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TargetMol产品目录中 "

endothelium dependent relaxation

"的结果
  • 抑制剂&激动剂
    7
    TargetMol | Inhibitors_Agonists
  • 多肽产品
    2
    TargetMol | Peptide_Products
  • 天然产物
    1
    TargetMol | Natural_Products
  • L-Nabe
    N(w)-nitroarginine benzyl ester, H-Arg(NO2)-Obzl, N-Nitro-L-argininebenzyl ester, NABE, Benzyl Nw-nitro-L-argininate
    T257487672-27-7
    L-Nabe (H-Arg(NO2)-Obzl) 是一种有效的不可逆内皮依赖性舒张抑制剂。
    • ¥ 10600
    6-8周
    规格
    数量
  • CGP48369
    T14942135689-23-5In house
    CGP48369 是一种有效的血管紧张素 II 受体 (angiotensin II receptor) 拮抗剂,具有降血压作用,可增强自发性高血压大鼠冠状动脉的内皮依赖性松弛。
    • ¥ 4900
    In stock
    规格
    数量
  • ZM 169369
    ICI169369,ICI-169369
    T2757485273-95-6
    ICI 169369, a 5-HT2 5-HT1C antagonist, can evoke endothelium-dependent relaxation in rabbit aorta.
    • ¥ 10600
    6-8周
    规格
    数量
  • Nolpitantium Free Base
    T70456155418-05-6
    Nolpitantium Free Base is a highly selective nonpeptide antagonist of neurokinin-1 (NK1) receptor. Nolpitantium potently, selectively and competitively inhibited substance P binding to NK1 receptors from various animal species, including humans. In vitro, it was a potent antagonist in functional assays for NK1 receptors such as [Sar9, Met(O2)11]substance P-induced endothelium-dependent relaxation of rabbit pulmonary artery and contraction of guinea-pig ileum. Up to 1 mkM, Nolpitantium had no effect in bioassays for NK2 and NK3 receptors. The antagonism exerted by Nolpitantium toward NK1 receptors was apparently non-competitive, with pD2' values between 9.65 and 10.16 in the different assays. Nolpitantium also blocked in vitro [Sar9, Met(O2)11]substance P-induced release of acetylcholine from rat striatum. In vivo, Nolpitantium exerted highly potent antagonism toward [Sar9, Met(O2)11]substance P-induced hypotension in dogs, bronchoconstriction in guinea-pig) and plasma extrava......
    • ¥ 21600
    10-14周
    规格
    数量
  • Quercetin-3-O-(2′′-O-galloyl)-β-D-glucopyranoside
    T8132469624-79-9
    Quercetin-3-O-(2′′-O-galloyl)-β-D-glucopyranoside 是一种从天竺葵属植物中分离的酚类化合物,具有口服活性和抗炎特性,可能在治疗水肿和改善主动脉内皮依赖性舒张损伤方面有应用潜力。
    • 待询
    规格
    数量
  • Adrenomedullin (porcine)
    T83164912862-96-5
    Adrenomedullin(porcine)是一種多肽,具有调节血管舒张的功能。它在内皮依赖性条件下能诱导大鼠主动脉舒张,IC50为2.4 nM;在内皮非依赖性条件下则能诱导猪冠状动脉舒张,IC50为27.6 nM。
    • 待询
    规格
    数量
  • IRL-1038 TFA
    IRL-1038 TFA(144602-02-8 Free base)
    TP2262L1
    IRL-1038 TFA 是一种具有选择性和高效性的内皮素 B(ETB)受体拮抗剂, 抑制内皮素诱导的内皮依赖性松弛,可用于研究心血管疾病。
    • ¥ 130
    In stock
    规格
    数量