trv 120056

TRV120056 is a Gq-biased agonist that demonstrates a molecular efficacy ten times greater at the AT1R-Gq fusion protein than at the AT1R-βarr2 fusion protein.

TRV120056 acetate 是一种 Gq 偏向激动剂，对 AT1R-Gq 融合蛋白的分子效率比 AT1R-βarr2 融合蛋白高 10 倍。