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Phage-derived 12/1 peptide通过靶向MDM2和MDMX破坏 MDM2-p53 和 MDMX-p53 相互作用,发挥抗肿瘤活性,IC50为0.15和1.25 μM。

Phage-derived 12/1 peptide通过靶向MDM2和MDMX破坏 MDM2-p53 和 MDMX-p53 相互作用,发挥抗肿瘤活性,IC50为0.15和1.25 μM。
| 规格 | 价格 | 库存 | 数量 |
|---|---|---|---|
| 10 mg | 待询 | 待询 | |
| 50 mg | 待询 | 待询 |
Phage-derived 12/1 peptide 相关产品
| 产品描述 | Phage-derived 12/1 peptide demonstrates antitumor activity by targeting MDM2 and MDMX, thereby disrupting the MDM2-p53 and MDMX-p53 interactions, with IC50 values of 0.15 and 1.25 μM, respectively [1]. |
| 分子量 | 1558.78 |
| 分子式 | C71H99N17O19S2 |
| CAS No. | 186180-20-1 |
| Sequence | Met-Pro-Arg-Phe-Met-Asp-Tyr-Trp-Glu-Gly-Leu-Asn |
| Sequence Short | MPRFMDYWEGLN |
| 存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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