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TargetMol | Compound Library

代谢化合物库现货

Metabolism Compound Library
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货号 L2560

代谢是生物体内发生的用于维持生命的一系列有序化学反应的总称。这些反应使得生物体能够生长、繁殖以及对外界环境做出反应。代谢通常分为两类:分解代谢和合成代谢;分解代谢又称为异化作用,可以将环境中或细胞存储的营养物质进行分解以获得能量;合成代谢又称为同化作用,可以利用能量来合成细胞中的各个组分,二者的平衡使生物体保持自身的稳定,以适应环境。代谢中的化学反应几乎都是在酶的催化下进行的,从一个代谢物到另一个代谢物的代谢过程是通过一系列连续的酶促反应实现的,这种连续的酶促反应称为代谢途径。代谢紊乱、机体代谢途径的失调或中断会引发一系列代谢相关疾病。如糖尿病、肥胖、高血压、心血管疾病、癌症等。
Targetmol 代谢化合物库收集了3059 种代谢途径相关的化合物,是研究代谢相关疾病有用的工具。

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货号 L2560

代谢化合物库

规格

  • 1 mg
  • 10 μL x 10 mM (in DMSO)
  • 20 μL x 10 mM (in DMSO)
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

特点 特点

  • 3059种代谢途径相关生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 靶向糖代谢、脂质代谢、核苷酸代谢等多个代谢途径;靶点包括GLUT、Hexokinase、Pyruvate Kinase;ATGL、MAGL、FAAH等代谢相关热门靶点;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;

优势介绍 优势介绍

靶向脂代谢、糖代谢、核苷酸代谢、线粒体代谢等代谢通路相关靶点。

 Metabolism Compound Library
注:仅分析分布数量大于等于10个以上的通路。

涉及靶点相关性高,靶点数量多,包括Fatty Acid Synthase、Lipoxygenase、Mitochondrial Metabolism、α-glucosidase等。

 Metabolism Compound Library
注:仅分析分布数量大于等于20个以上的靶点。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

Apoptosis
Autophagy
Calcium Channel
PI3K
ROS
Reactive Oxygen Species
Dehydrogenase
Cytochromes P450
PDE
PPAR
Antibacterial
Endogenous Metabolite
Phosphatase
mTOR
Akt
NF-κB
AMPK
GSK-3
HIF/HIF Prolyl-Hydroxylase
COX
Lipoxygenase
Parasite
HSP
Phospholipase
Mitochondrial Metabolism
Antibiotic
CDK
DNA/RNA Synthesis
Casein Kinase
Carbonic Anhydrase
Glucosidase
Ferroptosis
Antifungal
Reductase
ERK
Potassium Channel
Transferase
p53
Retinoid Receptor
HIF
IGF-1R
MDM-2/p53
Serine/threonin kinase
Caspase
DNA-PK
glycosidase
FAAH
S6 Kinase
Glucokinase
Acyltransferase
TNF
Antioxidant
AChR
Interleukin
transporter
Influenza Virus
ATM/ATR
HIV Protease
Fatty Acid Synthase
p38 MAPK
PKA
PKC
Proteasome
NADPH
Wnt/beta-catenin
FXR
HMG-CoA Reductase
DPP-4
Virus Protease
Sodium Channel
Glutathione Peroxidase
VEGFR
IDO
Indoleamine 2,3-Dioxygenase (IDO)
DHFR
ROR
PDK
Hydroxylase
Lipase
JNK
Factor Xa
SGLT
STAT
Src
Mitophagy
Bcl-2 Family
Glucocorticoid Receptor
MAGL
Epoxide Hydrolase
Adrenergic Receptor
SARS-CoV
Nrf2
GABA Receptor
Ras
NO Synthase
Amino Acids and Derivatives
Histamine Receptor
PARP
Serine Protease
Liver X Receptor
Isocitrate Dehydrogenase (IDH)
IL Receptor
Prostaglandin Receptor
MMP
5-HT Receptor
Antifolate
TRP/TRPV Channel
Xanthine Oxidase
EGFR
PI4K
Mdm2
Stearoyl-CoA Desaturase (SCD)
HSV
TGF-beta/Smad
Cholinesterase (ChE)
Aminopeptidase
Sirtuin
Beta Amyloid
Cannabinoid Receptor
Anti-infection
Microtubule Associated
Aurora Kinase
P-gp
PAI-1
Acetyl-CoA Carboxylase
Tyrosinase
Adenosine Receptor
Estrogen Receptor/ERR
E1/E2/E3 Enzyme
LDL
Angiotensin-converting Enzyme (ACE)
Lipid
ALK
MEK
FLT
FAK
PKM
GPCR
Estrogen/progestogen Receptor
c-Met/HGFR
NAMPT
ROCK
Drug Metabolite
PTEN
CaMK
ATP Citrate Lyase
HDAC
HCV Protease
HBV
Immunology/Inflammation related
UGT
Phosphorylase
Antifection
Androgen Receptor
OXPHOS
MAPK
TLR
IκB/IKK
Neprilysin
SGK
Monoamine Oxidase
ATPase
Dopamine Receptor
Leukotriene Receptor
MAO
SIK
Topoisomerase
Chk
MTP
LTR
RAAS
Amylase
Aryl Hydrocarbon Receptor
iGluR
Opioid Receptor
FGFR
Vitamin
Proton pump
RAR/RXR
Integrin
DYRK
Pim
Bcr-Abl
Hedgehog/Smoothened
Trk receptor
MELK
Adenosine Deaminase
Syk
ROS Kinase
Chloride channel
CETP
PERK
Tyrosine Kinases
Raf
JAK
PDGFR
GPCR19
RSV
GST
FKBP
NADPH-oxidase
NOD-like Receptor (NLR)
NOS
NPC1L1
Monocarboxylate transporter
Histone Methyltransferase
NEDD8
BACE
Na+/Ca2+ Exchanger
Cysteine Protease
Myosin
NMDAR
Hexokinase
GluR
Antiviral
Reverse Transcriptase
Aromatase
PLK
NOD
Thrombin
CFTR
CAT
DNA Alkylator/Crosslinker
c-Myc
Cholecystokinin Receptor
Nucleoside Antimetabolite/Analog
PYK2
Glutaminase
LDLR
IAP
Prolyl Endopeptidase (PREP)
RIP kinase
PAFR
Gamma-secretase
P2X Receptor
ABC Transporter
PAK
CXCR
cAMP
Epigenetic Reader Domain
Beta-Secretase
PGE Synthase
Survivin
STING
CPT
Decarboxylase
Pyroptosis
GPX
Kras
c-RET
c-Kit
DNA Methyltransferase
TAM Receptor
AhR
MLK
PD-1/PD-L1
ADC Cytotoxin
Taste receptor
GSNOR
Transaminase
NUDIX hydrolase
YAP
P2Y Receptor
IFNAR
Necroptosis
Tie-2
GTPase
MRP
AAK1
Rho
Cell Cycle Arrest
Adenylate cyclase
FLAP
Monoamine Transporter
Molecular Glues
DNA Alkylation
Cadherin
DNA
BCRP
Glutathione reductase
Free radical scavengers
Urea Transporter
Histone Acetyltransferase
AIM2
hCE
c-Fms
ribosome
Cuproptosis
Complement System
Liposome
S1P Receptor
HER
Kinesin
FOXO3
PGK1
MicroRNA
Hydrogenase
Dynamin
MyD88
DprE1
Y Box Binding Protein 1
Arginase
Procollagen C Proteinase
Factor VIIa
LPL Receptor
Aconitase
Histone Demethylase
gp120/CD4
Progesterone Receptor
Melatonin Receptor
OCT
CaSR
N-Acetylglucosaminyltransferase
GNRH Receptor
ATG
NR4A
RANKL/RANK
CSF-1R
FABP
GRK
AAK1 (AP2 associated kinase 1)
DNA gyrase
Na-K-Cl cotransporter
Anion Exchanger
Guanylate cyclase
PROTAC Linker
Ligands for E3 Ligase
Thioredoxin
Bombesin Receptor
CCR
ACK1
Somatostatin
PAD
Transketolase
Norepinephrine
DUB
Telomerase
MNK
OAT
Porcupine
LRRK2
cGAS
GluCls
p62
Carboxypeptidase
TMV
LPA Receptor
CRISPR/Cas9
Aquaporin
FOXO
REV-ERB
Gap Junction Protein
Neurokinin receptor
DAPK
Platelet aggregation
APC/C
IRAK
Protease-activated Receptor
Imidazoline Receptor
Glyoxalase
PGC-1α
BTK

Keywords

MetabolismCompoundLibrary