(rac)pyrotinib

(Rac)-Pyrotinib ((Rac)-SHR-1258) is the racemate of Pyrotinib. Pyrotinib is a potent and selective EGFR/HER2 dual inhibitor.

Pyrotinib dimaleate 是选择性的 EGFR/HER2双重抑制剂，IC50值分别为 13 和 38 nM，用于治疗HER2阳性乳腺癌。