Cat. No. | Product Name | CAS No. | Purity | Chemical Structure |
---|---|---|---|---|
T32208 | Isogentisin
异龙胆黄素
|
491-64-5 | 95.1% |
|
Isogentisin (BRN 0258402) 是一种从龙胆科植物中分离出来的化合物,是一种用于预防吸烟引起的内皮损伤的新型化合物。Isogentisin 对单胺氧化酶具有抑制作用。 | ||||
T10617 | Brofaromine
化合物 T10617
|
63638-91-5 | 98% |
|
Brofaromine (CGP 11305A) is an MAO inhibitor (IC50: 0.2 μM for MAO-A). | ||||
TN3294 | 8alpha-(2-Methylacryloyloxy)hirsutinolide 13-O-acetate
化合物 TN3294
|
67667-71-4 | 98% |
|
8alpha-(2-Methylacryloyloxy)hirsutinolide 13-O-acetate shows inhibitory activity toward CYP2A6 and MAO-A and MAO-B enzymes. | ||||
TN2553 | 1-Methyl-2-undecyl-4(1H)-quinolone
化合物 TN2553
|
59443-02-6 | 98% |
|
1-Methyl-2-undecyl-4(1H)-quinolone, and dihydroevocarpine should also be served as the chemical markers together with evodiamine for the quality control of Evodi... | ||||
TN3300 | 8alpha-Tigloyloxyhirsutinolide 13-O-acetate
化合物 TN3300
|
83182-58-5 | 98% |
|
8alpha-Tigloyloxyhirsutinolide 13-O-acetate shows inhibitory activity toward CYP2A6 and MAO-A and MAO-B enzymes. 8alpha-Tigloyloxyhirsutinolide 13-O-acetate has ... | ||||
TN4137 | Glicoricone
化合物 TN4137
|
161099-37-2 | 98% |
|
Glicoricone acts as a partial estrogen antagonist. Glicoricone inhibited the monoamine oxidase with the IC50 values of 6.0 x 10(-5)-1.4 x 10(-4) M. | ||||
T5470 | LAZABEMIDE
拉扎贝胺
|
103878-84-8 | 98% |
|
Lazabemide (Ro 19-6327) 是一种单胺氧化酶 B 的选择性的可逆抑制剂 ,但对 MAO-A 活性较低。它高浓度时具有抑制单胺摄取的作用,能够抑制去甲肾上腺素、血清素和多巴胺摄取,其IC50值分别为 86 μM、123 μM 和 >500 μM。它可用于研究帕金森和阿尔茨海默病。 | ||||
T16770 | Ro 41-1049 hydrochloride
化合物 T16770
|
127917-66-2 | 98% |
|
Ro 41-1049 hydrochloride is a reversible and selective inhibitor of monoamine oxidase-A (Kd: 16.5 and 64.4 nM, respectively). | ||||
TN1099 | Dihydroevocarpine
二氢吴茱萸卡品碱
|
15266-35-0 | 98% |
|
Dihydroevocarpine shows potent anti-Helicobacter pylori activity with the minimum inhibitory concentration (MIC) value of 10-20 microg/ml. Dihydroevocarpine is a... | ||||
TN2790 | 2'-O-Methylperlatolic acid
化合物 TN2790
|
38968-07-9 | 98% |
|
2'-O-Methylperlatolic acid and confluentic acid are monoamine oxidase B inhibitors in a Brazilian plant, Himatanthus sucuuba. | ||||
TN3024 | 4'-Demethyleucomin
化合物 TN3024
|
34818-83-2 | 98% |
|
4'-Demethyleucomin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3024,CAS号为 34818-83-2。 | ||||
TN3918 | Echitovenidine
化合物 TN3918
|
7222-35-7 | 98% |
|
Echitovenidine shows monoamine oxidase inhibitor activity. | ||||
TN3116 | 5-Hydroxy-1-methoxyxanthone
化合物 TN3116
|
27770-13-4 | 98% |
|
5-Hydroxy-1-methoxyxanthone, 1,5-dihydroxyxanthone and 6-deoxyjacareubin are all antifungal against Cladosporium cucumerinum, while they show differing degrees o... | ||||
TN3726 | Cudraflavone B
化合物 TN3726
|
19275-49-1 | 98% |
|
Cudraflavone B has anti-proliferative activity, mouse brain monoamine oxidase (MAO) inhibitory effects, apoptotic actions in human gastric carcinoma cells and mo... | ||||
T15023 | CX-157
化合物 T15023
|
205187-53-7 | 98% |
|
CX-157 is a reversible monoamine oxidase-A (MAO-A) inhibitor (EC50:19.3 ng/mL). | ||||
T18918 | Azure B
天青 B
|
531-55-5 | BS |
|
Azure B (Azure B chloride) 是一种 Methylene blue 的主要代谢物,是一种阳离子染料,用于 Azure 曙红染色剂以进行血液涂片染色。它是高选择性和可逆的抑制单胺氧化酶(MAO)-A 的抑制剂,对重组人的 MAO-A 和 MAO-B 的IC50分别为 11 和 968 nM。它具有显... | ||||
T0751 | Furazolidone
呋喃唑酮
|
67-45-8 | 99.98% |
|
Furazolidone (Furoxone) 是一种具有抗菌和抗原虫活性的硝基呋喃衍生物,抑制AML1-ETO 转化细胞,IC50为12.7 μM。 | ||||
T8907 | Minaprine dihydrochloride
米那卜林二盐酸盐
|
25953-17-7 | 99.97% |
|
Minaprine dihydrochloride 是一种可逆的单胺氧化酶 MAO-A 抑制剂,对乙酰胆碱酯酶有微弱抑制,是一种抗抑郁类化合物。 | ||||
T0369 | Ethaverine hydrochloride
盐酸依沙维林
|
985-13-7 | 99.90% |
|
Ethaverine hydrochloride (Ethaquin) 是罂粟碱的同系物。 | ||||
T6651L | Safinamide
沙芬酰胺
|
133865-89-1 | 99.9% |
|
Safinamide (FCE-26743) 是一种可逆选择性单胺氧化酶 B (IC50 0.098μM)抑制剂,可减少多巴胺的降解,也是一种谷氨酸释放抑制剂(IC50 8μM)。它还能抑制多巴胺的再摄取。 Safinamide 还能阻断钠和钙通道。 Safinamide 的潜在的其他用途可能是帕金森病、不宁腿综合征和癫... |