drak2-in-1

Drak2-in-1, a potent, selective and ATP-competitive DRAK2 inhibitor, has an IC50 and KIvalue of 3 nM and 0.26 nM, respectively.Drak2-in-1 also had an effect on DRAK1 (IC50=51 nM).

DRAK1 2-IN-1 是一种活性的DRAK1和DRAK2双重抑制剂，Kd 值分别为 1 μM 和 6 μM。