AC-178335 is a pure somatostatin (SRIF) antagonist with an affinity constant (Ki) of 172 +/- 12 nM. AC-178335 blocks SRIF inhibition of adenylate cyclase in vitro (IC50 = 5.1 +/- 1.4 microM). It induces GH release when given alone (50 micrograms intraveno
4,6-Pregnadien-6-Me-16-Methylene-17-Ol-3,20-Dione-D2 Ac (Standard) 是 4,6-Pregnadien-6-Me-16-Methylene-17-Ol-3,20-Dione-D2 Ac 的标准品,适用于定量分析、质量控制及生化实验等相关研究。