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TargetMol | Compound Library

人代谢物化合物库现货

Human Metabolite Library
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货号 L2570

人代谢物包括内源性代谢物和外源性代谢物;内源性代谢物,顾名思义,就是人体内产生和发现的一些代谢产物,如柠檬酸循环的任何中间代谢物,这些代谢物参与机体重要的生理过程,可作为潜在的药物先导物。外源性代谢物不在机体内产生与发现,来源于外界,包括药物、毒素和食品添加剂等,研究外源性代谢物在人体内如何发生代谢,有助于加快药物发现和毒理学的研究。在药物发现中,了解药物的代谢物有助于对药物作用机理的研究。
TargetMol 人代谢物化合物库收集了6030 种内源性和外源性代谢物,包括羧酸、氨基酸、生物胺、核苷酸、维生素、单糖、双糖、脂类、碳水化合物等不同种类代谢物。

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货号 L2570

人代谢物化合物库

规格

  • 1 mg
  • 10 μL x 10 mM (in DMSO)
  • 20 μL x 10 mM (in DMSO)
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 6030种人代谢物的独特集合,用于高通量、高内涵筛选;
  • 研究人体代谢疾病、探索癌症发病机制和寻找新药的有效工具;
  • 部分化合物已上市或进入临床,具有生物安全保障和良好的生物活性;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

Endogenous Metabolite
Apoptosis
Antibacterial
Autophagy
Antibiotic
ROS
NF-κB
Antifungal
Parasite
COX
DNA/RNA Synthesis
Reactive Oxygen Species
5-HT Receptor
Cytochromes P450
Adrenergic Receptor
HIV Protease
Interleukin
Akt
Antioxidant
Calcium Channel
TNF
AChR
Caspase
Drug Metabolite
Potassium Channel
p38 MAPK
PPAR
Dopamine Receptor
NO Synthase
Histamine Receptor
GABA Receptor
ERK
Influenza Virus
PI3K
Virus Protease
Sodium Channel
PDE
Ferroptosis
Nucleoside Antimetabolite/Analog
Nrf2
Cholinesterase (ChE)
Glucocorticoid Receptor
STAT
Estrogen Receptor/ERR
SARS-CoV
Estrogen/progestogen Receptor
Dehydrogenase
Prostaglandin Receptor
MMP
Bcl-2 Family
AMPK
JNK
iGluR
Topoisomerase
Microtubule Associated
VEGFR
Tyrosinase
HSV
EGFR
Amino Acids and Derivatives
mTOR
TRP/TRPV Channel
Phosphatase
IL Receptor
RAAS
Mitophagy
Beta Amyloid
Adenosine Receptor
PKC
Mitochondrial Metabolism
Reverse Transcriptase
HCV Protease
TLR
Wnt/beta-catenin
PARP
Lipoxygenase
HDAC
ATPase
P-gp
Anti-infection
NMDAR
JAK
Monoamine Oxidase
Androgen Receptor
HIF/HIF Prolyl-Hydroxylase
Glucosidase
Carbonic Anhydrase
HBV
CDK
Antifection
Antiviral
Reductase
Opioid Receptor
glycosidase
Proteasome
PDGFR
Angiotensin-converting Enzyme (ACE)
GluR
GPCR
Progesterone Receptor
TGF-beta/Smad
HSP
c-Kit
DNA Alkylator/Crosslinker
Serotonin Transporter
MAO
GSK-3
Phospholipase
Transferase
Src
FGFR
MDM-2/p53
FLT
Ras
Chloride channel
PKA
Aryl Hydrocarbon Receptor
NOS
Glutathione Peroxidase
HMG-CoA Reductase
Thrombin
IGF-1R
Norepinephrine
NOD-like Receptor (NLR)
Immunology/Inflammation related
Gamma-secretase
Sirtuin
MEK
Thyroid hormone receptor(THR)
Proton pump
c-Met/HGFR
MRP
Serine Protease
Xanthine Oxidase
IκB/IKK
ribosome
Integrin
PERK
Tyrosine Kinases
Fatty Acid Synthase
CaMK
Retinoid Receptor
HIF
Cannabinoid Receptor
NADPH
FXR
Raf
DPP-4
DNA Alkylation
Epigenetic Reader Domain
MAPK
DHFR
Leukotriene Receptor
Hedgehog/Smoothened
Lipid
transporter
Aromatase
Melatonin Receptor
Antifolate
Cysteine Protease
UGT
Bcr-Abl
DNA
Neurokinin receptor
NOD
p53
ADC Cytotoxin
CXCR
Trk receptor
GPCR19
Hydroxylase
DNA Methyltransferase
ROS Kinase
AhR
CFTR
Histone Methyltransferase
P2Y Receptor
IFNAR
Necroptosis
Factor Xa
E1/E2/E3 Enzyme
ABC Transporter
CCR
SGLT
PGE Synthase
Acyltransferase
Free radical scavengers
Pyroptosis
c-RET
Platelet aggregation
Liposome
FAK
GNRH Receptor
Serine/threonin kinase
P2X Receptor
PROTAC Linker
ALK
GST
LTR
LDLR
Amylase
PAFR
MT Receptor
Monoamine Transporter
Molecular Glues
Endothelin Receptor
OXPHOS
OAT
Sigma receptor
PD-1/PD-L1
S1P Receptor
Vitamin
Arginase
LPL Receptor
BACE
Histone Demethylase
Lipase
Photosensitizer
Liver X Receptor
IDO
Phosphorylase
GlyT
Guanylate cyclase
Smo
Ligands for E3 Ligase
Indoleamine 2,3-Dioxygenase (IDO)
Telomerase
ATP Citrate Lyase
Aminopeptidase
Casein Kinase
Adenosine Deaminase
c-Myc
CaSR
Cholecystokinin Receptor
ATG
Cell Cycle Arrest
Glucokinase
IAP
Adenylate cyclase
Annexin A
LDL
DNA gyrase
FAAH
Bradykinin Receptor
Aurora Kinase
Survivin
STING
Histone Acetyltransferase
PAI-1
ATM/ATR
FKBP
PLK
Complement System
Syk
TAM Receptor
Imidazoline Receptor
HER
MicroRNA
Monocarboxylate transporter
MTP
CETP
ROCK
IRE1
Adiponectin Receptor
Na-K-Cl cotransporter
HCAR
PTEN
Epoxide Hydrolase
Thrombopoietin Receptor
DUB
BCRP
Beta-Secretase
Ephrin Receptor
Decarboxylase
RSV
Neprilysin
c-Fms
FOXO
S6 Kinase
NPC1L1
ROR
DNA-PK
YAP
Na+/Ca2+ Exchanger
gp120/CD4
Tie-2
Glutaminase
RANKL/RANK
CSF-1R
Prolyl Endopeptidase (PREP)
RIP kinase
Isocitrate Dehydrogenase (IDH)
Vasopressin Receptor
Chk
cAMP
Mucin
Carboxypeptidase
GPX
Melanocortin Receptor
Oxytocin Receptor
GHSR
CGRP Receptor
Gap Junction Protein
ADC Linker
Kras
Advanced Glycation End Products
Mdm2
Taste receptor
CAT
ASBT
CYP19A1
CRM1
MyD88
Ligands for Target Protein for PROTAC
Aconitase
Cell wall
MIF
VDA
Galectin
Bcl-6
Rho
NR4A
Glucagon Receptor
Hexokinase
PAK
Bombesin Receptor
Stearoyl-CoA Desaturase (SCD)
OX Receptor
Orphan receptor
Wee1
Glutathione reductase
LRRK2
cGAS
GluCls
CRFR
Acetyl-CoA Carboxylase
p62
Protease
CRISPR/Cas9
Cuproptosis
NADPH-oxidase
IRAK
Protease-activated Receptor
BTK
IKZF
Transaminase
Hydrogenase
stilbene oxidase
RAR/RXR
CD38
GDNF
Dynamin
NEDD8
DYRK
TOPK
N-Acetylglucosaminyltransferase
ASCT
Hck
Neurotensin Receptor
NAMPT
Myosin
Photosystem (PS)
FLAP
MTH1
Fas/FasL
Anion Exchanger
HCN Channel
MAGL
ACK1
Somatostatin
PAD
KSP
Cadherin
Transketolase
Huntingtin
PSMA
E3 Ligase Ligand-Linker Conjugates
Urea Transporter
CPT
ASK
hCE
LPA Receptor
PDK
Aquaporin
DAPK
APC/C
Tight Junction Protein
p97
Enteropeptidase (EP)
MLK
Kinesin
PKM
Ferroportin
Drug-Linker Conjugates for ADC
PGC-1α

Keywords