adrenoreceptor

(±)-Befunolol is a blocking agent of β-adrenoceptor.

Fenoterol hydrobromide (Phenoterol hydrobromide) 是一种具有口服活性和选择性的 β2-肾上腺素受体激动剂，也是支气管扩张剂，可用于研究哮喘和支气管炎等心血管疾病。

Higenamine hydrochloride (norcoclaurine HCl) 是一种 β2-AR 激动剂，是用于心力衰竭相关研究的中药乌头的关键成分，具有抗凋亡活性。

Quetiapine (ICI204636) 是5-HT 受体激动剂和多巴胺受体拮抗剂，对人5-HT1A 的 pEC50值为 4.77，对人 D2的 pIC50值为 6.33。它用于治疗精神分裂症，以及治疗与 I 型双相情感障碍相关的急性躁狂发作。它对人 D2、HT1、5-HT2A、5-HT2C 受体具有中高等亲和力，pKi 值为 7.25、5.74、7.54和5.55。

Taprizosin (UK-338003) mesylate 是 α 肾上腺素 (α-adrenoreceptor) 拮抗剂。

Bufuralol hydrochloride (盐酸布呋洛尔) 属于 beta-肾上腺素受体拮抗剂，是一种强效的非选择性 beta-adrenoreceptor 拮抗剂，具有部分激动活性且口服有效。Bufuralol hydrochloride 是 CYP2D6 的典型探针底物 (Km = 5-50 microM)，广泛用于表征 CYP2D6 的酶活性、其遗传变异的功能评价以及药物代谢动力学分析。

α2-adrenoreceptor antagonist

Broxaterol is a β2 adrenoreceptor agonist. It is part of a class of drugs that affect the smooth muscle receptors in the body.

L-Mabuterol HCl is a selective agonist of β2 adrenoreceptor.

Befunolol is a beta blocker with intrinsic sympathomimetic activity and also acts as a β adrenoreceptor partial agonist.

Hexoprenaline Sulfate is a selective beta2-adrenoreceptor agonist. Hexoprenaline Sulfate is active in man as a bronchodilator by the oral or intravenous routes and by inhalation. Hexoprenaline Sulfate is indicated for use in the treatment of bronchospasm

Mabuterol is a selective agonist of β2 adrenoreceptor with no beta 1-stimulation. Mabuterol inhibited the positive inotropic effect of isoprenaline at 10(-7) g/ml and decreased the maximum driving frequency at 3 X 10(-6) g/ml. Mabuterol was 3 times more p

Pirbuterol, a short-acting β2 adrenoreceptor agonist, has bronchodilating action used in the treatment of asthma.

Reproterol hydrochloride, a β2 adrenoreceptor agonist, is used to treat asthma and chronic obstructive pulmonary disease (COPD).

Ro 16-8714 is an agonist of beta-adrenoreceptor with antihyperglycemic and thermogenic properties.

Vatinoxan is a peripheral α2 adrenoreceptor antagonist.

Etiguanfacine(SSP-1871) is a agonist of α2-adrenoreceptor.

Fasobegron is a agonist of β3-adrenoreceptor .

Lubabegron(LY488756) is used as an agonist of β3-adrenoreceptor in veterinary.

Ronactolol is an aminopropanol derivative with beta-adrenoreceptor blocking activity.

Zoleprodolol is a antagonist of adrenoreceptor.

Povafonidine (PGE-6201204) 是一种有效的 α-2 肾上腺素受体激动剂。Povafonidine 可以收缩血管，减轻粘膜充血，可用于鼻塞研究。

Oxyfedrine 是具有口服活性的 β-肾上腺素受体的激动剂。Oxyfedrine 是一种血管扩张剂，可降低冠状动脉血管的张力，用于研究心血管疾病。

Aminomenthylnorepinephrine is a partial agonist of the beta-adrenoreceptor that causes irreversible inactivation.