racemate

BPO-27 racemate (BPO-27(racemate)) 是一种CFTR 抑制剂，IC50为8 nM。

ELN318463 racemate (ELN 318463 racemate) 是 ELN318463 的外消旋体，ELN318463 是一种淀粉样前体蛋白 (APP) 选择性 γ-分泌酶抑制剂。

SCH 42495 racemate is the racemate of SCH 42495. SCH 42495 is an orally active neutral inhibitor of metalloendopeptidase (NEP), with antihypertensive effect.

Seviteronel racemate is the racemate form of Seviteronel and is a potent inhibitor of CYP17 lyase.

GNE-140 is a potent inhibitor of lactate dehydrogenase A (LDHA). GNE-140 is a racemate mixture of (R)-GNE-140 and (S)-GNE-140.

Ibrutinib is a selective, irreversible Btk inhibitor (IC50: 0.5 nM). Ibrutinib Racemate is the racemate of Ibrutinib.

Streptonigrin is an aminoquinone antitumor and antibacterial antibiotic produced by Streptomyces flocculus. Streptonigrin inhibits β-Catenin/Tcf signaling and shows cytotoxicity in β-catenin-activated cells. Streptonigrin induces delayed chromosomal instability involving interstitial telomeric sequences in Chinese hamster ovary cells. Note: Streptonigrin from natural resource is (-)-rotation, has CAS#3930-19-6 and is a R-isomer.

GSK963 是手性的选择性受体相互作用蛋白 1 酶抑制剂，其IC50值为 29 nM。它在体外强效选择性抑制小鼠和人细胞的坏死。

Cobimetinib racemate (Cobimetinib (racemate)) 是 Cobimetinib 的外消旋体，是一种选择性 MEK 抑制剂。

(Rac)-SAR131675 是一种有效的、选择性的VEGFR3抑制剂，其IC50=23 nM。

(Rac)-ABT-202 dihydrochloride 是 ABT-202 的外消旋体。ABT-202 是烟碱乙酰胆碱受体激动剂，可用作镇痛剂。

(Rac)-BRD0705 是 BRD0705 的活性较低的外消旋体。 BRD0705 是一种有效的特异性 GSK3α 抑制剂。

(Rac)-Byakangelicin (7H-Furo[3,2-g][1]benzopyran-7-one, 9-(2,3-dihydroxy-3-methylbutoxy)-4-methoxy-) 是一种 Byakangelicin 的外消旋体，主要分离自 Angelica 属中。其中 Byakangelicin 是醛糖还原酶抑制剂(IC50:6.2 μM)，可用作抗肿瘤剂。

(Rac)-JBJ-04-125-02 (JBJ-04-125-02) 是 JBJ-04-125-02 的消旋体，是选择性突变，可口服的 EGFR 变构抑制剂，对EGFRL858R/T790M 的IC50为 0.26 nM。

DHMEQ racemate is an NF-κB inhibitor. The activity of DHMEQ racemate is lower than (-)-DHMEQ.

N-0861 racemate is the racemate of N-0861.

LY 344864 racemate 是一种 5-HT1F 受体激动剂。

Implitapide Racemate is the racemate of Implitapide. Implitapide is an inhibitor of microsomal triglyceride transfer protein (MTP).

CAL-130 Racemate is the racemate of CAL-130. CAL-130 is a PI3Kδ and PI3Kγ inhibitor (IC50s: 1.3 and 6.1 nM).

Derazantinib Racemate (ARQ-087 Racemate) 是 Derazantinib 的外消旋体。Derazantinib 是一种有效的，ATP 竞争型的，具有口服活性的酪氨酸激酶抑制剂，能够抑制软骨细胞 FGFR1 (IC50:4.5 nM)、FGFR2 (IC50:1.8 nM)、FGFR3 (IC50:4.5nM)。

GDC-0834 Racemate is the racemate form of GDC-0834, which is an effective and selective BTK inhibitor

INCB054329 Racemate is an inhibitor of BET protein.

KUL 7211 is a selective β-adrenoceptor agonist. KUL 7211 racemate is the racemate of KUL 7211.

Litronesib is a selective, allosteric inhibitor of kinesin Eg5.Litronesib (Racemate) is the racemate of litronesib.