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TargetMol | Compound Library

代谢化合物库现货

Metabolism Compound Library
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货号 L2560

代谢是生物体内发生的用于维持生命的一系列有序化学反应的总称。这些反应使得生物体能够生长、繁殖以及对外界环境做出反应。代谢通常分为两类:分解代谢和合成代谢;分解代谢又称为异化作用,可以将环境中或细胞存储的营养物质进行分解以获得能量;合成代谢又称为同化作用,可以利用能量来合成细胞中的各个组分,二者的平衡使生物体保持自身的稳定,以适应环境。代谢中的化学反应几乎都是在酶的催化下进行的,从一个代谢物到另一个代谢物的代谢过程是通过一系列连续的酶促反应实现的,这种连续的酶促反应称为代谢途径。代谢紊乱、机体代谢途径的失调或中断会引发一系列代谢相关疾病。如糖尿病、肥胖、高血压、心血管疾病、癌症等。
Targetmol 代谢化合物库收集了3059 种代谢途径相关的化合物,是研究代谢相关疾病有用的工具。

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货号 L2560

代谢化合物库

规格

  • 1 mg
  • 10 μL x 10 mM (in DMSO)
  • 20 μL x 10 mM (in DMSO)
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

特点 特点

  • 3059种代谢途径相关生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 靶向糖代谢、脂质代谢、核苷酸代谢等多个代谢途径;靶点包括GLUT、Hexokinase、Pyruvate Kinase;ATGL、MAGL、FAAH等代谢相关热门靶点;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;

优势介绍 优势介绍

靶向脂代谢、糖代谢、核苷酸代谢、线粒体代谢等代谢通路相关靶点。

 Metabolism Compound Library
注:仅分析分布数量大于等于10个以上的通路。

涉及靶点相关性高,靶点数量多,包括Fatty Acid Synthase、Lipoxygenase、Mitochondrial Metabolism、α-glucosidase等。

 Metabolism Compound Library
注:仅分析分布数量大于等于20个以上的靶点。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

Apoptosis
Autophagy
Calcium Channel
PI3K
ROS
Reactive Oxygen Species
Dehydrogenase
Cytochromes P450
PDE
PPAR
Antibacterial
Endogenous Metabolite
Phosphatase
mTOR
Akt
NF-κB
AMPK
GSK-3
HIF/HIF Prolyl-Hydroxylase
COX
Lipoxygenase
Parasite
HSP
Phospholipase
Mitochondrial Metabolism
Antibiotic
CDK
DNA/RNA Synthesis
Casein Kinase
Glucosidase
Carbonic Anhydrase
Antifungal
Potassium Channel
Ferroptosis
ERK
Reductase
p53
Transferase
Retinoid Receptor
HIF
IGF-1R
MDM-2/p53
Serine/threonin kinase
Caspase
DNA-PK
glycosidase
S6 Kinase
FAAH
Acyltransferase
TNF
Glucokinase
AChR
Antioxidant
Interleukin
Fatty Acid Synthase
Influenza Virus
ATM/ATR
transporter
HIV Protease
p38 MAPK
PKA
PKC
Proteasome
HMG-CoA Reductase
FXR
NADPH
Wnt/beta-catenin
DPP-4
Virus Protease
Sodium Channel
Indoleamine 2,3-Dioxygenase (IDO)
VEGFR
Glutathione Peroxidase
IDO
ROR
DHFR
PDK
Hydroxylase
Lipase
JNK
SGLT
STAT
Factor Xa
Mitophagy
Src
Bcl-2 Family
MAGL
Epoxide Hydrolase
Glucocorticoid Receptor
Ras
SARS-CoV
Nrf2
NO Synthase
Adrenergic Receptor
GABA Receptor
Amino Acids and Derivatives
Serine Protease
IL Receptor
Histamine Receptor
Prostaglandin Receptor
PARP
Liver X Receptor
Isocitrate Dehydrogenase (IDH)
MMP
PI4K
5-HT Receptor
Antifolate
Xanthine Oxidase
TRP/TRPV Channel
EGFR
TGF-beta/Smad
Stearoyl-CoA Desaturase (SCD)
HSV
Mdm2
Aminopeptidase
Microtubule Associated
Cannabinoid Receptor
Beta Amyloid
Anti-infection
Cholinesterase (ChE)
Sirtuin
Aurora Kinase
P-gp
Acetyl-CoA Carboxylase
Tyrosinase
Lipid
PAI-1
FAK
Angiotensin-converting Enzyme (ACE)
Estrogen Receptor/ERR
LDL
PKM
MEK
FLT
E1/E2/E3 Enzyme
Adenosine Receptor
ALK
Estrogen/progestogen Receptor
Drug Metabolite
PTEN
ROCK
CaMK
ATP Citrate Lyase
HDAC
GPCR
c-Met/HGFR
NAMPT
UGT
Antifection
Androgen Receptor
Immunology/Inflammation related
MAPK
Neprilysin
IκB/IKK
HCV Protease
OXPHOS
TLR
Phosphorylase
SGK
Monoamine Oxidase
HBV
Dopamine Receptor
Chk
SIK
Leukotriene Receptor
Topoisomerase
ATPase
MAO
MTP
FGFR
RAAS
Amylase
Aryl Hydrocarbon Receptor
Opioid Receptor
LTR
iGluR
Vitamin
Bcr-Abl
Trk receptor
Syk
Integrin
Hedgehog/Smoothened
Adenosine Deaminase
Proton pump
RAR/RXR
Pim
DYRK
MELK
ROS Kinase
GPCR19
RSV
JAK
Chloride channel
FKBP
NADPH-oxidase
CETP
Raf
Antiviral
NOD-like Receptor (NLR)
PERK
Tyrosine Kinases
PDGFR
GST
Reverse Transcriptase
Histone Methyltransferase
NMDAR
Hexokinase
PLK
NPC1L1
Myosin
NOS
Monocarboxylate transporter
Cysteine Protease
Prolyl Endopeptidase (PREP)
BACE
Thrombin
NEDD8
GluR
CFTR
Na+/Ca2+ Exchanger
Aromatase
NOD
PYK2
Glutaminase
RIP kinase
P2X Receptor
PGE Synthase
Survivin
PAFR
Gamma-secretase
Cholecystokinin Receptor
LDLR
Epigenetic Reader Domain
Beta-Secretase
Decarboxylase
c-RET
TAM Receptor
DNA Alkylator/Crosslinker
CXCR
STING
Pyroptosis
GPX
MLK
c-Kit
DNA Methyltransferase
AhR
Nucleoside Antimetabolite/Analog
IAP
ABC Transporter
KRas
CAT
c-Myc
PAK
cAMP
CPT
PD-1/PD-L1
ADC Cytotoxin
Transaminase
MRP
Adenylate cyclase
BCRP
Urea Transporter
Cuproptosis
Kinesin
P2Y Receptor
Cell Cycle Arrest
c-Fms
Complement System
S1P Receptor
Taste receptor
Tie-2
AAK1
FLAP
DNA Alkylation
Glutathione reductase
Liposome
Cadherin
Free radical scavengers
NUDIX hydrolase
YAP
IFNAR
Necroptosis
Molecular Glues
hCE
Monoamine Transporter
DNA
ribosome
HER
GSNOR
GTPase
Rho
Histone Acetyltransferase
AIM2
PGK1
FOXO3
LPL Receptor
Ligands for E3 Ligase
Somatostatin
PAD
Aquaporin
DAPK
Protease-activated Receptor
MicroRNA
Dynamin
DUB
OAT
MNK
Aconitase
CSF-1R
Thioredoxin
FOXO
Neurokinin receptor
APC/C
MyD88
DprE1
Melatonin Receptor
FABP
DNA gyrase
Guanylate cyclase
Norepinephrine
LRRK2
GluCls
Glyoxalase
Procollagen C Proteinase
OCT
RANKL/RANK
GRK
AAK1 (AP2 associated kinase 1)
Na-K-Cl cotransporter
Bombesin Receptor
ACK1
Telomerase
TMV
LPA Receptor
Hydrogenase
Factor VIIa
Histone Demethylase
N-Acetylglucosaminyltransferase
ATG
NR4A
Anion Exchanger
PROTAC Linker
CCR
Transketolase
Porcupine
cGAS
p62
CRISPR/Cas9
Imidazoline Receptor
Y Box Binding Protein 1
Arginase
gp120/CD4
Progesterone Receptor
CaSR
GNRH Receptor
Carboxypeptidase
REV-ERB
Gap Junction Protein
Platelet aggregation
IRAK
PGC-1α
BTK

Keywords

MetabolismCompoundLibrary