规格

价格

库存

数量

1 mg

¥ 328

现货

5 mg

¥ 828

现货

10 mg

¥ 1,320

现货

25 mg

¥ 2,880

现货

50 mg

¥ 4,330

现货

100 mg

¥ 6,180

现货

200 mg

¥ 8,490

现货

1 mL x 10 mM (in DMSO)

¥ 768

现货

生物活性

产品描述	BAY-4931 is a powerful, covalent, and selective inverse-agonist of PPARγ, exhibiting an IC50 value of 0.17 nM.
靶点活性	UM-UC-9 cells:3.4 nM, PPARγ(RT112-FABP4-NLucP cellular):0.17 nM, PPARγ (mouse):0.14 nM, PPARγ (human):0.40 nM
体外活性	通过RP-HPLC和LC-MS对培养提取物的分级显示，含有Questin的样本对人类A549肺细胞系具有毒性。[1]

化学信息

分子量	421.83
分子式	C₂₂H₁₆ClN₃O₄
CAS No.	423150-91-8
Smiles	N(C(=O)C1=CC(N(=O)=O)=CC=C1Cl)C=2C=C3C(OC(=N3)C4=CC=C(CC)C=C4)=CC2
密度	no data available

储存&溶解度

存储

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

溶解度信息

DMSO: 112.5 mg/mL (266.7 mM), Sonication and heating to 70℃ are recommended.

溶液配制表

DMSO