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TargetMol | Compound Library

神经保护化合物库现货

Neuroprotective Compound Library

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产品编号 L2640

神经保护(Neuroprotection)是指通过各种机制和手段来防止神经元受到损伤或促进神经元的修复,从而保护神经系统功能的过程。这一领域的研究主要集中在防止神经元凋亡、减少炎症反应、减少氧化应激和促进神经再生等方面。神经保护在许多神经退行性疾病(如阿尔茨海默病、帕金森病、多发性硬化症)以及急性神经损伤(如中风和脊髓损伤)中具有重要意义。研究揭示了多个关键靶点,如抗氧化,神经营养因子,钙离子通道等在预防神经元损伤、促进神经再生以及对抗神经退行性疾病方面展现出潜力。
TargetMol神经保护化合物库收集了1120种具有神经保护活性及潜在的神经保护活性化合物,可用于神经保护相关的药物研发,神经保护相关机制探索。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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产品编号 L2640

神经保护化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 1120种神经保护相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 靶点包括BDNF、Calcium Channel、Sodium Channel、NMDAR/TRPM4等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

Calcium Channel
Sodium Channel
Apoptosis
Wnt/beta-catenin
Potassium Channel
NO Synthase
iGluR
Endogenous Metabolite
Autophagy
GSK-3
GABA Receptor
NMDAR
GluR
NF-κB
AMPK
Reactive Oxygen Species
Antibacterial
COX
AChR
Akt
Parasite
CDK
5-HT Receptor
ERK
Cytochromes P450
TNF
NOS
Antioxidant
Caspase
PARP
Dopamine Receptor
Cholinesterase (ChE)
Beta Amyloid
PDE
Interleukin
p38 MAPK
PI3K
IL Receptor
Histamine Receptor
Mitophagy
PPAR
TRP/TRPV Channel
Adrenergic Receptor
Prostaglandin Receptor
ROS
Antibiotic
Monoamine Oxidase
Adenosine Receptor
MAO
Bcl-2 Family
Influenza Virus
HIF/HIF Prolyl-Hydroxylase
JNK
PKC
mTOR
EGFR
Tyrosinase
Ferroptosis
Virus Protease
Glucosidase
MMP
DNA/RNA Synthesis
STAT
Anti-infection
HIV Protease
Na+/Ca2+ Exchanger
Phosphatase
PKA
HSV
TGF-beta/Smad
MAPK
Nrf2
S6 Kinase
Microtubule Associated
GPCR
Carbonic Anhydrase
Src
RAAS
Mitochondrial Metabolism
Casein Kinase
HDAC
MEK
Ras
Sigma receptor
ATPase
Antifungal
Serotonin Transporter
Serine/threonin kinase
VEGFR
Glucocorticoid Receptor
Gamma-secretase
Drug Metabolite
Antifection
Molecular Glues
JAK
Aurora Kinase
Lipoxygenase
Epigenetic Reader Domain
Lipid
P-gp
Porcupine
SARS-CoV
transporter
Phospholipase
NOD
Chloride channel
Estrogen/progestogen Receptor
DYRK
Estrogen Receptor/ERR
Serine Protease
E1/E2/E3 Enzyme
LDL
Opioid Receptor
PTEN
Chk
Norepinephrine
CaMK
Beta-Secretase
PGE Synthase
Antiviral
TLR
Trk receptor
Sirtuin
Pyroptosis
Cannabinoid Receptor
MDM-2/p53
FLT
HMG-CoA Reductase
Imidazoline Receptor
S1P Receptor
Proteasome
HCV Protease
Integrin
Arginase
LPL Receptor
Reductase
BACE
PERK
Cysteine Protease
Leukotriene Receptor
ROCK
NR4A
Amylase
Aryl Hydrocarbon Receptor
Immunology/Inflammation related
Topoisomerase
Bcr-Abl
P2X Receptor
Monoamine Transporter
Guanylate cyclase
Somatostatin
Xanthine Oxidase
cAMP
IGF-1R
ATP Citrate Lyase
LRRK2
RSV
IκB/IKK
PDK
HIF
FGFR
ROS Kinase
AhR
p53
FOXO3
PGK1
Thyroid hormone receptor(THR)
Proton pump
Adenylyl Cyclase
DHFR
Piezo Channel
Amino Acids and Derivatives
YAP
Dehydrogenase
c-Met/HGFR
LTR
Arrestin
gp120/CD4
GTPase
Progesterone Receptor
OCT
CaSR
MRP
HBV
Tyrosine Kinases
Cholecystokinin Receptor
ASCT
Cell Cycle Arrest
Nucleoside Antimetabolite/Analog
Liver X Receptor
Glucokinase
NAMPT
Glutaminase
IDO
CSF-1R
Prolyl Endopeptidase (PREP)
Myosin
UGT
Raf
DNA gyrase
HCN Channel
DPP-4
Fatty Acid Synthase
PDGFR
Stearoyl-CoA Desaturase (SCD)
CXCR
OX Receptor
Indoleamine 2,3-Dioxygenase (IDO)
Androgen Receptor
Telomerase
SGLT
OXPHOS
Survivin
HSP
Ephrin Receptor
Histone Acetyltransferase
Methionine Adenosyltransferase (MAT)
Hippo pathway
GST
Acetyl-CoA Carboxylase
FKBP
Retinoid Receptor
Kras
c-Fms
ribosome
Adenosine Deaminase
DAPK
NADPH-oxidase
DNA Methyltransferase
TAM Receptor
NOD-like Receptor (NLR)
Glyoxalase
PD-1/PD-L1
Sodium-dependent phosphate transporter

Keywords