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表观遗传库

表观遗传库

现 货
产品编号 L1200 Epigenetics Compound Library
  库化合物信息   Excel SDF

表观遗传学主要研究“表观遗传现象”的机制,包括:基因选择性转录的调控,有DNA 甲基化、基因印记、组蛋白共价修饰和染色质重塑;和基因转录后的调控,有基因组中非编码RNA、微小RNA、反义RNA、内含子及核糖开关等。表征遗传具有解释老化机制、人类发育和癌症起源等疾病的潜力。例如,文献报道原癌基因区的表征遗传控制和肿瘤抑制序列可通过组蛋白构象变化而直接影响癌症的形成和进展。

TargetMol 表观遗传库收集960 种表观遗传相关的活性小分子,适用于表观遗传学研究,可用于高通量、高内涵筛选。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
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产品描述

  • 数量:精选960种表观遗传相关活性的化合物,且含有多种结构新颖的小分子,用于表观遗传学研究及其相关的检测和高通量、高内涵筛选;
  • 靶点含HDAC、SIRT、HAT以及HMT等十多种表观遗传相关靶点;
  • 信息详尽:化合物结构、靶点信息、活性描述等,为活性实验开展提供参考;
  • NMR、LCMS/HPLC检测技术保证产品高纯度和高质量。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L1200)
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客户使用化合物库发表的文献

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化合物库组成

Apoptosis (156)
Epigenetic Reader Domain (144)
Histone Methyltransferase (117)
HDAC (111)
Autophagy (100)
JAK (98)
PKC (78)
AMPK (77)
PARP (75)
Sirtuin (58)
Aurora Kinase (53)
HIF/HIF Prolyl-Hydroxylase (49)
HIF (36)
Histone Demethylase (36)
Histone Acetyltransferase (29)
Tyrosine Kinases (27)
CDK (27)
Endogenous Metabolite (25)
FLT (24)
Antibacterial (23)
DNA Methyltransferase (23)
Pim (21)
STAT (20)
HIV Protease (18)
Influenza Virus (16)
PKA (16)
Akt (16)
VEGFR (15)
Mitophagy (15)
Src (15)
Antibiotic (14)
Parasite (13)
Caspase (13)
EGFR (13)
ERK (12)
Wnt/beta-catenin (12)
FGFR (10)
NF-κB (10)
COX (10)
PDGFR (10)
BCL (10)
Reactive Oxygen Species (10)
PPAR (9)
Bcr-Abl (9)
Virus Protease (9)
p38 MAPK (9)
Topoisomerase (8)
c-RET (8)
ROCK (8)
Syk (8)
P450 (7)
PAD (7)
DNA/RNA Synthesis (7)
TNF (7)
MEK (7)
Casein Kinase (7)
PI3K (7)
GSK-3 (7)
IL Receptor (6)
PLK (6)
JNK (6)
Nrf2 (6)
Antifungal (6)
Adenosine Receptor (5)
AChR (5)
PDE (5)
Ferroptosis (5)
Methionine Adenosyltransferase (MAT) (5)
Calcium Channel (5)
Dehydrogenase (5)
S6 Kinase (5)
CaMK (5)
Serine/threonin kinase (5)
HSV (4)
NO Synthase (4)
MAO (4)
IκB/IKK (4)
Chk (4)
p53 (4)
Monoamine Oxidase (3)
IGF-1R (3)
c-Fms (3)
MAPK (3)
HER (3)
MMP (3)
mTOR (3)
GABA Receptor (3)
HBV (3)
DYRK (3)
IFNAR (3)
Trk receptor (3)
RAAS (3)
Histamine Receptor (3)
Nucleoside Antimetabolite/Analog (3)
Potassium Channel (3)
BTK (3)
SGK (3)
Ligand for E3 Ligase (2)
cholecystokinin (2)
MLK (2)
Hippo pathway (2)
ATP Citrate Lyase (2)
TLR (2)
PROTACs (2)
Phosphatase (2)
Sodium Channel (2)
AChE (2)
TGF-beta/Smad (2)
Serine Protease (2)
Antiviral (2)
YAP (2)
Anti-infection (2)
Dopamine Receptor (2)
Carboxypeptidase (2)
DNA Alkylation (2)
Tyrosinase (2)
Ligands for Target Protein for PROTAC (2)
transporter (2)
LDL (2)
Gamma-secretase (2)
5-HT Receptor (2)
Fatty Acid Synthase (2)
Integrin (2)
Microtubule Associated (2)
Myosin (2)
HCV Protease (2)
DUB (2)
Indoleamine 2,3-Dioxygenase (IDO) (2)
c-Kit (2)
Proteasome (1)
ribosome (1)
Phospholipase (1)
Cannabinoid Receptor (1)
DAPK (1)
NADPH-oxidase (1)
NOD (1)
BMI-1 (1)
TAM Receptor (1)
CFTR (1)
PD-1/PD-L1 (1)
Reverse Transcriptase (1)
PTEN (1)
Beta Amyloid (1)
NADPH (1)
SIK (1)
IAP (1)
Adrenergic Receptor (1)
Glucokinase (1)
Antifolate (1)
Estrogen Receptor/ERR (1)
c-Myc (1)
Tie-2 (1)
PERK (1)
BACE (1)
UGT (1)
Antioxidant (1)
c-Met/HGFR (1)
Estrogen/progestogen Receptor (1)
DNA-PK (1)
NPC1L1 (1)
Transferase (1)
Carbonic Anhydrase (1)
NOS (1)
Proton pump (1)
Chloride channel (1)
E1/E2/E3 Enzyme (1)
GRK (1)
GST (1)
Lipoxygenase (1)
Free radical scavengers (1)
LRRK2 (1)
SARS-CoV (1)
HSP (1)
P-gp (1)
Beta-Secretase (1)
SGLT (1)
Telomerase (1)
Interleukin (1)
Androgen Receptor (1)
GluR (1)
Raf (1)
Mdm2 (1)
CCR (1)
Hedgehog/Smoothened (1)
Guanylate cyclase (1)
ROS (1)
Antifection (1)
Mitochondrial Metabolism (1)
DNA gyrase (1)
NMDAR (1)
P2X Receptor (1)
S1P Receptor (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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