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gs9876 monosuccinate

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  • Lanraplenib monosuccinate
    GS-9876 monosuccinate
    T11824L1800046-97-2
    Lanraplenib monosuccinate inhibits SYK activity in platelets via the glycoprotein VI (GPVI) receptor without prolonging bleeding time (BT) in monkeys or humans. Lanraplenib monosuccinate is a highly selective and orally active SYK inhibitor (IC50=9.5 nM) in development for the treatment of inflammatory diseases.
    • ¥ 10600
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