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MLS0315771 是来源于磷酸甘露糖异构酶的竞争性抑制剂, 其 IC50值为~1 μM,Ki=为 1.4 μM。
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MLS0315771 是来源于磷酸甘露糖异构酶的竞争性抑制剂, 其 IC50值为~1 μM,Ki=为 1.4 μM。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
1 mg | ¥ 478 | In stock | |
5 mg | ¥ 1,160 | In stock | |
10 mg | ¥ 1,730 | In stock | |
25 mg | ¥ 3,230 | In stock | |
50 mg | ¥ 4,320 | In stock | |
100 mg | ¥ 5,730 | In stock | |
1 mL x 10 mM (in DMSO) | ¥ 1,280 | In stock |
产品描述 | MLS0315771 is an effective and biologically active competitive phosphomannose isomerase (MPI) inhibitor (IC50: ~1 μM and a Ki: 1.4 μM). |
靶点活性 | MPI:1 μM (IC50) |
体外活性 | MLS0315771 is toxic to the zebrafish embryos above 2 μM. MLS0315771 toxicity at higher concentrations is an off-target effect. MLS0315771 enhances mannose flux toward glycosylation. It ~50% of embryos appeared sick within 20 min at 8-10 μM, and most of them die by 30-60 min. |
分子量 | 273.33 |
分子式 | C15H12FNOS |
CAS No. | 727664-91-7 |
Smiles | Cc1ccc(C)c(c1)-n1sc2cc(F)ccc2c1=O |
密度 | no data available |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||
溶解度信息 | DMSO: 11 mg/mL (40.24 mM), Sonication is recommended. ![]() | |||||||||||||||||||||||||
溶液配制表 | ||||||||||||||||||||||||||
DMSO
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以上为“体内实验配液计算器”的使用方法举例,并不是具体某个化合物的推荐配制方式,请根据您的实验动物和给药方式选择适当的溶解方案。
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