isometheptene

Dexisometheptene is an antimigraine drug candidate. Dexisometheptene significantly increases the pain threshold of acute pain response, and potently and selectively binds to receptors in the central nervous system known as imidazoline type-1 (I1) receptor

Isometheptene mucate 是一种拟交感神经剂，是间接作用的肾上腺素能受体 (adrenergic receptor) 激动剂，能够用于研究偏头痛。