyrosine Kinases
PDGFR
CETP
Pim
Raf
Antiviral
NOD-like Receptor (NLR)
NMDAR
Hexokinase
PLK
Na+/Ca2+ Exchanger
c-Myc
Aromatase
Monocarboxylate transporter
Cysteine Protease
Prolyl Endopeptidase (PREP)
NEDD8
GluR
CFTR
Histone Methyltransferase
NPC1L1
Myosin
JAK
BACE
Thrombin
Gamma-secretase
CAT
PAK
cAMP
CPT
NOD
PD-1/PD-L1
NOS
DNA Alkylator/Crosslinker
CXCR
STING
Pyroptosis
GPX
MLK
Nucleoside Antimetabolite/Analog
IAP
ABC Transporter
Kras
PYK2
Glutaminase
RIP kinase
P2X Receptor
Survivin
Cholecystokinin Receptor
AAK1
LDLR
Epigenetic Reader Domain
Beta-Secretase
Decarboxylase
c-RET
TAM Receptor
c-Kit
DNA Methyltransferase
AhR
ADC Cytotoxin
P2Y Receptor
Cell Cycle Arrest
PAFR
c-Fms
Complement System
S1P Receptor
GSNOR
GTPase
Rho
AIM2
Histone Acetyltransferase
Cadherin
Free radical scavengers
Monoamine Transporter
DNA
ribosome
HER
Transaminase
MRP
BCRP
PGE Synthase
Urea Transporter
Cuproptosis
Kinesin
Taste receptor
Tie-2
FLAP
DNA Alkylation
Glutathione reductase
Liposome
NUDIX hydrolase
YAP
IFNAR
Necroptosis
Molecular Glues
hCE
PGK1
FOXO3
MicroRNA
Dynamin
LIM Kinase
DUB
OAT
MNK
Y Box Binding Protein 1
Arginase
gp120/CD4
Progesterone Receptor
CaSR
GNRH Receptor
Carboxypeptidase
REV-ERB
Gap Junction Protein
Platelet aggregation
IRAK
MyD88
DprE1
Melatonin Receptor
DNA gyrase
Guanylate cyclase
Norepinephrine
LRRK2
GluCls
Hydrogenase
Factor VIIa
Histone Demethylase
N-Acetylglucosaminyltransferase
ATG
NR4A
Anion Exchanger
PROTAC Linker
CCR
Transketolase
Porcupine
cGAS
p62
CRISPR/Cas9
Imidazoline Receptor
LPL Receptor
Adenylate cyclase
Ligands for E3 Ligase
Somatostatin
PAD
Aquaporin
DAPK
Protease-activated Receptor
Aconitase
CSF-1R
Thioredoxin
FOXO
Neurokinin receptor
APC/C
Procollagen C Proteinase
OCT
RANKL/RANK
GRK
AAK1 (AP2 associated kinase 1)
Na-K-Cl cotransporter
Bombesin Receptor
ACK1
Telomerase
TMV
LPA Receptor
PGC-1α
BTK

Keywords

MetabolismCompoundLibrary