vardenafil

Vardenafil (Vivanza) 是选择性、高效的、具有口服活性的磷酸二酯酶5抑制剂，IC50=0.7 nM。它能够非竞争性地抑制环磷酸鸟苷水解，从而提高 cGMP 水平。它对 PDE1 (180 nM)，PDE6 (11 nM)，PDE2，PDE3，PDE4 (>1000 nM) 具有选择性。它可用于研究勃起功能障碍。

Vardenafil hydrochloride trihydrate (BAY38-9456) 是一种新型 PDE 抑制剂，对 PDE5 和 PDE1 的 IC50 分别为 0.7 和 180 nM。

Vardenafil hydrochloride 是口服具有活性的、高效的、选择性的磷酸二酯酶 5抑制剂。它对 PDE1 (180 nM)，PDE6 (11 nM)，PDE2，PDE3，PDE4 (>1000 nM) 具有选择性。它能够非竞争性地抑制环磷酸鸟苷水解，提高 cGMP 水平。它可用于勃起功能障碍的研究。

Vardenafil dihydrochloride (Levitra) 是一种新型 PDE 抑制剂，对 PDE5 和 PDE1 的 IC50 分别为 0.7 和 180 nM。

N-Desethyl vardenafil is a metabolite of vardenafil , a phosphodiesterase 5 inhibitor, that is formed by the action of cytochrome P450 (CYP)3A4 and CYP3A5.

Vardenafil oxopiperazine is an inhibitor of phosphodiesterase-5.

N-Desethyl-N-methyl Vardenafil, a potential impurity in commercial vardenafil preparations, functions as a phosphodiesterase 5 (PDE5) inhibitor, similar to its parent compound. With an IC50 value of 2 nM, it exhibits potent inhibitory activity against PDE5.

N-Desethyl Vardenafil (Standard) is the standard substance of N-Desethyl Vardenafil, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. N-Desethyl vardenafil is a metabolite of vardenafil , a phosphodiesterase 5 inhibitor, that is formed by the action of cytochrome P450 (CYP)3A4 and CYP3A5.

Vardenafil-d5 是 Vardenafil 的氘代化合物。Vardenafil 的 CAS 号为 224785-90-4。Vardenafil 是选择性、高效的、具有口服活性的磷酸二酯酶5抑制剂，IC50=0.7 nM。它能够非竞争性地抑制环磷酸鸟苷水解，从而提高 cGMP 水平。它对 PDE1 (180 nM)，PDE6 (11 nM)，PDE2，PDE3，PDE4 (>1000 nM) 具有选择性。它可用于研究勃起功能障碍。

N-Desethyl-N-Methyl Vardenafil (Standard) is the standard substance of N-Desethyl-N-Methyl Vardenafil, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. N-Desethyl-N-methyl Vardenafil, a potential impurity in commercial vardenafil preparations, functions as a phosphodiesterase 5 (PDE5) inhibitor, similar to its parent compound. With an IC50 value of 2 nM, it exhibits potent inhibitory activity against PDE5.

Vardenafil (Standard) 是 Vardenafil 的标准品，适用于定量分析、质量控制及生化实验等相关研究。Vardenafil (Vivanza) 是选择性、高效的、具有口服活性的磷酸二酯酶5抑制剂，IC50=0.7 nM。它能够非竞争性地抑制环磷酸鸟苷水解，从而提高 cGMP 水平。它对 PDE1 (180 nM)，PDE6 (11 nM)，PDE2，PDE3，PDE4 (>1000 nM) 具有选择性。它可用于研究勃起功能障碍。

Vardenafil hydrochloride (Standard) 是 Vardenafil hydrochloride 的标准品，适用于定量分析、质量控制及生化实验等相关研究。Vardenafil hydrochloride 是口服具有活性的、高效的、选择性的磷酸二酯酶 5抑制剂。它对 PDE1 (180 nM)，PDE6 (11 nM)，PDE2，PDE3，PDE4 (>1000 nM) 具有选择性。它能够非竞争性地抑制环磷酸鸟苷水解，提高 cGMP 水平。它可用于勃起功能障碍的研究。

Vardenafil Oxopiperazine (Standard) is the standard substance of Vardenafil Oxopiperazine, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Vardenafil oxopiperazine is an inhibitor of phosphodiesterase-5.

Acetylvardenafil 是一种新型的Vardenafil类似物，其结构中的磺酰基被乙酰基取代。作为一种PDE-5抑制剂，Acetylvardenafil 可用于研究勃起功能障碍 (ED)。

Thiovardenafil is the thiol analogue of the PDE 5 inhibitor Vardenafil.