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Targets Recommended: Microtubule Associated

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Cat. No. Product Name Target Signaling Pathways
T12823 S516

Microtubule Associated Cytoskeletal Signaling
S516 is an active CKD-516 metabolite and is a potent inhibitor of tubulin polymerization(IC50 of 4.29 μM), has marked antitumor activity.
T13278 Valecobulin hydrochloride

CKD-516 hydrochloride

Microtubule Associated Cytoskeletal Signaling
Valecobulin hydrochloride (CKD-516 hydrochloride) 是 S516 的缬氨酸前体药和血管阻断剂。Valecobulin hydrochloride 对β-微管蛋白聚合有强效的抑制作用,对小鼠和人类的实体肿瘤具有显著的抗肿瘤活性。
T4327 Prexasertib dihydrochloride

LY2606368 (dihydrochloride),Prexasertib HCl,LY2606368

Apoptosis; Chk; S6 Kinase Apoptosis; Cell Cycle/Checkpoint; MAPK; PI3K/Akt/mTOR signaling
Prexasertib dihydrochloride (LY2606368) 是一种选择性的,ATP 竞争性的细胞周期检测点激酶 1 抑制剂,Ki 为 0.9 nM,IC50为 <1 nM。它抑制 CHK2(IC50=8 nM) 和 RSK1 (IC50=9 nM)。它引起双链 DNA 断裂和复制突变,导致细胞凋亡,有抗肿瘤活性。
T4310 Prexasertib

5-[[5-[2-(3-氨基丙氧基)-6-甲氧基苯基]-1H-吡唑-3-基]氨基]-2-吡嗪甲腈,LY2606368

Apoptosis; Chk Apoptosis; Cell Cycle/Checkpoint
Prexasertib (LY2606368) 是一种具有潜在抗肿瘤活性的检查点激酶 1 抑制剂。它可引起双链 DNA 断裂和复制突变,导致细胞凋亡。
T2477 UNBS5162

UNBS 5162,UNBS-5162

CXCR; Autophagy Autophagy; GPCR/G Protein; Immunology/Inflammation
UNBS5162 (UNBS-5162) 是一种新型萘酰亚胺,可降低实验性前列腺癌中 CXCL 趋化因子的表达。它是一种广谱趋化因子配体CXCL 拮抗剂,具有抗肿瘤活性。
T13278L Valecobulin

CKD-516

Others Others
Valecobulin is a potent β-tubulin polymerization inhibitor. Valecobulin is a valine prodrug of (S516) and an avascular disrupting compound.

化合物

S516
Cat.No: T12823
Synonym:
Target: Microtubule Associated
Valecobulin hydrochloride
Cat.No: T13278
Synonym: CKD-516 hydrochloride
Target: Microtubule Associated
Prexasertib dihydrochloride
Cat.No: T4327
Synonym: LY2606368 (dihydrochloride),Prexasertib HCl,LY2606368
Target: Apoptosis, Chk, S6 Kinase
Prexasertib
Cat.No: T4310
Synonym: 5-[[5-[2-(3-氨基丙氧基)-6-甲氧基苯基]-1H-吡唑-3-基]氨基]-2-吡嗪甲腈,LY2606368
Target: Apoptosis, Chk
UNBS5162
Cat.No: T2477
Synonym: UNBS 5162,UNBS-5162
Target: CXCR, Autophagy
Valecobulin
Cat.No: T13278L
Synonym: CKD-516
Target: Others
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