GV150013

Name: GV150013
Brand: TargetMol
SKU: T27503
Price: 1380 CNY
Availability: InStock
Rating: 5 (10 reviews)

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纯度: 99.93%

货号 T27503Cas号 167355-22-8

别名 GV-150013, GV 150013

GV150013是一种 cholecystokinin-2 (CCK2)受体拮抗剂。

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GV150013

一键复制产品信息

很棒

纯度: 99.93%

货号 T27503 别名 GV-150013, GV 150013Cas号 167355-22-8

GV150013是一种 cholecystokinin-2 (CCK2)受体拮抗剂。

规格	价格	库存
1 mg	¥ 1,380	现货
5 mg	¥ 3,330	现货
10 mg	¥ 4,670	现货
25 mg	¥ 6,900	现货
50 mg	¥ 9,360	现货
100 mg	¥ 12,300	现货
200 mg	¥ 16,800	现货
1 mL x 10 mM (in DMSO)	¥ 4,790	现货

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ee: 98.56%

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产品介绍

GV150013 AI Summary

GV150013 exhibits a high affinity for Cholecystokinin type B (CCK-B) receptors, with a Ki value of 0.955 nM, signifying its potent ability to displace tritiated CCK-8S bound on guinea pig brain CCK-B receptors. In contrast, it demonstrates a significantly lower affinity for Cholecystokinin type A (CCK-A) receptors, with a Ki value of 1122.02 nM in rat pancreas. The ratio of CCK-B to CCK-A receptor affinity is 1175.0, showing a pronounced preference for CCK-B receptors. Moreover, GV150013 displays notable anxiolytic activity in mice when administered orally, with an effective dose (ED50) in the black/white box test determined to be 0.00005 mg/kg..

Note: Summary generated by AI. Data source: ChEMBL

生物活性

产品描述	GV150013 is an antagonist of cholecystokinin-2 (CCK2) receptor.
别名	GV-150013, GV 150013

化学信息

分子量	534.65
分子式	C₃₃H₃₄N₄O₃
CAS No.	167355-22-8
Smiles	C(C12CC3CC(C1)CC(C2)C3)N4C=5C(N(C(=O)[C@H](NC(NC6=CC=CC=C6)=O)C4=O)C7=CC=CC=C7)=CC=CC5
密度	1.34 g/cm3 (Predicted)

储存&溶解度

存储

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

溶解度信息

DMSO: 50 mg/mL (93.52 mM), Sonication is recommended.

溶液配制表

DMSO

	1mg	5mg	10mg	50mg
1 mM	1.8704 mL	9.3519 mL	18.7038 mL	93.5191 mL
5 mM	0.3741 mL	1.8704 mL	3.7408 mL	18.7038 mL
10 mM	0.1870 mL	0.9352 mL	1.8704 mL	9.3519 mL
20 mM	0.0935 mL	0.4676 mL	0.9352 mL	4.6760 mL
50 mM	0.0374 mL	0.1870 mL	0.3741 mL	1.8704 mL