Name: TLQP 21 acetate
Brand: TargetMol
SKU: TP2296L
Price: 1060 CNY
Availability: InStock
Rating: 5 (10 reviews)

规格

价格

库存

数量

1 mg

¥ 1,060

现货

5 mg

¥ 2,680

现货

10 mg

¥ 4,570

现货

25 mg

¥ 8,220

现货

50 mg

¥ 11,900

现货

100 mg

¥ 15,900

现货

生物活性

产品描述	TLQP 21 acetate is a potent agonist of G-protein-coupled receptor complement-3a receptor 1 (C3aR1). The EC50 values are 10.3 μM for mouse and 68.8 μM for human. TLQP 21 acetate is a VGF-derived peptide with endocrine and extraendocrine properties.
靶点活性	C3aR1:10.3 μM(EC50,mouse), C3aR1:68.8 μM(EC50,human)
体外活性	TLQP 21 acetate 通过激活 C3aR1 导致细胞内 Ca2+ 的增加。TLQP 21 acetate (3 μM)诱导的收缩效果可达乙酰胆碱促进的相应收缩效果的约69%[1]。

化学信息

分子量	2492.8
分子式	C₁₀₉H₁₇₄N₄₀O₂₈
Smiles	CC(O)=O.N=C(N)NCCC[C@@H](C(O)=O)NC([C@H](C)NC([C@H]1N(C([C@H]2N(C([C@H](CC(C)C)NC([C@H](C)NC([C@H](CC3=CNC=N3)NC([C@H](CC4=CNC=N4)NC([C@H](CC5=CC=CC=C5)NC([C@H](CC6=CNC=N6)NC([C@H](CCCNC(N)=N)NC([C@H](CCCNC(N)=N)NC([C@H](CCCNC(N)=N)NC([C@H](CO)NC([C@H](CO)NC([C@H](C)NC([C@H]7N(C([C@H]8N(C([C@H](CCC(N)=O)NC([C@H](CC(C)C)NC([C@H]([C@H](O)C)N)=O)=O)=O)CCC8)=O)CCC7)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)CCC2)=O)CCC1)=O)=O
Sequence	Thr-Leu-Gln-Pro-Pro-Ala-Ser-Ser-Arg-Arg-Arg-His-Phe-His-His-Ala-Leu-Pro-Pro-Ala-Arg
Sequence Short	TLQPPASSRRRHFHHALPPAR

储存&溶解度

存储	store at low temperature,keep away from moisture \| Powder: -20°C for 3 years \| In solvent: -80°C for 1 year \| Shipping with blue ice/Shipping at ambient temperature.