Elacestrant S enantiomer (RAD1901 S enantiomer) is a low activity enantiomer of elacestrant. Elacestrant, also known as RAD1901, is an orally available and selective estrogen receptor ( ERR ) degrader. It exhibits IC50 values of 48 nM and 870 nM for ERα and ERβ, respectively.
Elacestrant S enantiomer is a selective and orally available estrogen receptor (ERR) degrader with IC50 values of 48 and 870 nM for ERα and ERβ, respectively.
Elacestrant (RAD1901) dihydrochloride is a selective and orally available estrogen receptor (ERR) degrader with IC50 values of 48 and 870 nM for ERα and ERβ, respectively. Elacestrant S enantiomer dihydrochloride is an low activity enantiomer of elacestrant dihydrochloride.