- 全部删除
您的购物车当前为空
LY231617是一种可口服和能穿透血脑屏障的抗氧化剂,能够减轻大鼠全身缺血性神经元损伤。LY231617能够对H2O2诱导的毒性具有神经保护作用,抑制脂质过氧化。


为众多的药物研发团队赋能,
让新药发现更简单!
LY231617是一种可口服和能穿透血脑屏障的抗氧化剂,能够减轻大鼠全身缺血性神经元损伤。LY231617能够对H2O2诱导的毒性具有神经保护作用,抑制脂质过氧化。
| 规格 | 价格 | 库存 | 数量 |
|---|---|---|---|
| 1 mg | ¥ 315 | In stock | |
| 5 mg | ¥ 745 | In stock | |
| 10 mg | ¥ 1,160 | In stock | |
| 25 mg | ¥ 2,380 | In stock | |
| 50 mg | ¥ 3,480 | In stock | |
| 100 mg | ¥ 4,960 | In stock | |
| 200 mg | ¥ 6,860 | In stock | |
| 1 mL x 10 mM (in DMSO) | ¥ 818 | In stock |
LY231617 相关产品
| 产品描述 | LY231617 is an orally bioavailable, blood-brain barrier-penetrant antioxidant that mitigates systemic ischaemic neuronal injury in rats. It exerts neuroprotective effects against H₂O₂-induced toxicity by inhibiting lipid peroxidation. |
| 体外活性 | LY231617(0.25-25 μM)与海马细胞共孵育一夜后,可削弱 H₂O₂ 对海马细胞培养物的毒性,10 μM 时效果最显著[1]。 |
| 体内活性 | 在大鼠四血管闭塞模型中,LY231617(50 mg/kg)在缺血前30分钟通过口服给药,能够显著减轻神经元损伤[2]。LY231617(20 mg/kg)在缺血后30分钟经静脉给药,可有效保护海马和纹状体免受四血管闭塞所导致的损害[2]。 |
| 别名 | LY-231617 |
| 分子量 | 299.88 |
| 分子式 | C17H30ClNO |
| CAS No. | 141545-89-3 |
| Smiles | Cl.OC=1C(=CC(=CC1C(C)(C)C)CNCC)C(C)(C)C |
| 密度 | no data available |
| 颜色 | Yellow |
| 物理性状 | Solid |
| 存储 | store under nitrogen | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. | |||||||||||||||||||||||||||||||||||
| 溶解度信息 | DMSO: 200 mg/mL (666.93 mM), Sonication is recommended. Ethanol: <29.99 mg/mL, Sonication is recommended. | |||||||||||||||||||||||||||||||||||
溶液配制表 | ||||||||||||||||||||||||||||||||||||
DMSO
| ||||||||||||||||||||||||||||||||||||
评论内容