trpa1in1

TRPA1-IN-1 is a potent, selective antagonist of the TRPA1 channel, demonstrating significant oral bioavailability as a small molecule.

hTRPA1-IN-1 (19) 是从海绵Diacarnus spinipoculum中提取的一种倍半萜化合物，作为瞬时受体电位阳离子通道苜蓿素1 (TRPA1) 的抑制剂，其IC50为2 μM。