cckb receptor

Itriglumide (CR-2945) 是一种胆囊收缩素 （CCK）-2 受体拮抗剂，具有抗分泌和抗溃疡作用。

CCK-B Receptor Antagonist 2 is a potent and orally active antagonist of Gastrin CCK-B (IC50: 0.43 nM). It also inhibits gastrin CCK-A activity (IC50: 1.82 μM).

CCK-B Receptor Antagonist 1 is a cholecystokinin B (CCK-B) receptor agonist and has the potential of reducing the secretion of gastric acid.

PD 135158 is a CCK2 receptor antagonist.

PD-149164 is an agonist of the CCK-A receptor.

TP-680 is a antagonist of cholecystokininA receptor.

Selective CCK2 receptor antagonist

RP-72540 is a cholecystokinin B receptor antagonist. RP 72540 showed selectivity factors in express of 200 for CCKA versus CCKB receptors and also had high affinity for gastrin binding sites in the stomach. Administration of RP-72540 resulted in a dose-de

Pentagastrin (ICI-50123) 是一种选择性的胆囊收缩素 B(CCKB) 受体激动剂，IC50=11 nM。它能够增强胃粘膜对酸的防御机制，并保护胃粘膜免受损伤。