erkin3

ERK-IN-3 (ASN007 free base) 是一种有效的口服活性 ERK 抑制剂，以低 IC50 值抑制 ERK1 2，可用于研究由 RAS 突变驱动的癌症。

ERK-IN-3 benzenesulfonate is a potent and orally active inhibitor of ERK . ERK-IN-3 benzenesulfonate inhibits ERK1 2 with low single-digit nM IC 50 values. ERK-IN-3 benzenesulfonate can be used for the research of cancers driven by RAS mutations.

PERK-IN-3 is a potent inhibitor of PERK(IC50 of 7.4 nM).