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TargetMol | Compound Library

人代谢物化合物库现货

Human Metabolite Library
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货号 L2570

人代谢物包括内源性代谢物和外源性代谢物;内源性代谢物,顾名思义,就是人体内产生和发现的一些代谢产物,如柠檬酸循环的任何中间代谢物,这些代谢物参与机体重要的生理过程,可作为潜在的药物先导物。外源性代谢物不在机体内产生与发现,来源于外界,包括药物、毒素和食品添加剂等,研究外源性代谢物在人体内如何发生代谢,有助于加快药物发现和毒理学的研究。在药物发现中,了解药物的代谢物有助于对药物作用机理的研究。
TargetMol 人代谢物化合物库收集了6030 种内源性和外源性代谢物,包括羧酸、氨基酸、生物胺、核苷酸、维生素、单糖、双糖、脂类、碳水化合物等不同种类代谢物。

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货号 L2570

人代谢物化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 6030种人代谢物的独特集合,用于高通量、高内涵筛选;
  • 研究人体代谢疾病、探索癌症发病机制和寻找新药的有效工具;
  • 部分化合物已上市或进入临床,具有生物安全保障和良好的生物活性;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

Endogenous Metabolite
Apoptosis
Antibacterial
Autophagy
Antibiotic
ROS
NF-κB
Antifungal
Parasite
COX
DNA/RNA Synthesis
Reactive Oxygen Species
5-HT Receptor
Cytochromes P450
Adrenergic Receptor
HIV Protease
Akt
Interleukin
Antioxidant
Calcium Channel
TNF
AChR
Caspase
p38 MAPK
Drug Metabolite
Potassium Channel
Dopamine Receptor
PPAR
NO Synthase
GABA Receptor
Histamine Receptor
ERK
PI3K
Influenza Virus
Virus Protease
Sodium Channel
Nucleoside Antimetabolite/Analog
PDE
Ferroptosis
Nrf2
Cholinesterase (ChE)
Prostaglandin Receptor
SARS-CoV
STAT
Estrogen/progestogen Receptor
Glucocorticoid Receptor
Bcl-2 Family
MMP
Dehydrogenase
Estrogen Receptor/ERR
AMPK
iGluR
JNK
Microtubule Associated
VEGFR
Topoisomerase
Tyrosinase
HSV
EGFR
mTOR
Amino Acids and Derivatives
TRP/TRPV Channel
Phosphatase
RAAS
Mitophagy
IL Receptor
PKC
Beta Amyloid
Adenosine Receptor
Mitochondrial Metabolism
Reverse Transcriptase
HCV Protease
Wnt/beta-catenin
ATPase
TLR
PARP
Lipoxygenase
P-gp
HDAC
Anti-infection
NMDAR
Androgen Receptor
JAK
Monoamine Oxidase
Reductase
Glucosidase
Carbonic Anhydrase
HBV
CDK
Antiviral
HIF/HIF Prolyl-Hydroxylase
Proteasome
Antifection
Opioid Receptor
PDGFR
glycosidase
Progesterone Receptor
Angiotensin-converting Enzyme (ACE)
GPCR
GluR
TGF-beta/Smad
DNA Alkylator/Crosslinker
HSP
c-Kit
Serotonin Transporter
MAO
GSK-3
Phospholipase
Chloride channel
Transferase
Src
FGFR
MDM-2/p53
Ras
PKA
FLT
Aryl Hydrocarbon Receptor
Glutathione Peroxidase
HMG-CoA Reductase
Thrombin
Immunology/Inflammation related
Norepinephrine
Sirtuin
NOD-like Receptor (NLR)
NOS
Gamma-secretase
Xanthine Oxidase
IGF-1R
ribosome
Proton pump
c-Met/HGFR
MRP
Fatty Acid Synthase
IκB/IKK
MEK
Cannabinoid Receptor
Thyroid hormone receptor(THR)
Integrin
NADPH
PERK
Tyrosine Kinases
Serine Protease
DPP-4
CaMK
Retinoid Receptor
FXR
Raf
DNA Alkylation
Epigenetic Reader Domain
DHFR
Melatonin Receptor
Hedgehog/Smoothened
Lipid
MAPK
transporter
Aromatase
HIF
Neurokinin receptor
p53
Antifolate
Cysteine Protease
Leukotriene Receptor
UGT
Bcr-Abl
DNA
DNA Methyltransferase
Factor Xa
E1/E2/E3 Enzyme
CXCR
Trk receptor
GPCR19
Hydroxylase
Platelet aggregation
NOD
ROS Kinase
AhR
CFTR
ADC Cytotoxin
P2Y Receptor
IFNAR
Necroptosis
ABC Transporter
Molecular Glues
CCR
SGLT
Acyltransferase
Free radical scavengers
Pyroptosis
FAK
Liposome
Histone Methyltransferase
GNRH Receptor
Serine/threonin kinase
P2X Receptor
PGE Synthase
c-RET
BACE
LDLR
Amylase
PAFR
MT Receptor
Monoamine Transporter
PROTAC Linker
Endothelin Receptor
OXPHOS
OAT
ALK
GST
PD-1/PD-L1
S1P Receptor
Vitamin
Arginase
LPL Receptor
LTR
Histone Demethylase
Lipase
CaSR
Cholecystokinin Receptor
Photosensitizer
Liver X Receptor
IDO
LDL
Phosphorylase
GlyT
Guanylate cyclase
Smo
Indoleamine 2,3-Dioxygenase (IDO)
Telomerase
ATP Citrate Lyase
Aminopeptidase
Casein Kinase
Ligand for E3 Ligase
Adenosine Deaminase
c-Myc
ATG
Cell Cycle Arrest
Glucokinase
IAP
Annexin A
DNA gyrase
FAAH
Bradykinin Receptor
Aurora Kinase
Survivin
STING
Histone Acetyltransferase
PAI-1
Neprilysin
ATM/ATR
FKBP
PLK
Complement System
Syk
Sigma receptor
TAM Receptor
Imidazoline Receptor
HER
MicroRNA
Monocarboxylate transporter
MTP
YAP
CETP
ROCK
IRE1
Adiponectin Receptor
Na-K-Cl cotransporter
HCAR
PTEN
Epoxide Hydrolase
Thrombopoietin Receptor
DUB
BCRP
Beta-Secretase
Ephrin Receptor
Decarboxylase
RSV
c-Fms
FOXO
S6 Kinase
ROR
DNA-PK
Na+/Ca2+ Exchanger
Cell wall
Tie-2
gp120/CD4
Glutaminase
RANKL/RANK
CSF-1R
Prolyl Endopeptidase (PREP)
RIP kinase
Isocitrate Dehydrogenase (IDH)
Vasopressin Receptor
Chk
cAMP
Mucin
GPX
Protease
Melanocortin Receptor
Oxytocin Receptor
GHSR
CGRP Receptor
ADC Linker
Kras
Apelin receptor
Advanced Glycation End Products
Mdm2
Taste receptor
Adenylyl Cyclase
CAT
NPC1L1
ASBT
CYP19A1
CRM1
MyD88
Ligands for Target Protein for PROTAC
Aconitase
MIF
VDA
Galectin
Bcl-6
Rho
Neurotensin Receptor
NR4A
Glucagon Receptor
Hexokinase
Bombesin Receptor
PAK
Stearoyl-CoA Desaturase (SCD)
OX Receptor
Wee1
Glutathione reductase
LRRK2
cGAS
GluCls
Acetyl-CoA Carboxylase
p62
Carboxypeptidase
CRISPR/Cas9
PDK
Cuproptosis
Gap Junction Protein
NADPH-oxidase
IRAK
Protease-activated Receptor
BTK
IKZF
Transaminase
stilbene oxidase
Hydrogenase
RAR/RXR
CD38
GDNF
Dynamin
NEDD8
DYRK
TOPK
N-Acetylglucosaminyltransferase
ASCT
Hck
NAMPT
Myosin
Photosystem (PS)
FLAP
MTH1
Fas/FasL
Anion Exchanger
HCN Channel
MAGL
ACK1
Somatostatin
PAD
KSP
Cadherin
Transketolase
Orphan Receptor
Huntingtin
PSMA
Urea Transporter
CPT
ASK
hCE
CRFR
LPA Receptor
Aquaporin
DAPK
Tight Junction Protein
p97
Enteropeptidase (EP)
MLK
Kinesin
PKM
Ferroportin
Drug-Linker Conjugates for ADC
PGC-1α

Keywords