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NTRC-824 is >150-fold selectivity for NTS2 over NTS1 (Ki >30 μM). NTRC-824 is an effective, selective, and neurotensin-like nonpeptide neurotensin receptor type 2 (NTS2) antagonist (IC50: 38 nM and a Ki : 202 nM).
NTRC-824 is >150-fold selectivity for NTS2 over NTS1 (Ki >30 μM). NTRC-824 is an effective, selective, and neurotensin-like nonpeptide neurotensin receptor type 2 (NTS2) antagonist (IC50: 38 nM and a Ki : 202 nM).
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
50 mg | 待估 | 35日内发货 |
产品描述 | NTRC-824 is >150-fold selectivity for NTS2 over NTS1 (Ki >30 μM). NTRC-824 is an effective, selective, and neurotensin-like nonpeptide neurotensin receptor type 2 (NTS2) antagonist (IC50: 38 nM and a Ki : 202 nM). |
靶点活性 | NTS2:38 nM, NTS2:(ki)202 nM |
体外活性 | NTRC-824 is the first nonpeptide compound that behaves like and is more active than, the endogenous ligand. In the NTS1 assay up to 30 μM, Testing of NTRC-824 at the NTS1 receptor displays no binding activity, making NTRC-824 selective for NTS2 in both the binding and functional assays . |
分子量 | 553.55 |
分子式 | C25H26F3N3O6S |
CAS No. | 1623002-61-8 |
密度 | 1.41 g/cm3 (Predicted) |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
以上为“体内实验配液计算器”的使用方法举例,并不是具体某个化合物的推荐配制方式,请根据您的实验动物和给药方式选择适当的溶解方案。
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