5-ht1b/1d

Almotriptan Malate (PNU180638) 是一种选择性 5-HT1B 1D 受体激动剂，用于治疗成人偏头痛发作。

Almotriptan (LAS 31416) 是一种用于研究偏头痛的5-HT1B 1D 受体激动剂。

GR 125743 是选择性的5-HT1B 1D 受体拮抗剂，与野生型的人 h5-HT1B 和 5-HT1D 结合的pKi 分别为 8.85 和 8.31，可用于帕金森病和心血管疾病的研究。

AR-A 2 is a selective 5-HT1B receptor antagonist, with a high affinity to guinea pig cortex 5HT1B 1D and recombinant guinea pig 5-HT1B receptors (Ki: 0.24 and 0.47 nM) and with 10-fold lower affinity to guinea pig 5-HT1D receptor (Ki: 5 nM).

Donitriptan hydrochloride (Donitriptan monohydrochloride) 是一种有效的高亲和力 5-HT1B 1D 受体激动剂，pKi 分别为 9.4 和 9.3。

Sumatriptan succinate (GR 43175) 是一种5-HT1受体激动剂，可作用于偏头疼的急性治疗。

Eletriptan hydrobromide (Eletriptan HBr) 是一种口服活性激动剂，对 5-HT1B 1D 受体具有特异性亲和力，Ki 值分别为 0.92 和 3.14 nM。

Zolmitriptan (311C90) 是一种5-HT1B 1D 受体部分激动剂，可用于偏头痛的研究，对 5-HT1B、5-HT1D、5-HT1F 受体的Ki 分别为 5.01、0.63 和 63.09 nM。

Alniditan is a receptors agonist of 5-HT1B 1D in HEK 293 cells (IC50: 1.7 and 1.3 nM). For 5-HT1B 1D receptors, the pKi values are 8.96 and 9.40, respectively.

Frovatriptan Succinate is a synthetic triptan with 5-HT1B 1D receptors agonist activity. It is indicated for the acute treatment of migraine.

5-HT1B 1D receptor antagonist

Dual 5-HT1B 1D receptor antagonist

Donitriptan Mesylate, a 5-HT1B 1D agonist, is used potentially for the treatment of migraines.

GR-127935 is a potent and selective 5-HT1B 1D receptor antagonist.