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Perfluorinated SAHA is an HDAC inhibitor for use in cancer treatment regimens, with demonstrated greater antiproliferative properties than SAHA . PFSAHA has also been shown to have higher selectivity for PA3774, an HDAC-like enzyme from P. aeruginosa, as well as other HDACs, which may prove beneficial for developing novel chemotherapeutic treatments for cancer.

KSI-3716 是一种 c-Myc 抑制剂，是一种膀胱内化疗剂，阻断 c-MYC MAX 与靶基因启动子形成复合物，通过诱导细胞周期停滞和细胞凋亡发挥作用，可用于膀胱癌的研究。

KSI-6666作为一种口服有效的竞争性鞘氨醇1-磷酸受体1 (S1PR1) 拮抗剂，其IC50值仅为6.4 nM。在自身免疫性脑脊髓炎模型及T细胞转移性结肠炎模型中，KSI-6666展示了显著的抗炎效果。

PKSI-527 is an inhibitor of plasma kallikrein (Ki = 0.81 μM). It is selective for plasma kallikrein over glandular kallikrein, plasmin, thrombin, urokinase, and Factor Xa (Kis = >500, 390, >500, 200, and >500 μM, respectively). PKSI-527 reduces bradykinin generation induced by kaolin and λ-carrageenan ex vivo in human plasma. It also prolongs partial thromboplastin and euglobulin clot lysis times. In vivo, PKSI-527 (300 mg/kg per day) reduces hyperplasia, pannus formation, and infiltration of inflammatory cells in the tarsal joint of mice with collagen-induced arthritis.

AVSEHQLLHDKGKSIQDLRRRFFLHHLI-{Aib}-EIHTAYRFGG 促进骨化作用。该化合物适用于研究成骨缺陷或骨矿物质密度（BMD）降低相关疾病，如骨质疏松症。

Pinobanksin是一种天然黄酮类化合物，在B细胞淋巴瘤细胞系和SH-SY5Y细胞中诱导凋亡。是一种强效抗氧化剂，能够抑制低密度脂蛋白（LDL）的过氧化，能够占据黄嘌呤氧化酶（XO）的催化中心从而进行抑制。Pinobanksin还表现出抗菌、抗炎、抗寄生虫、抗突变、抗增殖和抗血管生成的作用。

10-Hydroxydihydroperaksine是一种天然产物，属于夹竹桃科萝芙木属，其产品编号为 TN2568，CAS号为 451478-47-0。10-Hydroxydihydroperaksine可用作对照参考。

3,7-O-Diacetylpinobanksin是一种天然产物，属于松科松属，其产品编号为 TN2910，CAS号为 103553-98-6。3,7-O-Diacetylpinobanksin可用作对照参考。

Pinobanksin 3-acetate (3-O-Acetylpinobanksin) 是一种短叶松素酯衍生物,是一种强抗氧化剂，存在于向日葵和蜂蜜中，可以抑制低密度脂蛋白的过氧化.

Dihydroperaksine是一种天然产物，属于夹竹桃科萝芙木属，其产品编号为 TN3860，CAS号为 16100-84-8。Dihydroperaksine可用作对照参考。

Pinobanksin 3-O-propanoate is a natiral product from forest trees.

Pinobanksin 5-methyl ether can induce detoxification genes.

Pinobanksin 3-(2-methyl)butyrate 是 Pinobanksin 衍生物。pinobanksin 是一种细胞凋亡诱导剂，可诱导 F6细胞凋亡。

Peraksine是一种天然产物，属于夹竹桃科萝芙木属，其产品编号为 TN6030，CAS号为 15527-80-7。Peraksine可用作对照参考。

KS I is a gonadotropin antagonist and is a cyclolignan isolated from extracts of Lycopus and Lithosperum after oxidation with caffeic acid.

PI5P4Ks-IN-2 是磷脂酰肌醇 5-磷酸 4-激酶 PI5P4Kγ 的抑制剂。PI5P4Ks-IN-2 靶向 PI5P4K 亚型，对 PI5P4Kα、PI5P4Kβ、PI5P4Kγ和PI5P4Kγ+具有抑制作用 ，IC50 值分别 <4.3、<4.6、6.2和0.32 。

DYRKs-IN-1 has antitumor activity. DYRKs-IN-1 is a potent DYRKs (Dual-specificity tyrosine-phosphorylation-regulated kinases) inhibitor with IC50s of 9 nM and 5 nM for DYRK1B and DYRK1A, respectively.

DYRKs-IN-2 has antitumor activity. DYRKs-IN-2 is a potent DYRKs inhibitor with IC50s of 30.6 nM and 12.8 nM for DYRK1B and DYRK1A, respectively.

TNKS-IN-41 highly potent and selective inhibitor of tankyrase.

Gentamicin (Centicin) 是一种广谱的氨基糖苷类抗生素，具有抗菌活性，抑制革兰氏阳性菌和革兰氏阴性细菌的生长，可用于研究眼部感染。

TNKS-IN-1 is a highly potent and selective inhibitor of tankyrase.

KS IV is a cyclolignan isolated from extract of Lycopus and Lithosperum after oxidation with caffeic acid.

PI5P4Ks-IN-1 (compound 7) 是一种与PI5P4Kγ结合的活性化合物。

LDHA PDKs-IN-2 (compound 20k) 是有效的 LDHA 和 PDKs 的双重抑制剂，IC50 值分别为 0.7 和 1.6 μM。LDHA PDKs-IN-2 会增加耗氧量并且减少乳酸的形成。LDHA PDKs-IN-2 显示了癌症研究的潜力，它可以减少 A549 细胞的增殖，EC50值为 15.7 μM。