tamoxifen-d5

Tamoxifen-d5 is a deuterium labeled Tamoxifen. Tamoxifen is a selective modulator of estrogen receptor (SERM). Tamoxifen is a potent activator of Hsp90 and enhances the Hsp90 molecular chaperone ATPase activity.

(E)-4-Hydroxytamoxifen-d5 ((E)-Afimoxifene-d5) 是 (E)-4-Hydroxytamoxifen 的氘取代形式。(E)-4-Hydroxytamoxifen ((E)-Afimoxifene) 是 (Z)-4-hydroxytamoxifen 的低活性异构体，并作为雌激素受体 (estrogen receptor) 的调节剂。