gs-2

Ganoderic acid GS-2 inhibits the activity of the human immunodeficiency virus-1 (HIV-1) protease.

GS-2278是一种高效的LPAR1 (溶血磷脂酸受体 1) 拮抗剂，预期可应用于特发性肺纤维化 (IPF) 的研究。

CGS-27023A is a novel matrix metalloproteinase inhibitor.

CM-352是一种金属蛋白酶抑制剂，可减少脑损伤并改善脑出血大鼠模型的功能恢复。

Letrozole (CGS 20267) 是一种可口服的，选择性可逆的非甾体类芳香化酶抑制剂，IC50值为 11.5 nM。它选择性抑制雌激素的生物合成，可研究乳腺癌。

CGS 21680 是一种选择性的腺苷和腺苷 A2A 受体激动剂，Ki 值为 27 nM。

GS 283 is a Ca(2+) antagonist. GS 283 is also a weak histamine and muscarinic receptor blocker in rat and guinea pig tracheal smooth muscles.

Compound AJ-3（RGS2–Galpha-q interaction-IN-1）是一种抑制RGS2-Galpha-q相互作用的化合物。它能有效抑制表达RGS2的癌细胞生长，并具有阻止细胞迁移的特性。

CGS 20625 是一种具有口服活性、特异性和高效性的中枢苯二氮卓受体的部分激动剂，具有抗焦虑和抗惊厥活性。CGS 20625 对 [3H]-氟硝西泮与中枢苯二氮卓受体的结合有抑制作用，可用于研究焦虑症和癫痫等神经系统疾病。

Cgs 25155 is an orally active inhibitor of NEP 24.11.

CGS 24012 is a bioactive chemical.

CGS 27023A 是一种非肽类强效口服活性基质溶解素抑制剂。

CGS 21680 Hydrochloride (CGS 21680 HCl) 是一种选择性腺苷 A2A 受体激动剂，Ki 值为 27 nM。

Dolispan is a Histamine H1 Antagonist.

VULM 993 is a calcium antagonist.

Cgs 27830 is an Endothelin Receptor Antagonist.

Cgs 26303 is a potent non-peptidic inhibitor of neutral endopeptidase capable of protecting atrial natriuretic peptide from enzymatic degradation.

Tofenacin (free base) is an antidepressant drug with a tricyclic-like structure. It acts as a serotonin-norepinephrine reuptake inhibitor, and based on its close relation to orphenadrine, may also possess anticholinergic and antihistamine properties. Tofenacin is also the major active metabolite of orphenadrine and likely plays a role in its beneficial effects against depressive symptoms seen in Parkinson's disease patients.

Cgs 25015 inhibits endothelin-converting enzyme.

Saussureamine C is an inhibitor of H274Y and N294S mutants.

CGS 25462 is a neutral endopeptidase (NEP) inhibitor.

Lu 26-046 is a muscarinic receptor agonist.

Cgs 22706 is an adenosine A2 receptor antagonist.

Smurf1 inhibitor 1 is a inhibitor that promotes bone formation.