ezetimibe

Ezetimibe (SCH 58235) 是一种膳食胆固醇吸收抑制剂。它是一种NPC1L1抑制剂，是有效的Nrf2激活剂。

Ezetimibe-d4-1是Ezetimibe的氘代物，Ezetimibe是一种有效的胆固醇吸收抑制剂和NPC1L1抑制剂，并具有Nrf2激活作用。

Ezetimibe Ring-Open Impurity-d4 是 Ezetimibe Ring-Open Impurity 的氘代化合物。Ezetimibe Ring-Open Impurity 的 CAS 号为 1197811-72-5。

Desfluoro-ezetimibe is the defluorinated impurity of ezetimibe. Ezetimibe is an effective, metabolically stable cholesterol absorption inhibitor. Ezetimibe is a Niemann-Pick C1-like1 (NPC1L1) inhibitor and an effective Nrf2 activator.

ent-Ezetimibe (ent-SCH 58235) 是 Ezetimibe 的 RRS 型对映体。其中Ezetimibe 是一种胆固醇吸收 (cholesterol-absorption) 抑制剂，是NPC1L1抑制剂，也是有效的Nrf2激活剂。

Ezetimibe D4, a deuterium-labeled variant of Ezetimibe, functions as an inhibitor of Niemann-Pick C1-like1 (NPC1L1) and is recognized for its potent activation of Nrf2.

Ezetimibe ketone (EZM-K) 是一种 Ezetimibe 代谢产物，具有抗氧化活性，可缓解 H2O2 诱导 NRK-52E 细胞凋亡和活性氧 （ROS），上调 Nrf2 和 HO-1 水平。

Ezetimibe phenoxy glucuronide (Ezetimibe glucuronide) is the active metabolite of Ezetimibe. Antihyperlipoproteinemic activity.

Ezetimibe phenoxy glucuronide-d4 (Ezetimibe glucuronide-d4) 是 2H 标记的 Ezetimibe phenoxy glucuronide。Ezetimibe phenoxy glucuronide 是 Ezetimibe 的活性代谢物，具有降脂活性，抑制肠道对胆固醇的吸收。phenoxy glucuronide。Ezetimibe phenoxy glucuronide 通过减少肠道对胆固醇的吸收来降低 LDL-C。

Sch 58053 is an analog of Ezetimibe and a selective inhibitor of lymphatic cholesterol transport in the intestine.