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Search Results for " noradrenaline "

46

抑制剂 & 化合物

10

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T0871	Noradrenaline bitartrate	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Noradrenaline bitartrate 直接作用于 α 和 β 肾上腺素能受体。它是去甲肾上腺素的酒石酸氢盐，去甲肾上腺素是一种合成苯乙胺，可模拟内源性去甲肾上腺素的拟交感神经作用。临床上，去甲肾上腺素用作外周血管收缩剂，通过其α-肾上腺素能作用导致动脉和静脉床收缩。它还被用作通过其 β-1 肾上腺素能作用介导的强效正性肌力和变时性心脏刺激剂。
T23070	Nisoxetine hydrochloride	Sodium Channel; Monoamine Transporter; Norepinephrine	Membrane transporter/Ion channel; Neuroscience
	Nisoxetine hydrochloride 是一种去甲肾上腺素转运蛋白 (NET) 抑制剂，Kd 值为 0.76 nM。它是抗抑郁药和局部麻药，可以阻断电压门控性钠通道。
T19654	Guanoclor 胍氯酚,VATENSOL	Others	Others
	Guanoclor (VATENSOL) 也称为guanochlor，是一种交感神经药物。已知它与猪肾膜中的非肾上腺素能位点结合。
T0166	Pancuronium dibromide Pancuronium bromide,Pavulon,泮库溴铵	AChR	Neuroscience
	Pancuronium dibromide (Pavulon) 是一种双季基类固醇，是一种神经肌肉松弛剂。它通过与乙酰胆碱竞争 nACh 受体上的结合位点来抑制神经肌肉传递。它还可抑制心脏毒蕈碱受体并具有拟交感神经作用。
T37015	Iprindole	5-HT Receptor	GPCR/G Protein; Neuroscience
	Iprindole, a tricyclic indole antidepressant, is a dual weak inhibitor of noradrenaline and 5-HT uptake [1].
T5327	Amezinium methylsulfate Amezinium metilsulfate,甲磺美嗪,Amezinium (methylsulfate),Lu-1631	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Amezinium methylsulfate (Lu-1631) 具有多种机制，包括刺激 α 和 β-1 受体以及抑制去甲肾上腺素和酪胺的摄取。
T16816	S 18986	GluR	Neuroscience
	S 18986 is a selective, orally active, brain penetrant positive allosteric modulator of AMPA-type receptors, showcasing cognitive-enhancing properties in rodents. It induces the release of noradrenaline and acetylcholine in the rat hippocampus, leading to enhanced object-recognition memory.
T0472	Venlafaxine hydrochloride Venlafaxine HCl,盐酸文拉法辛,Wy 45030 hydrochloride	5-HT Receptor; Serotonin Transporter	GPCR/G Protein; Neuroscience
	Venlafaxine hydrochloride (Wy 45030 hydrochloride) 是一种口服有效的 5-羟色胺 (5-HT)/去甲肾上腺素 (NE) 重摄取的双重抑制剂，具有抗抑郁活性。
T1471	Duloxetine hydrochloride Duloxetine HCl,盐酸度洛西汀,LY-248686 hydrochloride,(S)-Duloxetine hydrochloride,LY-248686 HCl	Dopamine Receptor; 5-HT Receptor; Serotonin Transporter; Norepinephrine	GPCR/G Protein; Neuroscience
	Duloxetine hydrochloride ((S)-Duloxetine hydrochloride) 是一种 5-羟色胺-去甲肾上腺素重吸收 (serotonin-norepinephrine reuptake) 抑制剂 (SNRI)，Ki=4.6 nM，可用于广泛性焦虑症的研究。
TP2106L	Urantide acetate(669089-53-6 free base)	Neurotensin Receptor	GPCR/G Protein
	Urantide acetate(669089-53-6 free base) 是一种选择性和竞争性的 urotensin-II (UT) 受体拮抗剂 (pKB = 8.3)。体外阻断 hU-II 诱导的胸主动脉收缩。对去甲肾上腺素或内皮素 1 诱导的收缩或乙酰胆碱诱导的松弛没有影响。在钙动员测定（在表达 hUT 受体的 CHO 细胞中）中表现为部分激动剂。
T69331	Ciclazindol (free base)
	Ciclazindol (free base) is a noradrenaline uptake inhibitor.
T36949	Niaprazine	5-HT Receptor; Adrenergic Receptor; Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Niaprazine 是有效的组胺 H1 受体拮抗剂，具有抗组胺和抗血清素活性。Niaprazine 在睡眠障碍方面有研究的价值。
T69389	Desethylreboxetine
	Desethylreboxetine is an desethylated metabolite of Reboxetine (R142000), a selective noradrenaline reuptake inhibitor and an antidepressant.
T28951	Tesofensine NS 2330,NS2330,NS-2330
	Tesofensine, a serotonin–noradrenaline–dopamine reuptake inhibitor, is used potentially for the treatment of obesity.
T69509	SCH-12650 maleate
	SCH-12650 maleate is a noradrenaline uptake and gastric secretion inhibitor.
T69335	Ciclazindol hydrochloride
	Ciclazindol hydrochloride is the salt from of Ciclazindol (free base), a noradrenaline uptake inhibitor.
T26970	CD-349 CD 349,CD349
	CD-349 is a calcium channel antagonist. CD-349 inhibits the noradrenaline (NA)-induced contraction of aortas in Ca2(+)-free medium.
T69568	FLA-63
	FLA-63 is a dopamine-beta-hydroxylase (DBH)-inhibitor and an inhibitor of the last step of noradrenaline biosynthesis.
T33006	LY-104119 LY 104119,LY104119
	LY-104119 is a thermogenic weight loss compound that rapidly reduces noradrenaline concentrations in brown adipose tissue between the scapulas, the heart, and the liver.
T7341	Diclofensine Ro 8-4650,(+/-)-双氮奋兴	Dopamine Receptor; Monoamine Transporter	GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
	Diclofensine (Ro 8-4650) 是一种高效单胺再摄取抑制剂，在大鼠脑突触体中能够阻断多巴胺 (IC50=0.74 nM)、去甲肾上腺素 (IC50=2.3 nM) 和 5-羟色胺 (IC50=3.7 nM)。
T69270	Amezinium
	Amezinium is a sympathomimetic drug used for the treatment of low blood pressure. It has multiple mechanisms, including stimulation of alpha and beta-1 receptors and inhibition of noradrenaline and tyramine uptake.
TP2106	Urantide
	Selective and competitive urotensin-II (UT) receptor antagonist (pKB = 8.3). Blocks hU-II induced contractions in thoracic aorta ex vivo. Exhibits no effect on noradrenaline or endothelin 1-induced contraction or on acetylcholine-induced relaxation. Behav
T10145	4-Hydroxyatomoxetine	Others	Others
	4-Hydroxyatomoxetine is an active metabolite of Atomoxetine. 4-Hydroxyatomoxetine is metabolized by CYP2D6. Atomoxetine is a noradrenaline reuptake inhibitor.
T68327	Dexnafenodone Free Base
	Dexnafenodone Free Base is a potent inhibitor of noradrenaline, and to a lesser degree of serotonin reuptake, induced changes in the pattern of sleep which are comparable to those of non‐sedating tricyclic antidepressants.
T69071	Secoverine
	Secoverine is a selective muscarinic receptor antagonist that was studied as a neurotropic spasmolytic agent. It was shown that the drug had no nicotinolytic or antihistaminic activity, a moderate antisterotonic activity, an inhibiting effect on the noradrenaline uptake mechanism of the vas deferens and marked local anesthetic activity.
T60368	Benzoctamine
	Benzoctamine 是一种口服有效作用精神剂，具有镇静作用。Benzoctamine 增加儿茶酚胺的周转率。Benzoctamine 增强大鼠心脏中 [3H] 去甲肾上腺素的摄取。Benzoctamine 也可加速脑内注射 [3H] 去甲肾上腺素的消失。
T11892	Lurasidone D8 Hydrochloride SM-13496 D8	Others	Others
	Lurasidone D8 Hydrochloride is an inhibitor of Dopamine D2, 5-HT2A, 5-HT7, 5-HT1A and noradrenaline α2C, and is the deuterium labeled Lurasidone.
T37699	Org 24598
	Potent and selective inhibitor of the glial glycine transporter GlyT1b (IC50 = 6.9 nM). Displays negligible activity at GlyT-2, adrenoreceptors, dopamine, 5HT receptors and noradrenaline, dopamine, 5HT and GABA transporters (pIC50 in vivo. Chue et al (2013) Glycine reuptake inhibition as a new therapeutic approach in schizophrenia: focus on the glycine transporter 1 (GlyT1). Curr.Pharm.Des. 19 1311 PMID:23194655 \|Brown et al (2001) Discovery and SAR of org 24598-a selective glycine uptake inhibi...
T10144	4-Hydroxyatomoxetine D3	Others	Others
	4-Hydroxyatomoxetine D3 is a deuterium labeled 4-Hydroxyatomoxetine. 4-Hydroxyatomoxetine is an active metabolite of Atomoxetine. 4-Hydroxyatomoxetine is metabolized by CYP2D6. Atomoxetine is a noradrenaline reuptake inhibitor.
T29002	Trazium Esilate EGYT3615,EGYT-3615,EGYT 3615
	Trazium esilate is an adrenergic receptor antagonist. Trazium esilate is a weak displacer on a1-, a2- and D2-receptors, however, it induced a2-receptor desenzitization after repeated treatment. It had no influence on rat brain cortical noradrenaline and s
T69133	Etozolin HCl
	Etozolin HCl is a safe and effective diuretic agent in the treatment of acute cardiac failure. In isolated rings of guinea-pig aorta not responding to acetylcholine, the diuretic dexetozoline did not influence basal vascular tone but inhibited noradrenaline- and histamine-induced contractions. Dexetozoline has a very high bioavailability after oral administration and is fairly lipohilic. The half-life of etozolin is 2.5 h. Dexetozoline accumulates in cirrhosis.
T73083	Nipradolol KT 210 ; K 351 ; Hypadil,Hypadil,KT 210,K 351
	Nipradolol (KT-210; K-351) 是一种有效的 α-1-肾上腺素能受体的阻滞剂。Nipradolol 还抑制白化兔模型中 Phenylephrine 诱导的眼压升高 (IOP)。Nipradolol 抑制去甲肾上腺素 (NA) 引起的肌肉收缩，对犬冠状动脉也有血管扩张剂活性。
T31582	DSP 4 DSP4,UNII-PQ1P7JP5C1,DSP-4,az-Dsp 4
	DSP 4 is a selective neurotoxin selective for noradrenergic neurons in the locus coeruleus noradrenergic system and capable of crossing the blood–brain barrier and cyclizes to a reactive aziridinium derivative that is accumulated into the noradrenergic ne
T69145	Nisoxetine 尼索西汀
	Nisoxetine 是一种有效的和选择性的去甲肾上腺素转运蛋白(NET)抑制剂，Kd 值为 0.76 nM。Nisoxetine 是一种抗抑郁试剂和局部麻药，它可以阻断电压门控性钠通道。
T71772	Bicifadine free base
	Bicifadine, also known as DOV-220075, CL 220,075, is a SNDR inhibitor potentially for the treatment of lower back pain. Bicifadine has a non-opioid, non-NSAID mechanism for the treatment of pain, which should have less abuse potential than opioid drugs and less propensity to cause gastric ulcers than NSAID drugs. While the drug is purported to be a serotonin (SERT) and noradrenaline transporter (NET) inhibitor, it also has effects at the dopamine transporter (DAT), effectively making it a broad...
T74045	H-Lys-Tyr-OH TFA
	H-Lys-Tyr-OH TFA (Lysyltyrosine TFA)为L-赖氨酸与L-酪氨酸构成的二肽。该化合物通过促进去甲肾上腺素与酪氨酸在大脑中的释放，用于预防神经系统疾病或提升大脑功能。
T1580	Desvenlafaxine 去甲文拉法辛,WY 45233 Succinate,O-Desmethylvenlafaxine	5-HT Receptor; Serotonin Transporter; Norepinephrine	GPCR/G Protein; Neuroscience
	Desvenlafaxine (O-Desmethylvenlafaxine) 是 Venlafaxine 主要代谢物的丁二酸盐形式，在人多巴胺转运体上显示弱的结合亲和力。它是一种具有口服活性的、能透过血脑屏障的5-HT 和去甲肾上腺素再摄取的抑制剂，对 hSERT 和 hNET 的IC50值分别为 47.3 nM 和 531.3 nM。
T72209	(R,R)-Reboxetine mesylate (R,R)-FCE20124 mesylate ; (R,R)-PNU155950E mesylate,(R,R)-PNU155950E mesylate,(R,R)-FCE20124 mesylate
	(R,R)-Reboxetine mesylate 是一种抗抑郁药，具有良好的生物利用度。(R,R)-Reboxetine 为 Reboxetine 的对映体之一，属于选择性去甲肾上腺素再摄取抑制剂。Reboxetine 本身包含 (R,R) 与 (S,S) 两种对映体，且对 α-肾上腺素能和毒蕈碱受体的亲和力较低，表现出较低的动物毒性。
T1735	Lurasidone hydrochloride Lurasidone HCl,SM-13496 (Hydrochloride),盐酸鲁拉西酮,SM-13496	Dopamine Receptor; 5-HT Receptor; Norepinephrine	GPCR/G Protein; Neuroscience
	Lurasidone hydrochloride (Lurasidone HCl) 是多巴胺 D2和5-HT7的拮抗剂，IC50值分别为 1.68 和 0.495 nM，用于治疗精神分裂症和双相情感障碍。它也是5-HT1A 受体的部分激动剂，IC50值为 6.75 nM。
T74582	Trimipramine N-oxide
	Trimipramine N-oxide 为三环抗抑郁药trimipramine的活性代谢物，其对人去甲肾上腺素单胺转运体(hNAT)、血清素(hSERT)、多巴胺(hDAT)以及人体有机阳离子转运蛋白(hOCT1与hOCT2)的IC50值分别为11.7、3.59、9.4、9.35及27.4 nM。因此，Trimipramine N-oxide在忧郁和焦虑研究中有应用价值。
T71356	Lanperisone HCl
	Lanperisone, also known as NK433, is a muscle relaxant. NK433 inhibited the facilitation of the flexor reflex mediated by group II afferent fibers that was induced by intrathecal administration of noradrenaline-HCl. NK433 had effects more than three times stronger and tending to be longer-lasting than those of eperisone-HCl. These results suggest that NK433 exerts a non-selective inhibition on spinal reflexes and that inhibition of the descending noradrenergic tonic facilitation within the spina...
T72701	Cavα2δ1&NET-IN-3
	Cavα2δ1&NET-IN-3 (example 216) 是电压门控钙通道 (VGCC) 的亚基 α2δ 和去甲肾上腺素转运蛋白 (NET) 抑制剂。Cavα2δ1&NET-IN-3 对人的 Cav2.2 钙通道 α2δ-1 亚基和 NET 的 Ki 均为 100-500 nM。
T68190	Carmoxirole (free base)
	Carmoxirole (free base) is a dopamine D2 receptor agonist with limited central activity that modulates sympathetic activation and subsequently reduces pre-load and afterload in animals. It was shown, that carmoxirole induced beneficial effects on hemodynamic and neurohumoral parameters in heart failure. In addition, experimental evidence showed that carmoxirole lowered blood pressure in various models of hypertension mainly or exclusively through inhibition of noradrenaline release from sympathe...
T28653	S-8510 free base SB 737552,SB-737552,S8510,SB737552,S-8510,S 8510
	S-8510 is a GABA-A receptor inverse agonist. S-8510 selectively potentiated pentylenetetrazol-induced convulsion without affecting minimal electroconvulsive shock- or strychnine-induced convulsion in ddY mice. S-8510 ameliorated memory impairment induced
T78126	Dothiepin Dosulepin,Dothep	Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Dothiepin（Dosulepin; Dothep）是一种具备镇静/抗焦虑作用的抗抑郁药物。该化合物主要通过抑制去甲肾上腺素的再摄取，而非血清素，以增强去肾上腺素能神经传递。同时，Dothiepin作为组胺H1受体的拮抗剂，具备显著的镇痛活性，适用于治疗心因性面部疼痛、特发性纤维肌痛综合征或类风湿关节炎，并且不具有心脏毒性。
T2306	Brexpiprazole 依匹哌唑,OPC-34712,依匹唑派	Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Brexpiprazole (OPC-34712) 是人5-HT1A 和多巴胺受体的部分激动剂，Ki 分别为0.12 和 0.3 nM。它也是5-HT2A 受体的拮抗剂，Ki 为 0.47 nM，可作为非典型抗精神病药。

化合物

Noradrenaline bitartrate

Cat.No: T0871

Target: Adrenergic Receptor

Nisoxetine hydrochloride

Cat.No: T23070

Target: Sodium Channel, Monoamine Transporter, Norepinephrine

Cat.No: T19654

Synonym: 胍氯酚,VATENSOL

Target: Others

Pancuronium dibromide

Cat.No: T0166

Synonym: Pancuronium bromide,Pavulon,泮库溴铵

Target: AChR

Cat.No: T37015

Target: 5-HT Receptor

Amezinium methylsulfate

Cat.No: T5327

Synonym: Amezinium metilsulfate,甲磺美嗪,Amezinium (methylsulfate),Lu-1631

Target: Adrenergic Receptor

Cat.No: T16816

Target: GluR

Venlafaxine hydrochloride

Cat.No: T0472

Synonym: Venlafaxine HCl,盐酸文拉法辛,Wy 45030 hydrochloride

Target: 5-HT Receptor, Serotonin Transporter

Duloxetine hydrochloride

Cat.No: T1471

Synonym: Duloxetine HCl,盐酸度洛西汀,LY-248686 hydrochloride,(S)-Duloxetine hydrochloride,LY-248686 HCl

Target: Dopamine Receptor, 5-HT Receptor, Serotonin Transporter, Norepinephrine

Urantide acetate(669089-53-6 free base)

Cat.No: TP2106L

Target: Neurotensin Receptor

Ciclazindol (free base)

Cat.No: T69331

Cat.No: T36949

Target: 5-HT Receptor, Adrenergic Receptor, Histamine Receptor

Desethylreboxetine

Cat.No: T69389

Cat.No: T28951

Synonym: NS 2330,NS2330,NS-2330

SCH-12650 maleate

Cat.No: T69509

Ciclazindol hydrochloride

Cat.No: T69335

Cat.No: T26970

Synonym: CD 349,CD349

Cat.No: T69568

Cat.No: T33006

Synonym: LY 104119,LY104119

Cat.No: T7341

Synonym: Ro 8-4650,(+/-)-双氮奋兴

Target: Dopamine Receptor, Monoamine Transporter

Cat.No: T69270

Cat.No: TP2106

4-Hydroxyatomoxetine

Cat.No: T10145

Target: Others

Dexnafenodone Free Base

Cat.No: T68327

Cat.No: T69071

Cat.No: T60368

Lurasidone D8 Hydrochloride

Cat.No: T11892

Synonym: SM-13496 D8

Target: Others

Cat.No: T37699

4-Hydroxyatomoxetine D3

Cat.No: T10144

Target: Others

Trazium Esilate

Cat.No: T29002

Synonym: EGYT3615,EGYT-3615,EGYT 3615

Cat.No: T69133

Cat.No: T73083

Synonym: KT 210 ; K 351 ; Hypadil,Hypadil,KT 210,K 351

Cat.No: T31582

Synonym: DSP4,UNII-PQ1P7JP5C1,DSP-4,az-Dsp 4

Cat.No: T69145

Synonym: 尼索西汀

Bicifadine free base

Cat.No: T71772

H-Lys-Tyr-OH TFA

Cat.No: T74045

Cat.No: T1580

Synonym: 去甲文拉法辛,WY 45233 Succinate,O-Desmethylvenlafaxine

Target: 5-HT Receptor, Serotonin Transporter, Norepinephrine

(R,R)-Reboxetine mesylate

Cat.No: T72209

Synonym: (R,R)-FCE20124 mesylate ; (R,R)-PNU155950E mesylate,(R,R)-PNU155950E mesylate,(R,R)-FCE20124 mesylate

Lurasidone hydrochloride

Cat.No: T1735

Synonym: Lurasidone HCl,SM-13496 (Hydrochloride),盐酸鲁拉西酮,SM-13496

Target: Dopamine Receptor, 5-HT Receptor, Norepinephrine

Trimipramine N-oxide

Cat.No: T74582

Lanperisone HCl

Cat.No: T71356

Cavα2δ1&NET-IN-3

Cat.No: T72701

Carmoxirole (free base)

Cat.No: T68190

S-8510 free base

Cat.No: T28653

Synonym: SB 737552,SB-737552,S8510,SB737552,S-8510,S 8510

Cat.No: T78126

Synonym: Dosulepin,Dothep

Target: Histamine Receptor

Cat.No: T2306

Synonym: 依匹哌唑,OPC-34712,依匹唑派

Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor

Cat. No.	Product Name	Target	Signaling Pathways
T20173	Noradrenaline tartrate NSC 169106,NSC-169106,l-Noradrenaline d-bitartrate,NSC169106,Norepinephrine bitartrate
	Norepinephrine bitartrate is a precursor of epinephrine. Norepinephrine is the principal transmitter of most postganglionic sympathetic fibers and of the diffuse projection system in the brain arising from the locus ceruleus.
T1064	Norepinephrine bitartrate monohydrate 酒石酸去甲肾上腺素,Levophed,Noradrenaline bitartrate monohydrate,降肾上腺素	Endogenous Metabolite; Adrenergic Receptor; Autophagy	Autophagy; GPCR/G Protein; Metabolism; Neuroscience
	Norepinephrine bitartrate monohydrate (Levophed) 是一种β1-选择性的肾上腺素能受体激动剂，EC50为 5.37 μM。
T7044	Norepinephrine 去甲肾上腺素,Levophed,Levonoradrenaline,Aktamin,Nor-Epirenan,Levonor,Arterenol	MMP; Endogenous Metabolite; Adrenergic Receptor; Autophagy	Autophagy; GPCR/G Protein; Metabolism; Neuroscience; Proteases/Proteasome
	Norepinephrine (Levophed) 是β1选择性的肾上腺素能受体激动剂，EC50值为 5.37 μM。它可上调鼻咽癌肿瘤细胞中血管内皮生长因子、基质金属蛋白酶MMP-2和MMP-9的表达。
T1045	Trimipramine maleate Surmontil maleate,马来酸三甲丙咪嗪,三甲丙咪嗪马来酸盐	Dopamine Receptor; 5-HT Receptor; Antibacterial; Adrenergic Receptor; Norepinephrine; Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience
	Trimipramine maleate (Surmontil maleate) 是一种 5-HT 受体拮抗剂，对 5-HT1C、5-HT2和 5-HT1A 受体的 pKi 值分别为 6.39、8.10和 4.66。
T0689	D-Phenylalanine	Endogenous Metabolite; Monocarboxylate transporter	Membrane transporter/Ion channel; Metabolism
	D-Phenylalanine 是一种苯丙氨酸的合成右旋异构体，可抑制Pseudoalteromonas sp.SC2014 的生物膜发育。
T0469	Octopamine hydrochloride 章鱼胺盐酸盐,(±)-p-Octopamine hydrochlorid,(+,-)-Octopamine HCl,章胺盐酸盐	Dopamine Receptor; Endogenous Metabolite; Adrenergic Receptor	GPCR/G Protein; Metabolism; Neuroscience
	Octopamine hydrochloride ((±)-p-Octopamine hydrochlorid) 是一种与去甲肾上腺素结构相关的生物单胺类物质，在无脊椎动物中起着神经调节剂、神经激素和神经递质的作用。它对转染人 alpha2-肾上腺素受体(ARs)的中国仓鼠卵巢细胞 α2-ARs 有刺激作用。它提高糖原分解、糖酵解、糖异生、摄氧量和门脉灌注压。
T4848	Mandelic acid acidomandelico,DL-Mandelic acid,扁桃酸	Others; Endogenous Metabolite; Antibacterial	Metabolism; Microbiology/Virology; Others
	DL-Mandelic acid (acidomandelico) 是一种 α-羟基羧酸，有抗菌活性，广泛用作医药和精细化学品的中间体，已用于研究尿路感染和阴道滴虫病，还具有较高的精子固定活性和较低的阴道刺激性。
T2S0118	Daurinoline	Calcium Channel; 5-HT Receptor; Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience
	Daurinoline is a non-competitive antagonist, it exerts marked relaxation effect on basilar artery of rabbits through non-competitive antagonism, it would have a protective function on microcirculation of cerebral pia mater, which may be beneficial to relieve cerebral ischemic injury. Daurinoline could significantly reverse noradrenaline induced constriction of pial arterioles and venules, and increase the number of blood vessels which were decreased by noradrenaline.
TN3368	Akuammigine	Opioid Receptor; Adrenergic Receptor	Endocrinology/Hormones; GPCR/G Protein; Neuroscience
	Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding pA2 values of 4.68. Akuammidine also shows a preference for mu-opioid binding sites with Ki val
T37911	cis-Resveratrol 顺式白藜芦醇,(Z)-Resveratrol
	Resveratrol is a potent phenolic antioxidant found in grapes, red wine, and various berries that also has antiproliferative and anti-inflammatory activity. cis-Resveratrol is the double bond isomer of trans-resveratrol, the more often studied and naturally abundant of the two resveratrol isomers. cis-Resveratrol exhibits antioxidant activity in the &#181M range similar to that observed with trans-resveratrol. It blocks production of reactive oxygen species (ROS) by inhibition of NAD(P)H oxidase ...

天然产物

Noradrenaline tartrate

Cat.No: T20173

Synonym: NSC 169106,NSC-169106,l-Noradrenaline d-bitartrate,NSC169106,Norepinephrine bitartrate

Norepinephrine bitartrate monohydrate

Cat.No: T1064

Synonym: 酒石酸去甲肾上腺素,Levophed,Noradrenaline bitartrate monohydrate,降肾上腺素

Target: Endogenous Metabolite, Adrenergic Receptor, Autophagy

Cat.No: T7044

Synonym: 去甲肾上腺素,Levophed,Levonoradrenaline,Aktamin,Nor-Epirenan,Levonor,Arterenol

Target: MMP, Endogenous Metabolite, Adrenergic Receptor, Autophagy

Trimipramine maleate

Cat.No: T1045

Synonym: Surmontil maleate,马来酸三甲丙咪嗪,三甲丙咪嗪马来酸盐

Target: Dopamine Receptor, 5-HT Receptor, Antibacterial, Adrenergic Receptor, Norepinephrine, Histamine Receptor

D-Phenylalanine

Cat.No: T0689

Target: Endogenous Metabolite, Monocarboxylate transporter

Octopamine hydrochloride

Cat.No: T0469

Synonym: 章鱼胺盐酸盐,(±)-p-Octopamine hydrochlorid,(+,-)-Octopamine HCl,章胺盐酸盐

Target: Dopamine Receptor, Endogenous Metabolite, Adrenergic Receptor

Cat.No: T4848

Synonym: acidomandelico,DL-Mandelic acid,扁桃酸

Target: Others, Endogenous Metabolite, Antibacterial

Cat.No: T2S0118

Target: Calcium Channel, 5-HT Receptor, Histamine Receptor

Cat.No: TN3368

Target: Opioid Receptor, Adrenergic Receptor

cis-Resveratrol

Cat.No: T37911

Synonym: 顺式白藜芦醇,(Z)-Resveratrol

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