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代谢化合物库

代谢化合物库

产品编号 L2560 Metabolism Compound Library
  库化合物信息   Excel SDF

代谢是生物体内发生的用于维持生命的一系列有序化学反应的总称。这些反应使得生物体能够生长、繁殖以及对外界环境做出反应。代谢通常分为两类:分解代谢和合成代谢;分解代谢又称为异化作用,可以将环境中或细胞存储的营养物质进行分解以获得能量;合成代谢又称为同化作用,可以利用能量来合成细胞中的各个组分,二者的平衡使生物体保持自身的稳定,以适应环境。代谢中的化学反应几乎都是在酶的催化下进行的,从一个代谢物到另一个代谢物的代谢过程是通过一系列连续的酶促反应实现的,这种连续的酶促反应称为代谢途径。代谢紊乱、机体代谢途径的失调或中断会引发一系列代谢相关疾病。如糖尿病、肥胖、高血压、心血管疾病、癌症等。

Targetmol 代谢化合物库收集了2350 种代谢途径相关的化合物,是研究代谢相关疾病有用的工具。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
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特点

  • 2350种代谢途径相关生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 靶向糖代谢、脂质代谢、核苷酸代谢等多个代谢途径;靶点包括GLUT、Hexokinase、Pyruvate Kinase;ATGL、MAGL、FAAH等代谢相关热门靶点;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;

化合物库定制

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包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L2560)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

Autophagy (305)
Apoptosis (290)
PI3K (192)
Endogenous Metabolite (164)
Reactive Oxygen Species (163)
Calcium Channel (159)
P450 (143)
Dehydrogenase (122)
PDE (114)
PPAR (111)
mTOR (101)
Akt (97)
Antibacterial (93)
AMPK (82)
Phosphatase (78)
GSK-3 (71)
COX (60)
Mitochondrial Metabolism (53)
NF-κB (51)
HSP (50)
Lipoxygenase (49)
Phospholipase (48)
Ferroptosis (46)
Antibiotic (46)
Parasite (45)
CDK (42)
HIF/HIF Prolyl-Hydroxylase (40)
DNA-PK (37)
Antifungal (35)
Transferase (34)
Casein Kinase (34)
Carbonic Anhydrase (34)
Serine/threonin kinase (33)
p53 (33)
DNA/RNA Synthesis (32)
IGF-1R (31)
S6 Kinase (30)
HIF (30)
Potassium Channel (30)
Retinoid Receptor (26)
AChR (26)
Reductase (26)
HIV Protease (26)
ERK (26)
Glucosidase (24)
Fatty Acid Synthase (24)
Influenza Virus (24)
NADPH (23)
DPP-4 (23)
ROS (22)
FAAH (22)
Proteasome (22)
Indoleamine 2,3-Dioxygenase (IDO) (22)
transporter (22)
ATM/ATR (22)
PKC (22)
FXR (21)
Amino Acids and Derivatives (21)
HMG-CoA Reductase (21)
PKA (21)
Antioxidant (20)
ROR (19)
PDK (19)
Wnt/beta-catenin (19)
Acyltransferase (19)
Glucokinase (19)
Sodium Channel (19)
Mitophagy (18)
Lipase (18)
Glutathione Peroxidase (17)
TNF (17)
Caspase (17)
Hydroxylase (17)
Src (17)
Glucocorticoid Receptor (16)
Epoxide Hydrolase (16)
GABA Receptor (16)
p38 MAPK (16)
VEGFR (16)
PARP (15)
SGLT (15)
Virus Protease (14)
Liver X Receptor (14)
IL Receptor (13)
Factor Xa (13)
DHFR (13)
STAT (13)
JNK (13)
P-gp (12)
Adrenergic Receptor (12)
Adenosine Receptor (12)
PI4K (12)
Xanthine Oxidase (12)
FLT (11)
5-HT Receptor (11)
IDO (11)
Antifolate (11)
Stearoyl-CoA Desaturase (SCD) (11)
TRP/TRPV Channel (11)
MMP (11)
Lipid (11)
Aminopeptidase (11)
Isocitrate Dehydrogenase (IDH) (11)
Acetyl-CoA Carboxylase (11)
Prostaglandin Receptor (10)
PAI-1 (10)
HSV (10)
Aurora Kinase (10)
Histamine Receptor (10)
UGT (9)
NO Synthase (9)
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MEK (9)
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SGK (9)
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PKM (8)
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Nrf2 (8)
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Chk (7)
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ALK (7)
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c-RET (3)
IAP (3)
HER (3)
Hexokinase (3)
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TAM Receptor (3)
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JAK (3)
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PLK (3)
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MRP (2)
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Glutaminase (2)
P2Y Receptor (2)
PAK (2)
IFNAR (2)
hCE (2)
PGC-1α (2)
LRRK2 (1)
stilbene oxidase (1)
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cAMP (1)
GSNOR (1)
Kinesin (1)
Telomerase (1)
Bombesin Receptor (1)
Thioredoxin (1)
LPA Receptor (1)
Tie-2 (1)
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Transaminase (1)
MyD88 (1)
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Pyroptosis (1)
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DUB (1)
Guanylate cyclase (1)
PD-1/PD-L1 (1)
DprE1 (1)
DNA Methyltransferase (1)
FABP (1)
Histone Demethylase (1)
PAFR (1)
PAD (1)
Histone Methyltransferase (1)
DNA (1)
Somatostatin (1)
DAPK (1)
ROS Kinase (1)
Hydrogenase (1)
GTPase (1)
CSF-1R (1)
CRISPR/Cas9 (1)
P2X Receptor (1)
Progesterone Receptor (1)
OAT (1)
NUDIX hydrolase (1)
Immunology/Inflammation related (1)
PGE Synthase (1)
Melatonin Receptor (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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