A2B receptor antagonist 1

Name: A2B receptor antagonist 1
Brand: TargetMol
SKU: T10058
Price: 3730 CNY
Availability: InStock
Rating: 5 (10 reviews)

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纯度: 99.53%

货号 T10058Cas号 531506-36-2

A2B receptor antagonist 1 是一个有效的 A2B 腺苷受体 (A2B adenosine receptor) 拮抗剂。

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A2B receptor antagonist 1

一键复制产品信息

很棒

纯度: 99.53%

货号 T10058Cas号 531506-36-2

A2B receptor antagonist 1 是一个有效的 A2B 腺苷受体 (A2B adenosine receptor) 拮抗剂。

规格	价格	库存
1 mg	¥ 3,730	现货
5 mg	¥ 7,380	现货
10 mg	¥ 9,870	现货
25 mg	¥ 14,800	现货
50 mg	¥ 19,800	现货
100 mg	¥ 27,300	现货
1 mL x 10 mM (in DMSO)	¥ 8,460	现货

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COA HNMR LCMS 产品操作手册

产品介绍

A2B receptor antagonist 1 AI Summary

A2B receptor antagonist 1 exhibits significant bioactivity associated with adenosine receptors, prominently showing high affinity for the adenosine A2b receptor with a Ki of 11.0 nM. It also demonstrates moderate affinity for the adenosine A3 receptor with a Ki of 76.0 nM and lower affinity for the adenosine A2a receptor with a Ki of 290.0 nM. Additionally, A2B receptor antagonist 1 exhibits selectivity for the A2b receptor over the A1 receptor with a ratio Ki of 7.0, over the A2a receptor with a ratio Ki of 26.0, and over the A3 receptor with a ratio Ki of 15.0. These affinities and selectivities highlight its potential as a targeted biological tool in studying adenosine receptor functions..

Note: Summary generated by AI. Data source: ChEMBL

生物活性

产品描述	A2B receptor antagonist 1 (EXAMPLE 9B) is a potent A2B adenosine receptor antagonist.

化学信息

分子量	392.45
分子式	C₂₁H₂₄N₆O₂
CAS No.	531506-36-2
Smiles	C(CC)N1C2=C(NC(=N2)C3=CN(CC4=CC=CC=C4)N=C3)C(=O)N(CCC)C1=O
密度	1.32 g/cm3 (Predicted)

储存&溶解度

存储

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

溶解度信息

DMSO: 15.47 mg/mL (39.42 mM), Sonication is recommended.

溶液配制表

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.5481 mL	12.7405 mL	25.4810 mL	127.4048 mL
5 mM	0.5096 mL	2.5481 mL	5.0962 mL	25.4810 mL
10 mM	0.2548 mL	1.2740 mL	2.5481 mL	12.7405 mL
20 mM	0.1274 mL	0.6370 mL	1.2740 mL	6.3702 mL