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TargetMol | Compound Library

代谢化合物库现货

Metabolism Compound Library
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货号 L2560

代谢是生物体内发生的用于维持生命的一系列有序化学反应的总称。这些反应使得生物体能够生长、繁殖以及对外界环境做出反应。代谢通常分为两类:分解代谢和合成代谢;分解代谢又称为异化作用,可以将环境中或细胞存储的营养物质进行分解以获得能量;合成代谢又称为同化作用,可以利用能量来合成细胞中的各个组分,二者的平衡使生物体保持自身的稳定,以适应环境。代谢中的化学反应几乎都是在酶的催化下进行的,从一个代谢物到另一个代谢物的代谢过程是通过一系列连续的酶促反应实现的,这种连续的酶促反应称为代谢途径。代谢紊乱、机体代谢途径的失调或中断会引发一系列代谢相关疾病。如糖尿病、肥胖、高血压、心血管疾病、癌症等。
Targetmol 代谢化合物库收集了3059 种代谢途径相关的化合物,是研究代谢相关疾病有用的工具。

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货号 L2560

代谢化合物库

规格

  • 1 mg
  • 10 μL x 10 mM (in DMSO)
  • 20 μL x 10 mM (in DMSO)
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

特点 特点

  • 3059种代谢途径相关生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 靶向糖代谢、脂质代谢、核苷酸代谢等多个代谢途径;靶点包括GLUT、Hexokinase、Pyruvate Kinase;ATGL、MAGL、FAAH等代谢相关热门靶点;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;

优势介绍 优势介绍

靶向脂代谢、糖代谢、核苷酸代谢、线粒体代谢等代谢通路相关靶点。

 Metabolism Compound Library
注:仅分析分布数量大于等于10个以上的通路。

涉及靶点相关性高,靶点数量多,包括Fatty Acid Synthase、Lipoxygenase、Mitochondrial Metabolism、α-glucosidase等。

 Metabolism Compound Library
注:仅分析分布数量大于等于20个以上的靶点。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

Apoptosis
ROS
Autophagy
Reactive Oxygen Species
PI3K
Cytochromes P450
Akt
Endogenous Metabolite
Dehydrogenase
PDE
Antibacterial
PPAR
NF-κB
mTOR
Phosphatase
AMPK
Mitochondrial Metabolism
GSK-3
COX
Amino Acids and Derivatives
HIF/HIF Prolyl-Hydroxylase
ERK
Parasite
Lipoxygenase
Phospholipase
Caspase
Antifungal
Antibiotic
Reductase
Transferase
p38 MAPK
DNA/RNA Synthesis
Ferroptosis
Interleukin
Glucosidase
Wnt/beta-catenin
glycosidase
Antioxidant
IGF-1R
p53
CDK
TNF
MDM-2/p53
HIF
NO Synthase
Nrf2
JNK
NADPH
STAT
Calcium Channel
Acyltransferase
Sirtuin
Fatty Acid Synthase
Potassium Channel
Glutathione Peroxidase
S6 Kinase
Bcl-2 Family
ATM/ATR
HIV Protease
Glucokinase
HMG-CoA Reductase
Ras
DNA-PK
Influenza Virus
FAAH
Lipase
DPP-4
MMP
PARP
Xanthine Oxidase
AChR
VEGFR
FXR
Retinoid Receptor
Virus Protease
PKC
Indoleamine 2,3-Dioxygenase (IDO)
DHFR
Hydroxylase
IDO
5-HT Receptor
Liver X Receptor
ROR
Lipid
PDK
IL Receptor
Src
GABA Receptor
EGFR
Aminopeptidase
Mitophagy
PKA
transporter
Prostaglandin Receptor
SARS-CoV
GPCR
MAGL
P-gp
TLR
SGLT
Drug Metabolite
Epoxide Hydrolase
Adrenergic Receptor
Stearoyl-CoA Desaturase (SCD)
Microtubule Associated
PI4K
Acetyl-CoA Carboxylase
Anti-infection
Monoamine Oxidase
Adenosine Receptor
Isocitrate Dehydrogenase (IDH)
TGF-beta/Smad
Beta Amyloid
Antifolate
HBV
TRP/TRPV Channel
Topoisomerase
OXPHOS
Tyrosinase
Estrogen Receptor/ERR
Aromatase
PKM
Cholinesterase (ChE)
HDAC
Phosphorylase
Mdm2
Sodium Channel
UGT
Aurora Kinase
FAK
Amylase
JAK
HSV
FLT
NOD-like Receptor (NLR)
Immunology/Inflammation related
MAPK
PTEN
Histamine Receptor
Casein Kinase
MEK
c-Met/HGFR
NAMPT
ALK
Antifection
Aryl Hydrocarbon Receptor
Opioid Receptor
Cannabinoid Receptor
IκB/IKK
Dopamine Receptor
Androgen Receptor
ATPase
PERK
iGluR
MAO
Estrogen/progestogen Receptor
HCV Protease
Epigenetic Reader Domain
Glucocorticoid Receptor
ROS Kinase
NOS
MTP
Leukotriene Receptor
GPX
NADPH-oxidase
Integrin
FOXO
E1/E2/E3 Enzyme
ATP Citrate Lyase
SGK
Chk
Proton pump
RAAS
HSP
Carbonic Anhydrase
Nucleoside Antimetabolite/Analog
ROCK
Raf
CaMK
Bcr-Abl
Serine Protease
Cell Cycle Arrest
LTR
Antiviral
Reverse Transcriptase
PGC-1α
Histone Methyltransferase
Survivin
FGFR
Chloride channel
RAR/RXR
LDL
Pyroptosis
Hedgehog/Smoothened
Decarboxylase
Adenosine Deaminase
PDGFR
CETP
GST
Kras
Angiotensin-converting Enzyme (ACE)
Trk receptor
Syk
Cysteine Protease
FKBP
Proteasome
DYRK
MELK
NOD
Gamma-secretase
NMDAR
GPCR19
Monocarboxylate transporter
LRRK2
Free radical scavengers
NPC1L1
Tyrosine Kinases
GluR
Molecular Glues
CAT
c-Myc
Photosensitizer
cAMP
PD-1/PD-L1
Hexokinase
DUB
RSV
PLK
S1P Receptor
MyD88
DNA Alkylator/Crosslinker
Serine/threonin kinase
FABP
CXCR
Myosin
Beta-Secretase
c-RET
ATG
IAP
DNA
CFTR
IFNAR
BACE
AhR
CPT
Gap Junction Protein
Transaminase
LPL Receptor
PYK2
BCRP
PGE Synthase
Glucagon Receptor
Prolyl Endopeptidase (PREP)
MLK
Cholecystokinin Receptor
LDLR
SIK
FLAP
DNA Alkylation
TAM Receptor
PROTACs
Histone Demethylase
NR4A
ABC Transporter
p62
ribosome
HER
Necroptosis
Pim
FOXO3
c-Kit
Arginase
ASCT
Dipeptidyl Peptidase
IRAK
PGK1
ADC Cytotoxin
MRP
Adenylate cyclase
RIP kinase
Urea Transporter
Cuproptosis
DAPK
Kinesin
P2Y Receptor
HCAR
c-Fms
Complement System
Arrestin
Norepinephrine
STING
Aconitase
Tie-2
Glutathione reductase
Liposome
PROTAC Linker
Transketolase
Sigma receptor
NUDIX hydrolase
YAP
GRK
Telomerase
DNA Methyltransferase
Thrombin
GSNOR
GTPase
Rho
PAK
Ephrin Receptor
AIM2
Histone Acetyltransferase
Platelet aggregation
IKZF
Glutaminase
Ligands for E3 Ligase
Somatostatin
PAD
Mucin
ASK
Methionine Adenosyltransferase (MAT)
Aquaporin
MicroRNA
Dynamin
B7
PAFR
Orphan Receptor
PANoptosis
OAT
MNK
AUTACs
NEDD4-1
Protease
Tight Junction Protein
DprE1
Melatonin Receptor
IRE1
Guanylate cyclase
Bradykinin Receptor
Cadherin
GluCls
Sulfotransferase
CGRP Receptor
Glyoxalase
Thyroid hormone receptor(THR)
Serotonin Transporter
CSF-1R
Neurokinin receptor
APC/C
stilbene oxidase
Hydrogenase
CD38
N-Acetylglucosaminyltransferase
Adiponectin Receptor
Monoamine Transporter
Anion Exchanger
CCR
FMO
Porcupine
CRISPR/Cas9
Imidazoline Receptor
Advanced Glycation End Products
Piezo Channel
OCT
RANKL/RANK
Annexin A
Na-K-Cl cotransporter
Bombesin Receptor
ACK1
Cholesterol synthesis
hCE
TMV
LPA Receptor
BMI-1
Y Box Binding Protein 1
gp120/CD4
GNRH Receptor
BTK
GHR
PAI-1
REV-ERB
Vitamin
Ferroportin
IGF-2R

Keywords

MetabolismCompoundLibrary