- 全部删除
- 您的购物车当前为空
Amisulpride (DAN 2163) 是多巴胺D2/D3受体拮抗剂,对于人多巴胺D2和D3的Ki 分别为 2.8 和 3.2 nM。
Amisulpride (DAN 2163) 是多巴胺D2/D3受体拮抗剂,对于人多巴胺D2和D3的Ki 分别为 2.8 和 3.2 nM。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
2 mg | ¥ 116 | In stock | |
5 mg | ¥ 169 | In stock | |
10 mg | ¥ 236 | In stock | |
25 mg | ¥ 375 | In stock | |
50 mg | ¥ 543 | In stock | |
100 mg | ¥ 795 | In stock | |
500 mg | ¥ 1,990 | In stock | |
1 mL x 10 mM (in DMSO) | ¥ 239 | In stock |
产品描述 | Amisulpride (DAN 2163) (trade name Solian) is an antipsychotic drug sold by Sanofi-Aventis. It is not approved for use in the United States, but is approved for use in Europe and Australia for the treatment of psychoses and schizophrenia. Additionally, it is approved in Italy for the treatment of dysthymia (under the brand name Deniban). Amisulpride is a selective dopamine antagonist. |
靶点活性 | D3 receptor:3.2 nM (Ki), D2 receptor:2.8 nM (Ki) |
别名 | 氨磺必利, 阿米舒必利, DAN 2163 |
分子量 | 369.48 |
分子式 | C17H27N3O4S |
CAS No. | 71675-85-9 |
Smiles | C(NCC1N(CC)CCC1)(=O)C2=C(OC)C=C(N)C(S(CC)(=O)=O)=C2 |
密度 | 1.2 g/cm3 |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
溶解度信息 | Ethanol: 65 mg/mL (175.92 mM), Sonication is recommended. H2O: < 1 mg/mL (insoluble or slightly soluble) DMSO: 50 mg/mL (135.33 mM), Sonication is recommended. ![]() | |||||||||||||||||||||||||||||||||||
溶液配制表 | ||||||||||||||||||||||||||||||||||||
DMSO/Ethanol
|
以上为“体内实验配液计算器”的使用方法举例,并不是具体某个化合物的推荐配制方式,请根据您的实验动物和给药方式选择适当的溶解方案。
评论内容