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造血毒性小分子库

造血毒性小分子库

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产品编号 L3100 Hematopoietic Toxicity Compound Library
  库化合物信息   Excel SDF

TargetMol 造血毒性小分子库汇集了 104 种小分子化合物,它们对造血系统功能具有不同程度的毒性作用,包括骨髓抑制、中性粒细胞减少、白细胞减少、贫血和其他功能,在结构和机制上都具有代表性。所有的产品都是经过生物活性测试的,可以查到相关的文献报道。其中部分产品为已经上市的小分子药物,这些小分子化合物可以提供1mg,5mg 不等的包装,并且绝大部分产品可以提供后期的重复供应,为生物和药理科学家们的工作提供了有用的实验工具进行细胞诱导以及药理和毒理的相关研究。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
咨询化合物库
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产品描述

  • 104种生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 靶点包括HDAC、PPAR、DNA Alkylating、EGFR等;?
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L3100)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

Autophagy (33)
Apoptosis (32)
Antibacterial (20)
Antibiotic (20)
Endogenous Metabolite (13)
DNA/RNA Synthesis (11)
DNA Alkylator/Crosslinker (10)
Parasite (8)
Potassium Channel (7)
Microtubule Associated (7)
Mitophagy (7)
Antifungal (7)
HIV Protease (6)
COX (6)
Sodium Channel (6)
Adrenergic Receptor (5)
Nucleoside Antimetabolite/Analog (5)
DNA Alkylation (5)
Topoisomerase (5)
AChR (5)
c-Kit (4)
Dopamine Receptor (4)
5-HT Receptor (4)
Estrogen/progestogen Receptor (3)
Ferroptosis (3)
HDAC (3)
EGFR (3)
PDGFR (3)
PDE (3)
Reactive Oxygen Species (3)
Bcr-Abl (3)
Antifection (3)
Thyroid hormone receptor(THR) (3)
HSV (3)
P450 (2)
Phosphatase (2)
Reverse Transcriptase (2)
NF-κB (2)
MRP (2)
Thrombin (2)
VEGFR (2)
MAO (2)
Histamine Receptor (2)
GABA Receptor (2)
Calcium Channel (2)
CRISPR/Cas9 (2)
Dehydrogenase (2)
DNA (2)
Estrogen Receptor/ERR (2)
FLT (2)
Virus Protease (2)
HIF/HIF Prolyl-Hydroxylase (2)
GPR (1)
TAM Receptor (1)
Ras (1)
c-Met/HGFR (1)
CAT (1)
Rho (1)
ribosome (1)
iGluR (1)
Src (1)
STAT (1)
Telomerase (1)
Taste receptor (1)
RAAS (1)
Antifolate (1)
AMPK (1)
TNF (1)
Adenosine Receptor (1)
TRP/TRPV Channel (1)
Tyrosinase (1)
Tyrosine Kinases (1)
Adenosine deaminase (1)
Raf (1)
PPAR (1)
Proteasome (1)
DNA Methyltransferase (1)
Gamma-secretase (1)
NADPH-oxidase (1)
Mitochondrial Metabolism (1)
NMDAR (1)
Norepinephrine (1)
NOS (1)
HBV (1)
Opioid Receptor (1)
P2Y Receptor (1)
p53 (1)
Molecular Glues (1)
DNA gyrase (1)
Ligand for E3 Ligase (1)
IRE1 (1)
Influenza Virus (1)
Phospholipase (1)
Hydroxylase (1)
PKC (1)
Platelet aggregation (1)
Complement System (1)
PI3K (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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