azd-9496 maleate

AZD9496 maleate is a highly potent and selective antagonist of the estrogen receptor alpha (ERα), exhibiting an IC50 value of 0.28 nM. This compound, AZD9496 maleate, is an orally bioavailable selective estrogen receptor degrader (SERD).

AZD9496 是口服有效的选择性雌激素受体降解剂，是一种选择性的雌激素受体拮抗剂(IC50:0.28 nM)。