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Kynurenic acid sodium是一种内源性色氨酸代谢物,作为靶向离子型谷氨酸受体(NMDA)、其他谷氨酸受体及α7烟碱型乙酰胆碱受体的广谱拮抗剂,同时还是G蛋白偶联受体GPR35/CXCR8的强效激动剂。
Kynurenic acid sodium是一种内源性色氨酸代谢物,作为靶向离子型谷氨酸受体(NMDA)、其他谷氨酸受体及α7烟碱型乙酰胆碱受体的广谱拮抗剂,同时还是G蛋白偶联受体GPR35/CXCR8的强效激动剂。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
25 mg | ¥ 198 | In stock | |
50 mg | ¥ 290 | In stock | |
1 mL x 10 mM (in DMSO) | ¥ 455 | In stock |
Kynurenic acid sodium 相关产品
产品描述 | Kynurenic acid sodium salt is an endogenous tryptophan metabolite that acts as a broad-spectrum antagonist targeting ionotropic glutamate receptors (NMDA), other glutamate receptors, and the α7 nicotinic acetylcholine receptor, while also functioning as a potent agonist for the G-protein coupled receptor GPR35/CXCR8. |
体外活性 | 方法:Kynurenic acid sodium (1-100μM,24-48小时)处理角膜上皮细胞和结膜上皮细胞,MTT法测定细胞活力。 |
别名 | 犬尿喹啉酸钠盐, Kynurenic acid sodium salt |
分子量 | 211.15 |
分子式 | C10H6NNaO3 |
CAS No. | 2439-02-3 |
Smiles | O=C(C1=CC(O)=C2C=CC=CC2=N1)[O-].[Na+] |
密度 | no data available |
存储 | keep away from moisture,store under nitrogen,store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. | |||||||||||||||||||||||||||||||||||
溶解度信息 | H2O: < 0.1 mg/mL (insoluble) DMSO: 40 mg/mL (189.44 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
溶液配制表 | ||||||||||||||||||||||||||||||||||||
DMSO
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以上为“体内实验配液计算器”的使用方法举例,并不是具体某个化合物的推荐配制方式,请根据您的实验动物和给药方式选择适当的溶解方案。
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