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核受体化合物库

核受体化合物库

产品编号 L1510 Nuclear Receptor Compound Library
  库化合物信息   Excel SDF

核受体是细胞内一类区别于膜受体的蛋白,它们与相应配体结合后,能够直接与基因组DNA 结合并调节相邻基因表达,因此这类受体被归类为转录因子。核受体在胚胎发育和机体内环境平衡中发挥关键作用。近年来,核受体家族在代谢性疾病领域受到广泛的关注,已有研究证明,它们与糖尿病、脂肪肝等疾病的发生发展密切相关,也被称为代谢性核受体。

TargetMol 汇集了546 种有文献报道的核受体相关化合物,适用于核受体相关信号通路及疾病研究,可用于高通量筛选和高内涵筛选。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
咨询化合物库
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产品描述

  • 546个核受体作用化合物的独特集合,可用于高通量筛选和高内涵筛选;
  • 提供产品的来源、化学信息和生物学信息,为筛选提供理论方向和研究基础;
  • 结构多样,药效显著,可渗透细胞;
  • NMR和HPLC技术保证产品高纯度。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L1510)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

PPAR (124)
Estrogen/progestogen Receptor (94)
Estrogen Receptor/ERR (86)
Autophagy (69)
Androgen Receptor (64)
Glucocorticoid Receptor (62)
Endogenous Metabolite (53)
Retinoid Receptor (40)
Apoptosis (31)
ROR (22)
Progesterone Receptor (21)
Thyroid hormone receptor(THR) (21)
FXR (21)
AhR (21)
Antibacterial (16)
Liver X Receptor (15)
COX (15)
Aryl Hydrocarbon Receptor (11)
P450 (10)
NF-κB (9)
Reactive Oxygen Species (8)
Ferroptosis (8)
Antifungal (6)
GPR (6)
Potassium Channel (5)
RAR/RXR  (5)
Akt (5)
AMPK (5)
Drug Metabolite (5)
Antibiotic (4)
TSH Receptor (4)
Prostaglandin Receptor (4)
Annexin A (4)
Influenza Virus (4)
Parasite (4)
Mitophagy (4)
MMP (4)
Adrenergic Receptor (4)
JNK (3)
Lipoxygenase (3)
GPCR19 (3)
Reductase (3)
IL Receptor (3)
TRP/TRPV Channel (3)
Tyrosinase (3)
GABA Receptor (2)
AChR (2)
Virus Protease (2)
Nrf2 (2)
p53 (2)
NO Synthase (2)
Cannabinoid Receptor (2)
PARP (2)
Smo (2)
PDE (2)
Phosphatase (2)
DNA/RNA Synthesis (2)
Sirtuin (2)
Interleukin (2)
HIV Protease (2)
transporter (2)
VEGFR (2)
Aromatase (2)
p38 MAPK (2)
Glutathione Peroxidase (2)
BCL (2)
ROS (2)
SARS-CoV (2)
PKC (2)
TNF (2)
S1P Receptor (1)
Sodium Channel (1)
PKA (1)
STAT (1)
Phospholipase (1)
TAM Receptor (1)
PAK (1)
Thrombin (1)
Proteasome (1)
Phosphorylase (1)
ABC (1)
Opioid Receptor (1)
c-Met/HGFR (1)
Epoxide Hydrolase (1)
Epigenetic Reader Domain (1)
EGFR (1)
DNA Methyltransferase (1)
Dehydrogenase (1)
Cysteine Protease (1)
Complement System (1)
c-Kit (1)
FLAP (1)
Caspase (1)
Carbonic Anhydrase (1)
CaMK (1)
Calcium Channel (1)
Antioxidant (1)
Antifection (1)
Adenylyl cyclase (1)
ERK (1)
FLT (1)
NOS (1)
Histone Methyltransferase (1)
MRP (1)
Melatonin Receptor (1)
MAO (1)
Ligands for Target Protein for PROTAC (1)
Ligand for E3 Ligase (1)
Leukotriene Receptor (1)
LDL (1)
HIF/HIF Prolyl-Hydroxylase (1)
Gamma-secretase (1)
HER (1)
HCV Protease (1)
HBV (1)
GSK-3 (1)
GluR (1)
Glucosidase (1)
Glucokinase (1)
Wnt/beta-catenin (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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