tpa-023

TPA 023 是 GABAA α2 α3 亚型的特异性激动剂 (Ki = 0.19 - 0.41 nM)。

TPA-023B is an orally active and high-affinity agonist of the GABAA receptor α2 α3 subtype (Kis: 0.73 nM 2 nM) partial and an antagonist α1 subtype (Ki: 1.8 nM), has non-sedating anxiolytic-like properties.