trpa1 antagonist 1

TRPA1 Antagonist 1 is an antagonist of TRPA1(IC50: 8 nM) and is a methylene phosphate prodrug which converts to its active parent drug.

TRPA1 Antagonist 3 is a compound with photoswitchable properties that acts as an agonist on the TRPA1 channel, providing the ability for optical control.

AMG9090 is a transient receptor potential ankyrin 1 (TRPA1) antagonist.

TRPA1-IN-1 is a potent, selective antagonist of the TRPA1 channel, demonstrating significant oral bioavailability as a small molecule.

PF-04745637 是TRPA1的选择性拮抗剂，对人 TRPA1 的IC50为 17 nM。