delequamine

Delequamine HCl is a potent and selective alpha 2-adrenoceptor antagonist. Delequamine HCl has a pKi of 9.45 for alpha 2-adrenoceptors in the rat cortex (pA2 in the guinea-pig ileum of 9.72).

Delequamine (RS 15385-197) 是一种有效的选择性 α2-肾上腺素受体拮抗剂。

RS 15385-198 是 Delequamine 的低活性异构体。Delequamine 是一种选择性 α2-肾上腺素受体拮抗剂。