mrs

BroMhexine IMpurity B 试剂用于制备 Ambroxol 和 Bromhexine (B678600) 代谢物 Ambroxol EP Impurity E。

MRS 1754 是A2B 腺苷受体选择性拮抗剂，对人和大鼠的 A1和 A3受体的亲和力非常低。

MRS-3777 hemioxalate 是一种选择性腺苷 A3 受体拮抗剂，可逆转其相应激动剂的抗伤害感受作用，可用于研究炎症性疼痛。

MRS-1191 is an effective and selective A3 adenosine receptor antagonist (KB: 92 nM, a Ki: 31.4 nM for human A3 receptor and an IC50: 120 nM for CHO cells).

MRS 1523 can exert an antihyperalgesic effect through N-type Ca channel block and action potential inhibition in isolated rat dorsal root ganglion (DRG) neurons. MRS 1523 is an effective and selective adenosine A3 receptor antagonist Ki: 18.9 nM and 113 n

MRS1177 is an effective and selective antagonist of the human Adenosine A3 receptor (hA3AR) (Ki: 0.3 nM).

MRS1186 is an effective and selective antagonist of the human Adenosine A3 receptor (Ki: 7.66 nM).

MRS2698 is an effective and highly selective agonist of the P2Y2 receptor (EC50: 8 nM). MRS2698 also is >300-fold P2Y2-selective versus the P2Y4 and P2Y6 receptors.

MRS4608是一种新型的P2Y14受体强效拮抗剂。

MRS4654 是一种新型的高效 P2Y14 受体拮抗剂，具有15 nM 的半最大抑制浓度 (IC50)。

MRS1220 是一种高效、选择性的人 A3 腺苷受体 (hA3AR) 拮抗剂，Ki 为 0.59 nM，可用于中枢神经系统疾病的研究。MRS1220 在体内还减少了胶质母细胞瘤的肿瘤大小和血管形成。

antagonist for the human adenosine A3 receptor

competitive antagonist at P2Y1 receptors

P2Y13 receptor antagonist

P2X1 receptor potentiator

Selective, high affinity competitive antagonist of the P2Y1 receptor

Highly potent, selective P2Y1 receptor agonist

Highly potent and selective antagonist of the platelet P2Y1 receptor

P2Y14 receptor agonist

MRS 2693 trisodium salt is a P2Y6 agonist.

MRS 2768 tetrasodium salt is a P2Y2 agonist.

MRS2500 is a highly potent and selective platelet P2Y1 receptor antagonist.

MRS4458 is an effective inhibitor of the P2Y14 Receptor.

MRS4478 is an effective inhibitor of the P2Y14 Receptor.