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PSMA-1007 is a novel Glu-Ureido-type prostate-specific membrane antigen (PSMA) inhibitor.

STK899704 is a tubulin inhibitor. It prevents the polymerization of purified tubulin in vitro and depolymerizes microtubule in cultured cells leading to mitotic arrest.

MK-8998 是一种T型钙通道拮抗剂，可能用于治疗精神分裂症。然而，在治疗急性精神病住院患者方面，根据第四周的PANSS评分，MK-8998未显示出有效性。

GSK 894281 is a ghrelin receptor agonist. It may produces myocardial degeneration necrosis in rats.

GSK-894490A is an agonist of ghrelin receptor. GSK-894490A crosses the blood brain barrier and elicit pro-cognitive effects.

MK-8970 is an acetal carbonate prodrug of raltegravir with enhanced colonic absorption.

BRF110 is a brain penetrant, potent and selective agonist of nuclear receptor-related 1 (Nurr1):Retinoid X receptor α (RXRα) heterodimer. BRF110 is a neuroprotective agent that prevents dopaminergic neuron demise and striatal dopaminergic denervation in vivo against PD-causing toxins. It induced dopamine biosynthesis in vivo. BRF110 chronic dosing does not induce dyskinesia in mice model.

U-78517F is a potent inhibitor of lipid peroxidation.

K-8986 is a novel h1-receptor antagonist

Racemic rasagiline，也称为 AGN-1135，是一种单胺氧化酶 B 型抑制剂(MAOI)。然而，在食用富含酪胺的食物的患者中，这种药物的应用可能导致致命的高血压危象。TVP-1022是雷沙吉兰的(S)异构体，具有心脏保护剂的作用。