k201

JTV-519 free base (K201 free base), recognized for its antiarrhythmic and cardioprotective properties, functions as a Ca2+-dependent blocker of sarcoplasmic reticulum Ca2+-stimulated ATPase (SERCA) and serves as a partial agonist of ryanodine receptors in striated muscle.

JTV-519 是一种 Ca2+ 依赖性阻滞剂，通过稳定兰尼碱受体来防止缺血性心脏和骨骼肌 (SkM) 中的肌质网异常 Ca(2+) 泄漏。

JTV-519 hemifumarate,Antiarrhythmic and cardioprotective properties. is a Ca2+-dependent blocker of sarcoplasmic reticulum Ca2+-stimulated ATPase (SERCA) and a partial agonist of ryanodine receptors in striated muscle.

GSK2018682 is a novel sphingosine-1-phosphate receptor 1 (s1p1) and 5 (s1p5) agonist.

GSK2018682 是 1-磷酸鞘氨醇受体S1P1和S1P5激动剂，pEC50值分别为 7.7 和 7.2，可用于多发性硬化的研究。

Dibenzosuberenol is a reactant involved in oxidation with tert-butylhydroperoxide in water for synthesis of carboxylic acids and ketones; Synthesis of tachykinin neurokinin-1 receptor antagonists; Pauson-Khand reaction mechanism studies; Mapping the active site of aziridination catalysts.

VK-2019是一种选择性EBNA1(爱泼斯坦-巴尔核抗原 1)抑制剂,具有口服活性,主要用于研究ebv相关癌症.

JTV-519 fumarate (K201 fumarate) 是 一种 SERCA 阻断剂和兰尼碱受体的部分激动剂，具有抗心律失常和心脏保护作用，可改善肌浆网钙渗漏，可用于研究焦虑症。